BE894927A - Derives de l'ergoline, procede pour leur preparation et medicaments les contenant - Google Patents

Derives de l'ergoline, procede pour leur preparation et medicaments les contenant

Info

Publication number
BE894927A
BE894927A BE0/209409A BE209409A BE894927A BE 894927 A BE894927 A BE 894927A BE 0/209409 A BE0/209409 A BE 0/209409A BE 209409 A BE209409 A BE 209409A BE 894927 A BE894927 A BE 894927A
Authority
BE
Belgium
Prior art keywords
preparation
medicaments containing
ergolin
derivatives
ergolin derivatives
Prior art date
Application number
BE0/209409A
Other languages
English (en)
Inventor
L Bernardi
A Temperilli
D Ruggieri
G Arcari
P Salvati
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of BE894927A publication Critical patent/BE894927A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12Nitrogen atoms
BE0/209409A 1981-11-06 1982-11-05 Derives de l'ergoline, procede pour leur preparation et medicaments les contenant BE894927A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8133631 1981-11-06

Publications (1)

Publication Number Publication Date
BE894927A true BE894927A (fr) 1983-05-05

Family

ID=10525712

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/209409A BE894927A (fr) 1981-11-06 1982-11-05 Derives de l'ergoline, procede pour leur preparation et medicaments les contenant

Country Status (21)

Country Link
US (1) US4500712A (fr)
JP (1) JPS5885886A (fr)
AT (1) AT381091B (fr)
AU (1) AU553903B2 (fr)
BE (1) BE894927A (fr)
CA (1) CA1191841A (fr)
CH (1) CH650506A5 (fr)
CS (1) CS232000B2 (fr)
DE (1) DE3240727A1 (fr)
DK (1) DK494882A (fr)
FI (1) FI73214C (fr)
FR (1) FR2516083A1 (fr)
GB (1) GB2112382B (fr)
GR (1) GR77055B (fr)
IE (1) IE54327B1 (fr)
IL (1) IL67155A (fr)
IT (1) IT1205272B (fr)
NL (1) NL8204225A (fr)
SE (1) SE452884B (fr)
SU (1) SU1189347A3 (fr)
ZA (1) ZA828095B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3151912A1 (de) * 1981-12-23 1983-06-30 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue ergolin-aminoderivate, verfahren zu ihrer herstellung und deren verwendung als arzneimittel
PH21123A (en) * 1983-04-28 1987-07-27 Erba Farmitalia Ergoline derivatives
DE3413657A1 (de) * 1984-04-09 1985-10-17 Schering AG, 1000 Berlin und 4709 Bergkamen Neue ergoline
EP0160842B1 (fr) * 1984-04-09 1994-06-22 Schering Aktiengesellschaft Dérivés d'ergoline substitués sur la position 2, procédés pour leur préparation et leur utilisation comme médicaments
GB2173189B (en) * 1985-02-21 1988-04-27 Maruko Pharmaceutical Co Ergoline derivatives and salts thereof and pharmaceutical compositions thereof
GB8515528D0 (en) * 1985-06-19 1985-07-24 Erba Farmitalia Ergoline derivatives
DE3528584A1 (de) * 1985-08-06 1987-02-19 Schering Ag Neue 1-alkyl-ergolin-thioharnstoffderivate
DE3533672A1 (de) * 1985-09-19 1987-03-26 Schering Ag Neue 12- und 13-substituierte ergolinderivate
DE3535930A1 (de) * 1985-10-04 1987-04-09 Schering Ag Neue 2-substituierte ergolinderivate
DE19832191A1 (de) * 1998-07-17 2000-01-27 Knoell Hans Forschung Ev Neuartige Ergolinamin-Derivate und ihre Verwendung
DE60231403D1 (de) 2001-06-08 2009-04-16 Sod Conseils Rech Applic Chimere somatostatin-dopamin-analoga
WO2006104141A1 (fr) * 2005-03-29 2006-10-05 Shionogi & Co., Ltd. Dérivé de 3-propénylcéphème
TWI523863B (zh) 2012-11-01 2016-03-01 艾普森藥品公司 體抑素-多巴胺嵌合體類似物
CN104768565B (zh) 2012-11-01 2017-04-26 益普生制药股份有限公司 促生长素抑制素类似物及其二聚体

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3238211A (en) * 1966-03-01 Derhvatives of g-methyl and i,g-dimethyl ergolhne
AT258479B (de) * 1961-05-29 1967-11-27 Farmaceutici Italia Verfahren zur Herstellung von neuen Verbindungen aus der Klasse des D-6-Methyl- (und -1,6-Dimethyl)-8-amino-methyl-ergolins I
GB1005880A (en) * 1961-11-10 1965-09-29 Sandoz Ag Ergolene and ergoline derivatives
GB1138419A (en) * 1966-07-29 1969-01-01 Farmaceutici Italia Ergoline derivatives
BE712054A (fr) * 1967-03-16 1968-07-15
BR6915443D0 (pt) * 1969-07-18 1973-03-13 Farmaceutici Italia Processo para a preparacao de derivados de ergolina
US3966941A (en) * 1970-09-23 1976-06-29 Spofa United Pharmaceutical Works Composition for preventing lactation or pregnancy in mammals and the method for using the same
DK140596B (da) * 1971-05-19 1979-10-08 Sandoz Ag Analogifremgangsmåde til fremstilling af 8beta-(ureidomethyl)-ergolenderivater.
NL7416120A (nl) * 1973-12-21 1975-06-24 Farmaceutici Italia Werkwijze voor het bereiden van pyrimidinoami- nomethylergolinederivaten.
US3996228A (en) * 1973-12-21 1976-12-07 Societa' Farmaceutici Italia S.P.A. Pyrimidinoaminoethyl ergoline derivatives
GB1573621A (en) * 1976-01-02 1980-08-28 Sandoz Ltd Acylated 6-methyl-8a-amino-ergoline i compounds
DE2656344A1 (de) * 1975-12-23 1977-07-07 Sandoz Ag Ergolinderivate, ihre verwendung und herstellung
HU178396B (en) * 1978-03-20 1982-04-28 Vianova Kunstharz Ag Process for producing new 8-beta-hydrazion-methyl-ergoline-and -ergolene derivatives
DD138979A1 (de) * 1978-09-27 1979-12-05 Karlheinz Seifert Verfahren zur herstellung von acylthioharnstoffen mit ergolinstruktur
US4201862A (en) * 1979-03-16 1980-05-06 Eli Lilly And Company 2-Azaergolines and 2-aza-8(or 9)-ergolenes
DE3129714A1 (de) * 1981-07-23 1983-02-10 Schering Ag, 1000 Berlin Und 4619 Bergkamen Anti-psychotikum

Also Published As

Publication number Publication date
US4500712A (en) 1985-02-19
CS232000B2 (en) 1985-01-16
FI73214B (fi) 1987-05-29
IL67155A (en) 1985-07-31
IT1205272B (it) 1989-03-15
DK494882A (da) 1983-05-07
SE8206282L (sv) 1983-05-07
CH650506A5 (de) 1985-07-31
AT381091B (de) 1986-08-25
CA1191841A (fr) 1985-08-13
NL8204225A (nl) 1983-06-01
CS775282A2 (en) 1984-01-16
DE3240727A1 (de) 1983-05-19
SE452884B (sv) 1987-12-21
FR2516083B1 (fr) 1984-05-25
IL67155A0 (en) 1983-03-31
IT8224077A0 (it) 1982-11-04
GB2112382B (en) 1985-03-06
IE54327B1 (en) 1989-08-30
SE8206282D0 (sv) 1982-11-04
FI823727A0 (fi) 1982-11-01
FI73214C (fi) 1987-09-10
FI823727L (fi) 1983-05-07
FR2516083A1 (fr) 1983-05-13
ATA399682A (de) 1986-01-15
GR77055B (fr) 1984-09-05
SU1189347A3 (ru) 1985-10-30
IE822614L (en) 1983-05-06
AU553903B2 (en) 1986-07-31
GB2112382A (en) 1983-07-20
ZA828095B (en) 1983-09-28
AU9009082A (en) 1983-05-12
JPS5885886A (ja) 1983-05-23
JPS628433B2 (fr) 1987-02-23

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A.

Effective date: 19891130