BG26526A3 - Метод за получаване на 1-(бензазолилалкил)пиперидинови производни - Google Patents

Метод за получаване на 1-(бензазолилалкил)пиперидинови производни

Info

Publication number
BG26526A3
BG26526A3 BG033791A BG3379176A BG26526A3 BG 26526 A3 BG26526 A3 BG 26526A3 BG 033791 A BG033791 A BG 033791A BG 3379176 A BG3379176 A BG 3379176A BG 26526 A3 BG26526 A3 BG 26526A3
Authority
BG
Bulgaria
Prior art keywords
benzazolylalkyl
preparation
piperidine derivatives
piperidine
derivatives
Prior art date
Application number
BG033791A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jan Vandenberk
Ludo Edmond Kennis
Marcel Van
Albert M.
Original Assignee
Неизвестен
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/687,139 external-priority patent/US4066772A/en
Application filed by Неизвестен filed Critical Неизвестен
Publication of BG26526A3 publication Critical patent/BG26526A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG033791A 1975-07-21 1976-07-20 Метод за получаване на 1-(бензазолилалкил)пиперидинови производни BG26526A3 (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US59779375A 1975-07-21 1975-07-21
US05/687,139 US4066772A (en) 1975-07-21 1976-05-17 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds
KR7601697A KR810000334B1 (ko) 1975-07-21 1976-07-12 1-(벤즈 아조릴알킬) 피페리딘 유도체의 제조방법

Publications (1)

Publication Number Publication Date
BG26526A3 true BG26526A3 (bg) 1979-04-12

Family

ID=27348142

Family Applications (1)

Application Number Title Priority Date Filing Date
BG033791A BG26526A3 (bg) 1975-07-21 1976-07-20 Метод за получаване на 1-(бензазолилалкил)пиперидинови производни

Country Status (25)

Country Link
JP (1) JPS5217475A (tr)
AT (1) AT364358B (tr)
AU (1) AU511027B2 (tr)
BG (1) BG26526A3 (tr)
CA (1) CA1085852A (tr)
CH (1) CH623820A5 (tr)
CS (1) CS202550B2 (tr)
DE (1) DE2632870A1 (tr)
DK (1) DK154950C (tr)
ES (3) ES449740A1 (tr)
FI (1) FI62667C (tr)
GB (1) GB1542514A (tr)
HK (1) HK14180A (tr)
IE (1) IE43496B1 (tr)
IT (1) IT1062614B (tr)
KE (1) KE3215A (tr)
LU (1) LU75354A1 (tr)
MY (1) MY8100017A (tr)
NL (1) NL187442C (tr)
NZ (1) NZ181256A (tr)
PH (1) PH13710A (tr)
PT (1) PT65387B (tr)
RO (1) RO70566A (tr)
SE (2) SE426490B (tr)
YU (1) YU39969B (tr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4501749A (en) * 1983-10-31 1985-02-26 Merck & Co., Inc. Peripherally selective dopamine antagonists in the treatment of ocular hypertension
JPS6248684A (ja) * 1985-08-26 1987-03-03 Sumitomo Chem Co Ltd 新規なヨ−ドブチロフエノン誘導体およびその製造法
JPS62251313A (ja) * 1986-04-25 1987-11-02 信越ポリマー株式会社 結束装置
US6355659B1 (en) 1994-07-29 2002-03-12 Laboratorios Del Dr. Esteve, S.A. 4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same
FR2723091B1 (fr) * 1994-07-29 1996-11-08 Esteve Labor Dr Tetrahydropyridine-(6,4-hydroxypiperidine) alkylazoles
PA8603801A1 (es) * 2003-05-27 2004-12-16 Janssen Pharmaceutica Nv Derivados de la quinazolina
CA2549869C (en) 2003-12-18 2015-05-05 Janssen Pharmaceutica N.V. Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
NI200700147A (es) 2004-12-08 2019-05-10 Janssen Pharmaceutica Nv Derivados de quinazolina inhibidores de cinasas dirigidos a multip
AU2007274284B2 (en) 2006-07-13 2012-04-26 Janssen Pharmaceutica N.V. Mtki quinazoline derivatives
EP1997805A1 (en) * 2007-06-01 2008-12-03 Commissariat à l'Energie Atomique Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans
ES2562218T3 (es) 2007-07-27 2016-03-03 Janssen Pharmaceutica, N.V. Pirrolopirimidinas útiles para el tratamiento de enfermedades proliferativas
RU2488585C2 (ru) 2007-08-31 2013-07-27 Пэдью Фарма Л.П. Замещенные пиперидиновые соединения хиноксалинового типа и их применение
WO2014102594A2 (en) 2012-12-27 2014-07-03 Purdue Pharma L.P. Substituted benzimidazole-type piperidine compounds and uses thereof
CN113995755A (zh) * 2016-02-04 2022-02-01 辛多美制药有限公司 氘代多潘立酮组合物和用于治疗病症的方法
KR20240125702A (ko) 2017-06-30 2024-08-19 신돔 파마, 인크. 중수소화 돔페리돈 조성물, 방법, 및 제조

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE633495A (tr) * 1962-06-13
BE633914A (tr) * 1962-06-22
US3629267A (en) * 1968-10-28 1971-12-21 Smith Kline French Lab Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione
AU4698672A (en) * 1972-09-22 1972-11-09 Ciba-Geigy Ag Azacycloaliphatic compounds, process for their manufacture and compositions containing them
FR2218100A1 (en) * 1973-02-20 1974-09-13 Janssen Pharmaceutica Nv Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones
US3989707A (en) * 1974-06-21 1976-11-02 Janssen Pharmaceutica N.V. Benzimidazolinone derivatives

Also Published As

Publication number Publication date
FI762086A (tr) 1977-01-22
ES449740A1 (es) 1978-02-16
AT364358B (de) 1981-10-12
HK14180A (en) 1980-03-28
ES461631A1 (es) 1978-12-01
PT65387A (en) 1976-08-01
FI62667B (fi) 1982-10-29
IT1062614B (it) 1984-10-20
JPS5217475A (en) 1977-02-09
GB1542514A (en) 1979-03-21
CS202550B2 (en) 1981-01-30
YU179476A (en) 1983-01-21
JPS6131109B2 (tr) 1986-07-17
DK327576A (da) 1977-01-22
DE2632870A1 (de) 1977-02-10
RO70566A (ro) 1982-10-11
AU511027B2 (en) 1980-07-24
CH623820A5 (en) 1981-06-30
CA1085852A (en) 1980-09-16
DK154950C (da) 1989-05-29
IE43496B1 (en) 1981-03-11
FI62667C (fi) 1983-02-10
DK154950B (da) 1989-01-09
SE435621B (sv) 1984-10-08
IE43496L (en) 1977-01-21
ATA534776A (de) 1981-03-15
SE7608265L (sv) 1977-01-22
ES461630A1 (es) 1978-06-16
DE2632870C2 (tr) 1989-02-16
SE426490B (sv) 1983-01-24
MY8100017A (en) 1981-12-31
PT65387B (en) 1978-06-09
YU39969B (en) 1985-06-30
LU75354A1 (tr) 1977-02-28
NZ181256A (en) 1978-04-28
NL187442C (nl) 1991-10-01
SE8008713L (sv) 1980-12-11
NL187442B (nl) 1991-05-01
AU1596476A (en) 1978-01-19
NL7608023A (nl) 1977-01-25
KE3215A (en) 1982-07-09
PH13710A (en) 1980-09-09

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