AU1596476A - 1-(benzazolylalkyl) piperidine derivatives - Google Patents
1-(benzazolylalkyl) piperidine derivativesInfo
- Publication number
- AU1596476A AU1596476A AU15964/76A AU1596476A AU1596476A AU 1596476 A AU1596476 A AU 1596476A AU 15964/76 A AU15964/76 A AU 15964/76A AU 1596476 A AU1596476 A AU 1596476A AU 1596476 A AU1596476 A AU 1596476A
- Authority
- AU
- Australia
- Prior art keywords
- benzazolylalkyl
- piperidine derivatives
- piperidine
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired, expires
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US59779375A | 1975-07-21 | 1975-07-21 | |
| US687139 | 1976-05-17 | ||
| US05/687,139 US4066772A (en) | 1975-07-21 | 1976-05-17 | 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds |
| KR7601697A KR810000334B1 (en) | 1975-07-21 | 1976-07-12 | Process for preparation 1-(benzazolylalkyl)-piperidine derivatives |
| US597793 | 1984-04-06 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU1596476A true AU1596476A (en) | 1978-01-19 |
| AU511027B2 AU511027B2 (en) | 1980-07-24 |
Family
ID=27348142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU15964/76A Expired AU511027B2 (en) | 1975-07-21 | 1976-07-16 | 1-(benzazolylalkyl) piperidine derivatives |
Country Status (25)
| Country | Link |
|---|---|
| JP (1) | JPS5217475A (en) |
| AT (1) | AT364358B (en) |
| AU (1) | AU511027B2 (en) |
| BG (1) | BG26526A3 (en) |
| CA (1) | CA1085852A (en) |
| CH (1) | CH623820A5 (en) |
| CS (1) | CS202550B2 (en) |
| DE (1) | DE2632870A1 (en) |
| DK (1) | DK154950C (en) |
| ES (3) | ES449740A1 (en) |
| FI (1) | FI62667C (en) |
| GB (1) | GB1542514A (en) |
| HK (1) | HK14180A (en) |
| IE (1) | IE43496B1 (en) |
| IT (1) | IT1062614B (en) |
| KE (1) | KE3215A (en) |
| LU (1) | LU75354A1 (en) |
| MY (1) | MY8100017A (en) |
| NL (1) | NL187442C (en) |
| NZ (1) | NZ181256A (en) |
| PH (1) | PH13710A (en) |
| PT (1) | PT65387B (en) |
| RO (1) | RO70566A (en) |
| SE (2) | SE426490B (en) |
| YU (1) | YU39969B (en) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4501749A (en) * | 1983-10-31 | 1985-02-26 | Merck & Co., Inc. | Peripherally selective dopamine antagonists in the treatment of ocular hypertension |
| JPS6248684A (en) * | 1985-08-26 | 1987-03-03 | Sumitomo Chem Co Ltd | Novel iodobutyrophenone derivative and production thereof |
| JPS62251313A (en) * | 1986-04-25 | 1987-11-02 | 信越ポリマー株式会社 | Bundling device |
| US6355659B1 (en) | 1994-07-29 | 2002-03-12 | Laboratorios Del Dr. Esteve, S.A. | 4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same |
| FR2723091B1 (en) * | 1994-07-29 | 1996-11-08 | Esteve Labor Dr | TETRAHYDROPYRIDINE- (6,4-HYDROXYPIPERIDINE) ALKYLAZOLES |
| JO2785B1 (en) * | 2003-05-27 | 2014-03-15 | شركة جانسين فارماسوتيكا ان. في | Quinazoline derivatives |
| JP4936897B2 (en) | 2003-12-18 | 2012-05-23 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Pyrido- and pyrimidopyrimidine derivatives as antiproliferative agents |
| NI200700147A (en) | 2004-12-08 | 2019-05-10 | Janssen Pharmaceutica Nv | QUINAZOLINE DERIVATIVES KINE INHIBITORS TARGETING MULTIP |
| JP2009542778A (en) | 2006-07-13 | 2009-12-03 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | MTKI quinazoline derivative |
| EP1997805A1 (en) * | 2007-06-01 | 2008-12-03 | Commissariat à l'Energie Atomique | Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans |
| WO2009016132A1 (en) | 2007-07-27 | 2009-02-05 | Janssen Pharmaceutica Nv | Pyrrolopyrimidines |
| KR20140139125A (en) | 2007-08-31 | 2014-12-04 | 퍼듀 퍼머 엘피 | Substituted-quinoxaline-type piperidine compounds and the uses thereof |
| US9090618B2 (en) | 2012-12-27 | 2015-07-28 | Purdue Pharma L.P. | Substituted benzimidazole-type piperidine compounds and uses thereof |
| CA3013123A1 (en) * | 2016-02-04 | 2017-08-10 | Cinrx Pharma, Llc | Deuterated domperidone compositions and methods for therapy of disorders |
| US11364226B2 (en) | 2017-06-30 | 2022-06-21 | Cinrx Pharma, Llc | Deuterated domperidone compositions, methods, and preparation |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE633495A (en) * | 1962-06-13 | |||
| BE633914A (en) * | 1962-06-22 | |||
| US3629267A (en) * | 1968-10-28 | 1971-12-21 | Smith Kline French Lab | Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione |
| AU4698672A (en) * | 1972-09-22 | 1972-11-09 | Ciba-Geigy Ag | Azacycloaliphatic compounds, process for their manufacture and compositions containing them |
| FR2218100A1 (en) * | 1973-02-20 | 1974-09-13 | Janssen Pharmaceutica Nv | Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones |
| US3989707A (en) * | 1974-06-21 | 1976-11-02 | Janssen Pharmaceutica N.V. | Benzimidazolinone derivatives |
-
1976
- 1976-06-23 NZ NZ181256A patent/NZ181256A/en unknown
- 1976-06-30 GB GB7627242A patent/GB1542514A/en not_active Expired
- 1976-07-07 CA CA256,450A patent/CA1085852A/en not_active Expired
- 1976-07-07 RO RO7686860A patent/RO70566A/en unknown
- 1976-07-08 PH PH18663A patent/PH13710A/en unknown
- 1976-07-09 ES ES449740A patent/ES449740A1/en not_active Expired
- 1976-07-09 LU LU75354A patent/LU75354A1/xx unknown
- 1976-07-16 AU AU15964/76A patent/AU511027B2/en not_active Expired
- 1976-07-16 CS CS764688A patent/CS202550B2/en unknown
- 1976-07-19 IT IT50499/76A patent/IT1062614B/en active
- 1976-07-19 JP JP51085216A patent/JPS5217475A/en active Granted
- 1976-07-20 CH CH929176A patent/CH623820A5/en not_active IP Right Cessation
- 1976-07-20 PT PT65387A patent/PT65387B/en unknown
- 1976-07-20 BG BG7633791A patent/BG26526A3/xx unknown
- 1976-07-20 IE IE1602/76A patent/IE43496B1/en not_active IP Right Cessation
- 1976-07-20 DK DK327576A patent/DK154950C/en not_active IP Right Cessation
- 1976-07-20 FI FI762086A patent/FI62667C/en not_active IP Right Cessation
- 1976-07-20 NL NLAANVRAGE7608023,A patent/NL187442C/en not_active IP Right Cessation
- 1976-07-20 SE SE7608265A patent/SE426490B/en not_active IP Right Cessation
- 1976-07-20 AT AT0534776A patent/AT364358B/en not_active IP Right Cessation
- 1976-07-21 YU YU1794/76A patent/YU39969B/en unknown
- 1976-07-21 DE DE19762632870 patent/DE2632870A1/en active Granted
-
1977
- 1977-08-16 ES ES461631A patent/ES461631A1/en not_active Expired
- 1977-08-16 ES ES461630A patent/ES461630A1/en not_active Expired
-
1980
- 1980-03-20 HK HK141/80A patent/HK14180A/en unknown
- 1980-12-11 SE SE8008713A patent/SE435621B/en not_active IP Right Cessation
-
1981
- 1981-12-30 MY MY17/81A patent/MY8100017A/en unknown
-
1982
- 1982-05-21 KE KE3215A patent/KE3215A/en unknown
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