BG37380A3 - Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid - Google Patents

Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid

Info

Publication number
BG37380A3
BG37380A3 BG055782A BG5578282A BG37380A3 BG 37380 A3 BG37380 A3 BG 37380A3 BG 055782 A BG055782 A BG 055782A BG 5578282 A BG5578282 A BG 5578282A BG 37380 A3 BG37380 A3 BG 37380A3
Authority
BG
Bulgaria
Prior art keywords
phenylacetamido
dioxo
halo
ester
preparing
Prior art date
Application number
BG055782A
Other languages
Bulgarian (bg)
English (en)
Inventor
Vytautas Jasys
Original Assignee
Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware filed Critical Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Publication of BG37380A3 publication Critical patent/BG37380A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Cephalosporin Compounds (AREA)
BG055782A 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid BG37380A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24645681A 1981-03-23 1981-03-23

Publications (1)

Publication Number Publication Date
BG37380A3 true BG37380A3 (en) 1985-05-15

Family

ID=22930766

Family Applications (2)

Application Number Title Priority Date Filing Date
BG055782A BG37380A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid
BG067396A BG38939A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG067396A BG38939A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid

Country Status (32)

Country Link
EP (1) EP0061274B1 (da)
JP (3) JPS57169493A (da)
KR (1) KR860001368B1 (da)
AU (1) AU531892B2 (da)
BG (2) BG37380A3 (da)
CA (1) CA1213581A (da)
CS (1) CS227345B2 (da)
DD (1) DD202163A5 (da)
DE (1) DE3267505D1 (da)
DK (3) DK162392C (da)
EG (1) EG15803A (da)
ES (2) ES510655A0 (da)
FI (1) FI74284C (da)
GB (1) GB2095250A (da)
GR (1) GR75935B (da)
GT (1) GT198274393A (da)
HK (1) HK52487A (da)
HU (2) HU187667B (da)
IE (1) IE52835B1 (da)
IL (1) IL65308A (da)
IN (1) IN159362B (da)
MY (1) MY8700499A (da)
NO (1) NO159658C (da)
NZ (1) NZ200066A (da)
PH (1) PH17602A (da)
PL (3) PL138851B1 (da)
PT (1) PT74621B (da)
RO (2) RO87946A (da)
SG (1) SG23387G (da)
SU (2) SU1277897A3 (da)
YU (2) YU42761B (da)
ZA (1) ZA821899B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0084730A1 (en) * 1982-01-22 1983-08-03 Beecham Group Plc Esters of penicillin derivatives with beta-lactamase inhibitors, their preparation and their use
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
GB8808701D0 (en) * 1988-04-13 1988-05-18 Erba Carlo Spa Beta-lactam derivatives
ES2039299B1 (es) * 1991-10-04 1994-05-16 Asturpharma S A Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) * 1995-06-02 1998-04-01 Asturpharma S A Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
CN112724162B (zh) * 2020-12-28 2022-06-10 华南农业大学 一种阿莫西林-舒巴坦杂合分子的合成方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) * 1979-03-05 1981-02-25 Pfizer Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof
IE50650B1 (en) * 1979-10-11 1986-06-11 Leo Pharm Prod Ltd Method for producing penicillanic acid derivatives

Also Published As

Publication number Publication date
SU1277897A3 (ru) 1986-12-15
SU1277898A3 (ru) 1986-12-15
GT198274393A (es) 1983-09-08
DK165746B (da) 1993-01-11
AU8176482A (en) 1982-11-04
DK162392C (da) 1992-03-09
IL65308A0 (en) 1982-05-31
CA1213581A (en) 1986-11-04
KR830009113A (ko) 1983-12-17
DK165746C (da) 1993-06-07
IE52835B1 (en) 1988-03-16
EP0061274B1 (en) 1985-11-21
DD202163A5 (de) 1983-08-31
JPS6345287A (ja) 1988-02-26
PT74621A (en) 1982-04-01
PL235578A1 (en) 1983-06-20
FI820991L (fi) 1982-09-24
NO159658B (no) 1988-10-17
RO87946A (ro) 1985-12-20
JPS63146886A (ja) 1988-06-18
FI74284B (fi) 1987-09-30
SG23387G (en) 1987-07-10
YU61982A (en) 1985-03-20
PL240664A1 (en) 1983-09-12
BG38939A3 (en) 1986-03-14
PL139261B1 (en) 1987-01-31
EP0061274A1 (en) 1982-09-29
DE3267505D1 (en) 1986-01-02
DK127182A (da) 1982-09-24
DK121491D0 (da) 1991-06-21
GB2095250A (en) 1982-09-29
HU189917B (en) 1986-08-28
DK162392B (da) 1991-10-21
PL240663A1 (en) 1983-09-12
PH17602A (en) 1984-10-05
JPS57169493A (en) 1982-10-19
YU43585B (en) 1989-08-31
NO159658C (no) 1989-01-25
ES8403132A1 (es) 1984-03-01
YU42761B (en) 1988-12-31
HUT34985A (en) 1985-05-28
FI74284C (fi) 1988-01-11
ES8305768A1 (es) 1983-04-16
YU181084A (en) 1987-06-30
IL65308A (en) 1985-03-31
RO84278B (ro) 1984-07-30
MY8700499A (en) 1987-12-31
EG15803A (en) 1990-08-30
ZA821899B (en) 1983-01-26
PL138851B1 (en) 1986-11-29
NZ200066A (en) 1985-08-16
DK21892D0 (da) 1992-02-20
RO87946B (ro) 1985-12-02
IE820659L (en) 1982-09-23
DK21892A (da) 1992-02-20
PT74621B (en) 1984-11-26
HU187667B (en) 1986-02-28
NO820898L (no) 1982-09-24
HK52487A (en) 1987-07-17
KR860001368B1 (ko) 1986-09-17
PL134250B1 (en) 1985-08-31
JPH0331717B2 (da) 1991-05-08
DK121491A (da) 1991-06-21
DK167119B1 (da) 1993-08-30
RO84278A (ro) 1984-05-23
ES518970A0 (es) 1984-03-01
CS227345B2 (en) 1984-04-16
IN159362B (da) 1987-05-09
AU531892B2 (en) 1983-09-08
ES510655A0 (es) 1983-04-16
GR75935B (da) 1984-08-02

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