JPS5217475A - New 11*benzoazolii*alkyl* piperidine derivatives - Google Patents
New 11*benzoazolii*alkyl* piperidine derivativesInfo
- Publication number
- JPS5217475A JPS5217475A JP51085216A JP8521676A JPS5217475A JP S5217475 A JPS5217475 A JP S5217475A JP 51085216 A JP51085216 A JP 51085216A JP 8521676 A JP8521676 A JP 8521676A JP S5217475 A JPS5217475 A JP S5217475A
- Authority
- JP
- Japan
- Prior art keywords
- benzoazolii
- alkyl
- new
- piperidine derivatives
- piperidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Otolaryngology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US59779375A | 1975-07-21 | 1975-07-21 | |
| US05/687,139 US4066772A (en) | 1975-07-21 | 1976-05-17 | 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds |
| KR7601697A KR810000334B1 (en) | 1975-07-21 | 1976-07-12 | Process for preparation 1-(benzazolylalkyl)-piperidine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5217475A true JPS5217475A (en) | 1977-02-09 |
| JPS6131109B2 JPS6131109B2 (en) | 1986-07-17 |
Family
ID=27348142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP51085216A Granted JPS5217475A (en) | 1975-07-21 | 1976-07-19 | New 11*benzoazolii*alkyl* piperidine derivatives |
Country Status (25)
| Country | Link |
|---|---|
| JP (1) | JPS5217475A (en) |
| AT (1) | AT364358B (en) |
| AU (1) | AU511027B2 (en) |
| BG (1) | BG26526A3 (en) |
| CA (1) | CA1085852A (en) |
| CH (1) | CH623820A5 (en) |
| CS (1) | CS202550B2 (en) |
| DE (1) | DE2632870A1 (en) |
| DK (1) | DK154950C (en) |
| ES (3) | ES449740A1 (en) |
| FI (1) | FI62667C (en) |
| GB (1) | GB1542514A (en) |
| HK (1) | HK14180A (en) |
| IE (1) | IE43496B1 (en) |
| IT (1) | IT1062614B (en) |
| KE (1) | KE3215A (en) |
| LU (1) | LU75354A1 (en) |
| MY (1) | MY8100017A (en) |
| NL (1) | NL187442C (en) |
| NZ (1) | NZ181256A (en) |
| PH (1) | PH13710A (en) |
| PT (1) | PT65387B (en) |
| RO (1) | RO70566A (en) |
| SE (2) | SE426490B (en) |
| YU (1) | YU39969B (en) |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6248684A (en) * | 1985-08-26 | 1987-03-03 | Sumitomo Chem Co Ltd | Novel iodobutyrophenone derivative and production thereof |
| JPS62251313A (en) * | 1986-04-25 | 1987-11-02 | 信越ポリマー株式会社 | Bundling device |
| JP2007051154A (en) * | 1994-07-29 | 2007-03-01 | Lab Del Dr Esteve Sa | Tetrahydropyridine-(or 4-hydroxypiperidine)alkylazole having activity on sigma and/or 5ht1a receptor |
| JP2010529011A (en) * | 2007-06-01 | 2010-08-26 | コミッサリア ア レネルジ アトミック | Compounds with antiparasitic activity, their application in the treatment of infections caused by apicomplexers |
| JP2010537969A (en) * | 2007-08-31 | 2010-12-09 | パーデュー、ファーマ、リミテッド、パートナーシップ | Substituted quinoxaline-type piperidine compounds and uses thereof |
| JP2020534246A (en) * | 2016-02-04 | 2020-11-26 | シンリックス ファーマ、エルエルシー | Deuterated domperidone compositions, methods, and preparations |
| US11364226B2 (en) | 2017-06-30 | 2022-06-21 | Cinrx Pharma, Llc | Deuterated domperidone compositions, methods, and preparation |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4501749A (en) * | 1983-10-31 | 1985-02-26 | Merck & Co., Inc. | Peripherally selective dopamine antagonists in the treatment of ocular hypertension |
| US6355659B1 (en) | 1994-07-29 | 2002-03-12 | Laboratorios Del Dr. Esteve, S.A. | 4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same |
| JO2785B1 (en) * | 2003-05-27 | 2014-03-15 | شركة جانسين فارماسوتيكا ان. في | Quinazoline derivatives |
| UA83881C2 (en) | 2003-12-18 | 2008-08-26 | Янссен Фармацевтика Н.В. | Pyrido- and pyrimidopyrimidine derivatives as anti-proliferative agents |
| NI200700147A (en) | 2004-12-08 | 2019-05-10 | Janssen Pharmaceutica Nv | QUINAZOLINE DERIVATIVES KINE INHIBITORS TARGETING MULTIP |
| MX2009000456A (en) | 2006-07-13 | 2009-01-27 | Janssen Pharmaceutica Nv | Mtki quinazoline derivatives. |
| EP2185562B1 (en) | 2007-07-27 | 2015-12-02 | Janssen Pharmaceutica, N.V. | Pyrrolopyrimidines useful for the treatment of proliferative diseases |
| US9090618B2 (en) | 2012-12-27 | 2015-07-28 | Purdue Pharma L.P. | Substituted benzimidazole-type piperidine compounds and uses thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE633495A (en) * | 1962-06-13 | |||
| BE633914A (en) * | 1962-06-22 | |||
| US3629267A (en) * | 1968-10-28 | 1971-12-21 | Smith Kline French Lab | Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione |
| AU4698672A (en) * | 1972-09-22 | 1972-11-09 | Ciba-Geigy Ag | Azacycloaliphatic compounds, process for their manufacture and compositions containing them |
| FR2218100A1 (en) * | 1973-02-20 | 1974-09-13 | Janssen Pharmaceutica Nv | Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones |
| US3989707A (en) * | 1974-06-21 | 1976-11-02 | Janssen Pharmaceutica N.V. | Benzimidazolinone derivatives |
-
1976
- 1976-06-23 NZ NZ181256A patent/NZ181256A/en unknown
- 1976-06-30 GB GB7627242A patent/GB1542514A/en not_active Expired
- 1976-07-07 RO RO7686860A patent/RO70566A/en unknown
- 1976-07-07 CA CA256,450A patent/CA1085852A/en not_active Expired
- 1976-07-08 PH PH18663A patent/PH13710A/en unknown
- 1976-07-09 LU LU75354A patent/LU75354A1/xx unknown
- 1976-07-09 ES ES449740A patent/ES449740A1/en not_active Expired
- 1976-07-16 CS CS764688A patent/CS202550B2/en unknown
- 1976-07-16 AU AU15964/76A patent/AU511027B2/en not_active Expired
- 1976-07-19 JP JP51085216A patent/JPS5217475A/en active Granted
- 1976-07-19 IT IT50499/76A patent/IT1062614B/en active
- 1976-07-20 PT PT65387A patent/PT65387B/en unknown
- 1976-07-20 BG BG7633791A patent/BG26526A3/xx unknown
- 1976-07-20 IE IE1602/76A patent/IE43496B1/en not_active IP Right Cessation
- 1976-07-20 CH CH929176A patent/CH623820A5/en not_active IP Right Cessation
- 1976-07-20 FI FI762086A patent/FI62667C/en not_active IP Right Cessation
- 1976-07-20 SE SE7608265A patent/SE426490B/en not_active IP Right Cessation
- 1976-07-20 DK DK327576A patent/DK154950C/en not_active IP Right Cessation
- 1976-07-20 AT AT0534776A patent/AT364358B/en not_active IP Right Cessation
- 1976-07-20 NL NLAANVRAGE7608023,A patent/NL187442C/en not_active IP Right Cessation
- 1976-07-21 DE DE19762632870 patent/DE2632870A1/en active Granted
- 1976-07-21 YU YU1794/76A patent/YU39969B/en unknown
-
1977
- 1977-08-16 ES ES461630A patent/ES461630A1/en not_active Expired
- 1977-08-16 ES ES461631A patent/ES461631A1/en not_active Expired
-
1980
- 1980-03-20 HK HK141/80A patent/HK14180A/en unknown
- 1980-12-11 SE SE8008713A patent/SE435621B/en not_active IP Right Cessation
-
1981
- 1981-12-30 MY MY17/81A patent/MY8100017A/en unknown
-
1982
- 1982-05-21 KE KE3215A patent/KE3215A/en unknown
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6248684A (en) * | 1985-08-26 | 1987-03-03 | Sumitomo Chem Co Ltd | Novel iodobutyrophenone derivative and production thereof |
| JPS62251313A (en) * | 1986-04-25 | 1987-11-02 | 信越ポリマー株式会社 | Bundling device |
| JP2007051154A (en) * | 1994-07-29 | 2007-03-01 | Lab Del Dr Esteve Sa | Tetrahydropyridine-(or 4-hydroxypiperidine)alkylazole having activity on sigma and/or 5ht1a receptor |
| JP2010529011A (en) * | 2007-06-01 | 2010-08-26 | コミッサリア ア レネルジ アトミック | Compounds with antiparasitic activity, their application in the treatment of infections caused by apicomplexers |
| JP2010537969A (en) * | 2007-08-31 | 2010-12-09 | パーデュー、ファーマ、リミテッド、パートナーシップ | Substituted quinoxaline-type piperidine compounds and uses thereof |
| JP2020534246A (en) * | 2016-02-04 | 2020-11-26 | シンリックス ファーマ、エルエルシー | Deuterated domperidone compositions, methods, and preparations |
| US11364226B2 (en) | 2017-06-30 | 2022-06-21 | Cinrx Pharma, Llc | Deuterated domperidone compositions, methods, and preparation |
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