BG108344A - ЦИТРАТНА СОЛ НА 5.8.14-ТРИАЗАТЕТРАЦИКЛО-(10.3.1.0на степен2,11 .0на степен4.9)- ХЕКСАДЕКА-2.(11),3,5,7,9-ПЕНТАЕН И НЕЙНИ ФАРМАЦЕВТИЧНИ СЪСТАВИ - Google Patents
ЦИТРАТНА СОЛ НА 5.8.14-ТРИАЗАТЕТРАЦИКЛО-(10.3.1.0на степен2,11 .0на степен4.9)- ХЕКСАДЕКА-2.(11),3,5,7,9-ПЕНТАЕН И НЕЙНИ ФАРМАЦЕВТИЧНИ СЪСТАВИ Download PDFInfo
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- BG108344A BG108344A BG108344A BG10834403A BG108344A BG 108344 A BG108344 A BG 108344A BG 108344 A BG108344 A BG 108344A BG 10834403 A BG10834403 A BG 10834403A BG 108344 A BG108344 A BG 108344A
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- triazatetracyclo
- hexadeca
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Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Veterinary Medicine (AREA)
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- Neurology (AREA)
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- Molecular Biology (AREA)
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- AIDS & HIV (AREA)
- Toxicology (AREA)
- Obesity (AREA)
- Hematology (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29086301P | 2001-05-14 | 2001-05-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG108344A true BG108344A (bg) | 2004-12-30 |
Family
ID=23117854
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG108344A BG108344A (bg) | 2001-05-14 | 2003-11-11 | ЦИТРАТНА СОЛ НА 5.8.14-ТРИАЗАТЕТРАЦИКЛО-(10.3.1.0на степен2,11 .0на степен4.9)- ХЕКСАДЕКА-2.(11),3,5,7,9-ПЕНТАЕН И НЕЙНИ ФАРМАЦЕВТИЧНИ СЪСТАВИ |
Country Status (37)
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
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| DE122008000038I1 (de) * | 1997-12-31 | 2008-11-13 | Pfizer Prod Inc | Arylkondensierte azapolycyclische derivate |
| AU2002351008B2 (en) * | 2001-11-30 | 2007-07-12 | Pfizer Products Inc. | Pharmaceutical compositions of 5,8,14-triazatetracyclo[10.3.1.0(2,11).0(4,9)]-hexadeca-2(11)3,5,7,9-pentaene |
| BRPI0410219A (pt) * | 2003-05-20 | 2006-05-09 | Pfizer Prod Inc | composições farmacêuticas de vareniclina |
| US20050043407A1 (en) * | 2003-08-22 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the prevention and treatment of addiction in a mammal |
| BRPI0718600A2 (pt) * | 2006-11-09 | 2013-12-10 | Pfizer Prod Inc | Polimorfos de intermediários nicotínicos. |
| US8440825B2 (en) | 2008-03-06 | 2013-05-14 | Medichem S.A. | Fumaric acid salt of varenicline |
| WO2009143347A2 (en) | 2008-05-22 | 2009-11-26 | Teva Pharmaceutical Industries Ltd. | Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate |
| US20090318460A1 (en) * | 2008-05-26 | 2009-12-24 | Glenmark | Amorphous varenicline tartrate and process for the preparation thereof |
| US20090318695A1 (en) * | 2008-06-19 | 2009-12-24 | Vinod Kumar Kansal | Processes for the preparation of varenicline and intermediates thereof |
| WO2010005643A1 (en) * | 2008-07-10 | 2010-01-14 | Teva Pharmaceutical Industries Ltd. | Processes for purifying varenicline l-tartrate salt and preparing crystalline forms of varenicline l-tartrate salt |
| MY160005A (en) * | 2008-12-11 | 2017-02-15 | Cti Biopharma Corp | 11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo(19.3.1.1(2,6).1(8,12))heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene citrate salt |
| US20100189791A1 (en) | 2009-01-23 | 2010-07-29 | Teva Pharmaceutical Industries, Ltd. | Delayed release rasagiline malate formulation |
| WO2010143070A2 (en) | 2009-06-10 | 2010-12-16 | Actavis Group Ptc Ehf | Amorphous varenicline tartrate co-precipitates |
| RU2012102052A (ru) | 2009-06-22 | 2013-11-20 | Тева Фармасьютикал Индастриз Лтд. | Твердые формы солей варениклина и способы их получения |
| WO2011140431A1 (en) | 2010-05-06 | 2011-11-10 | Teva Pharmaceutical Industries Ltd. | Varenicline salts and crystal forms thereof |
| PL2837632T3 (pl) | 2012-04-13 | 2017-01-31 | Lianyungang Jinkang Hexin Pharmaceutical Co. Ltd. | Pochodne triazabicyklo[3.2.1]oktanu użyteczne do leczenia chorób proliferacyjnych |
| WO2018154395A2 (en) | 2018-06-11 | 2018-08-30 | Alvogen Malta Operations (Row) Ltd | Controlled release pharmaceutical composition of varenicline |
| EP3756653A1 (en) | 2019-06-28 | 2020-12-30 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Microparticulate varenicline citrate |
| US20230105412A1 (en) * | 2020-03-16 | 2023-04-06 | Jinkun Huang | 5-ht3 receptor modulator, the crystalline form, methods of making, and use thereof |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE122008000038I1 (de) * | 1997-12-31 | 2008-11-13 | Pfizer Prod Inc | Arylkondensierte azapolycyclische derivate |
| IL137937A0 (en) * | 1999-08-27 | 2001-10-31 | Pfizer Prod Inc | A pharmaceutical composition for the prevention and treatment of nicotine addiction in a mammal |
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- 2002-04-26 AT AT02724553T patent/ATE303386T1/de not_active IP Right Cessation
- 2002-04-26 JP JP2002589481A patent/JP4137645B2/ja not_active Expired - Fee Related
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- 2002-04-26 SK SK1337-2003A patent/SK13372003A3/sk unknown
- 2002-04-26 UA UA20031110265A patent/UA73421C2/uk unknown
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- 2002-04-26 IL IL15787402A patent/IL157874A0/xx unknown
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