BE896609A - Derives de l'ergoline procede pour les preparer et leur emploi comme medicaments - Google Patents

Derives de l'ergoline procede pour les preparer et leur emploi comme medicaments

Info

Publication number
BE896609A
BE896609A BE0/210660A BE210660A BE896609A BE 896609 A BE896609 A BE 896609A BE 0/210660 A BE0/210660 A BE 0/210660A BE 210660 A BE210660 A BE 210660A BE 896609 A BE896609 A BE 896609A
Authority
BE
Belgium
Prior art keywords
medicines
preparation
ergoline derivatives
derivatives process
ergoline
Prior art date
Application number
BE0/210660A
Other languages
English (en)
Inventor
L Bernardi
A Temperilli
S Mantegani
G Traquandi
P Salvati
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of BE896609A publication Critical patent/BE896609A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
BE0/210660A 1982-04-30 1983-04-29 Derives de l'ergoline procede pour les preparer et leur emploi comme medicaments BE896609A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8212653 1982-04-30

Publications (1)

Publication Number Publication Date
BE896609A true BE896609A (fr) 1983-08-16

Family

ID=10530108

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/210660A BE896609A (fr) 1982-04-30 1983-04-29 Derives de l'ergoline procede pour les preparer et leur emploi comme medicaments

Country Status (21)

Country Link
US (1) US4657914A (fr)
JP (1) JPS58194884A (fr)
AT (1) AT385035B (fr)
AU (1) AU553851B2 (fr)
BE (1) BE896609A (fr)
CA (1) CA1210389A (fr)
CH (1) CH654305A5 (fr)
CS (1) CS236874B2 (fr)
DE (1) DE3314878A1 (fr)
DK (1) DK164058C (fr)
FI (1) FI73996C (fr)
FR (1) FR2526022B1 (fr)
GB (1) GB2120242A (fr)
GR (1) GR78842B (fr)
HU (1) HU193527B (fr)
IE (1) IE53950B1 (fr)
IL (1) IL68496A (fr)
IT (1) IT1215630B (fr)
NL (1) NL191709C (fr)
SE (1) SE460967B (fr)
ZA (1) ZA833008B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4713457A (en) * 1985-02-21 1987-12-15 Maruko Seiyaku Co., Ltd. Ergoline derivatives and acid addition salts thereof

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714767D0 (en) * 1987-06-24 1987-07-29 Erba Farmitalia Egoline derivatives
HU190105B (en) * 1983-06-03 1986-08-28 Gyogyszerkutato Intezet Process for production of pirazolyl-methyl-ergolin- derivatives and their acid additional salts
GB8702364D0 (en) * 1987-02-03 1987-03-11 Erba Farmitalia Ergolinyl heterocycles
EP2566333A4 (fr) 2010-05-07 2014-04-02 Univ Leland Stanford Junior Identification de stabilisants de protéines multimériques
US20160045609A1 (en) 2014-08-14 2016-02-18 Mamoun M. Alhamadsheh Conjugation of pharmaceutically active agents with transthyretin ligands through adjustable linkers to increase serum half-life
NZ755597A (en) 2017-02-17 2023-06-30 Eidos Therapeutics Inc Processes for preparing ag-10, its intermediates, and salts thereof
MA52137A (fr) 2018-03-23 2021-01-27 Eidos Therapeutics Inc Méthodes de traitement de l'amylose ttr à l'aide d'ag10
KR20210046708A (ko) 2018-08-17 2021-04-28 에이도스 테라퓨틱스, 인코포레이티드 Ag10의 제형

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3238211A (en) * 1966-03-01 Derhvatives of g-methyl and i,g-dimethyl ergolhne
US3296071A (en) * 1963-05-31 1967-01-03 Upjohn Co Reducing blood sugar with 3-alkyl-5-alkoxymethylisoxazole
BE712054A (fr) * 1967-03-16 1968-07-15
US3957785A (en) * 1971-12-02 1976-05-18 Societa' Farmaceutici Italia S.P.A. Bβ-Pyrimidino-aminomethyl-10α-ergoline and 10α-methoxyergoline derivatives
CH563376A5 (fr) * 1972-06-29 1975-06-30 Lonza Ag
US3996228A (en) * 1973-12-21 1976-12-07 Societa' Farmaceutici Italia S.P.A. Pyrimidinoaminoethyl ergoline derivatives
NL7416120A (nl) * 1973-12-21 1975-06-24 Farmaceutici Italia Werkwijze voor het bereiden van pyrimidinoami- nomethylergolinederivaten.
US4147789A (en) * 1974-03-14 1979-04-03 Sandoz Ltd. 6-Methyl-8-thiomethyl-ergolene derivatives
IE41533B1 (en) * 1974-03-14 1980-01-30 Sandoz Ltd Thiomethyl ergolene derivatives
CS171480B1 (fr) * 1974-03-19 1976-10-29
CS177530B1 (en) * 1974-07-19 1977-07-29 Miroslav Semonsky New nbeta-substituted derivatives of b-beta-aminoethyl-ergoline-i their salts and methods for the production thereof
CH617452A5 (fr) * 1974-10-25 1980-05-30 Hoffmann La Roche
CH615929A5 (en) * 1975-06-02 1980-02-29 Sandoz Ag Process for the preparation of novel ergoline compounds
CH622518A5 (en) * 1976-12-14 1981-04-15 Sandoz Ag Process for the preparation of novel ergoline compounds
AU526764B2 (en) * 1978-09-08 1983-01-27 Farmitalia Carlo Erba S.P.A. Ergoline derivatives
GB2056437A (en) * 1979-08-07 1981-03-18 Erba Farmitalia Secoergoline derivatives
US4382940A (en) * 1979-12-06 1983-05-10 Farmitalia Carlo Erba S.P.A. Ercoline derivatives and therapeutic compositions having CNS affecting activity

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4713457A (en) * 1985-02-21 1987-12-15 Maruko Seiyaku Co., Ltd. Ergoline derivatives and acid addition salts thereof

Also Published As

Publication number Publication date
CS236874B2 (en) 1985-05-15
ATA156783A (de) 1987-07-15
SE8302379D0 (sv) 1983-04-27
IL68496A0 (en) 1983-07-31
FI73996B (fi) 1987-08-31
FI831406A0 (fi) 1983-04-25
IL68496A (en) 1985-06-30
ZA833008B (en) 1984-01-25
FI73996C (fi) 1987-12-10
DK164058C (da) 1992-10-12
GB8310843D0 (en) 1983-05-25
DE3314878C2 (fr) 1993-09-23
AU1402983A (en) 1983-11-03
FR2526022A1 (fr) 1983-11-04
DK189983D0 (da) 1983-04-28
AT385035B (de) 1988-02-10
IE830932L (en) 1983-10-30
NL191709B (nl) 1995-12-01
SE8302379L (sv) 1983-10-31
FR2526022B1 (fr) 1985-06-14
IE53950B1 (en) 1989-04-26
JPH0354668B2 (fr) 1991-08-20
GR78842B (fr) 1984-10-02
US4657914A (en) 1987-04-14
JPS58194884A (ja) 1983-11-12
CH654305A5 (it) 1986-02-14
FI831406L (fi) 1983-10-31
AU553851B2 (en) 1986-07-31
SE460967B (sv) 1989-12-11
NL8301529A (nl) 1983-11-16
IT8320807A0 (it) 1983-04-27
CA1210389A (fr) 1986-08-26
HU193527B (en) 1987-10-28
DE3314878A1 (de) 1983-11-03
DK189983A (da) 1983-10-31
NL191709C (nl) 1996-04-02
IT1215630B (it) 1990-02-22
GB2120242A (en) 1983-11-30
DK164058B (da) 1992-05-04

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A.

Effective date: 19980430