FI824314L
(fi)
*
|
1981-12-16 |
1983-06-17 |
Sankyo Co |
Thienopyrimidin-derivater, deras framstaellning och deras medicinska anvaendning
|
JPS60146891A
(ja)
*
|
1984-01-05 |
1985-08-02 |
Mitsubishi Chem Ind Ltd |
〔2,3−d〕チエノピリミジン誘導体およびその塩
|
JPH068292B2
(ja)
*
|
1985-05-07 |
1994-02-02 |
アルカロイダ ベギエスゼティ ギャル |
トリアゾリルキノリン誘導体
|
US4670560A
(en)
*
|
1986-04-28 |
1987-06-02 |
Ortho Pharmaceutical Corporation |
Thienopyrimidine-2,4-dione derivatives and intermediates thereof
|
EP0364598A4
(en)
*
|
1988-03-02 |
1992-01-15 |
Yoshitomi Pharmaceutical Industries, Ltd. |
3,4-dihydrothieno 2,3-d¨pyrimidine compounds and pharmaceutical application thereof
|
US5280026A
(en)
*
|
1989-05-30 |
1994-01-18 |
Smithkline Beecham Intercredit B.V. |
Thienopyrimidines
|
GB8912335D0
(en)
*
|
1989-05-30 |
1989-07-12 |
Smithkline Beckman Intercredit |
Compounds
|
DE4008726A1
(de)
*
|
1990-03-19 |
1991-09-26 |
Basf Ag |
Thieno(2,3-d)pyrimidinderivate
|
BR9101256A
(pt)
*
|
1990-03-30 |
1991-11-05 |
Dowelanco |
Composto,composicao fungicida,processo fungicida,composicao inseticida ou acaricida e processo inseticida ou acaricida
|
US5869486A
(en)
*
|
1995-02-24 |
1999-02-09 |
Ono Pharmaceutical Co., Ltd. |
Fused pyrimidines and pyriazines as pharmaceutical compounds
|
DE69624536T2
(de)
*
|
1995-08-08 |
2003-06-05 |
Ono Pharmaceutical Co |
Hydroxamsäurederivate verwendbar zur Hemmung von Gelatinase
|
DE19632423A1
(de)
*
|
1996-08-12 |
1998-02-19 |
Merck Patent Gmbh |
Thienopyrimidine
|
DE19650378A1
(de)
*
|
1996-12-05 |
1998-06-10 |
Basf Ag |
Neue Pyrimidylverbindungen als Pflanzenschutzmittel
|
AU5698398A
(en)
*
|
1996-12-18 |
1998-07-15 |
Eli Lilly And Company |
Combinatorial process for preparing fused pyrimidine libraries
|
US20030162795A1
(en)
*
|
1998-10-22 |
2003-08-28 |
Pfizer Inc. |
Thienopyrimidine and thienopyridine derivatives useful as anticancer agents
|
US6133271A
(en)
*
|
1998-11-19 |
2000-10-17 |
Cell Pathways, Inc. |
Method for inhibiting neoplastic cells and related conditions by exposure thienopyrimidine derivatives
|
US6608053B2
(en)
*
|
2000-04-27 |
2003-08-19 |
Yamanouchi Pharmaceutical Co., Ltd. |
Fused heteroaryl derivatives
|
US6503914B1
(en)
*
|
2000-10-23 |
2003-01-07 |
Board Of Regents, The University Of Texas System |
Thienopyrimidine-based inhibitors of the Src family
|
WO2002088138A1
(fr)
*
|
2001-04-30 |
2002-11-07 |
Bayer Corporation |
Nouveaux thiopheno[2,3-d]pyrimidines 4-amino-5,6-substitutes
|
US6805491B2
(en)
*
|
2002-05-20 |
2004-10-19 |
Stratos International, Inc. |
Stub having an optical fiber
|
AR044743A1
(es)
*
|
2002-09-26 |
2005-10-05 |
Nihon Nohyaku Co Ltd |
Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,
|
US20050222175A1
(en)
*
|
2004-03-31 |
2005-10-06 |
Dhanoa Dale S |
New piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
EP1622914B1
(fr)
*
|
2003-03-31 |
2011-06-01 |
Trovis Pharmaceuticals LLC |
Nouveaux composes de piperidinylamino-thieno[2,3-d] pyrimidine
|
US7612078B2
(en)
*
|
2003-03-31 |
2009-11-03 |
Epix Delaware, Inc. |
Piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
GB0315950D0
(en)
|
2003-06-11 |
2003-08-13 |
Xention Discovery Ltd |
Compounds
|
US7488736B2
(en)
*
|
2004-05-17 |
2009-02-10 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
GB0412467D0
(en)
*
|
2004-06-04 |
2004-07-07 |
Astrazeneca Ab |
Chemical compounds
|
GB0412986D0
(en)
|
2004-06-10 |
2004-07-14 |
Xention Discovery Ltd |
Compounds
|
JP2008506714A
(ja)
*
|
2004-07-16 |
2008-03-06 |
サネシス ファーマシューティカルズ, インコーポレイテッド |
オーロラキナーゼインヒビターとして有用なチエノピリミジン
|
GB0420719D0
(en)
*
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
US7598265B2
(en)
*
|
2004-09-30 |
2009-10-06 |
Epix Delaware, Inc. |
Compositions and methods for treating CNS disorders
|
US7576211B2
(en)
*
|
2004-09-30 |
2009-08-18 |
Epix Delaware, Inc. |
Synthesis of thienopyridinone compounds and related intermediates
|
US7407966B2
(en)
*
|
2004-10-07 |
2008-08-05 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
CA2583259C
(fr)
*
|
2004-10-08 |
2011-08-02 |
Astellas Pharma Inc. |
Derive polycyclique aromatique de pyrimidine
|
EP1802632B1
(fr)
*
|
2004-10-21 |
2011-07-13 |
Dow AgroSciences LLC |
Composes de thieno-pyrimidine possedant une activite fongicide
|
GB0423653D0
(en)
|
2004-10-25 |
2004-11-24 |
Piramed Ltd |
Pharmaceutical compounds
|
US7576212B2
(en)
|
2004-12-09 |
2009-08-18 |
Xention Limited |
Thieno[2,3-B] pyridines as potassium channel inhibitors
|
US7576080B2
(en)
*
|
2004-12-23 |
2009-08-18 |
Memory Pharmaceuticals Corporation |
Certain thienopyrimidine derivatives as phosphodiesterase 10 inhibitors
|
US7816351B2
(en)
*
|
2005-09-23 |
2010-10-19 |
Equispharm Co., Ltd |
5,6-dimethylthieno[2,3-di] pyrimidine derivatives, the preparation method thereof and the pharmaceutical composition comprising the same for anti-virus
|
EP1937691A1
(fr)
*
|
2005-10-21 |
2008-07-02 |
Dow Agrosciences LLC |
Composes de thieno-pyrimidine a activite fongicide
|
US7531482B2
(en)
*
|
2005-10-21 |
2009-05-12 |
Dow Agrosciences Llc |
Thieno-pyrimidine compounds having fungicidal activity
|
WO2007056215A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc. |
N-aryl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation associee
|
US20070213305A1
(en)
*
|
2005-11-02 |
2007-09-13 |
Cytovia, Inc. |
N-alkyl-N-aryl-thienopyrimidin-4-amines and analogs as activators of caspases and inducers of apoptosis and the use thereof
|
WO2007056208A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc. |
N-arylalkyl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation de ceux-ci
|
GB0525164D0
(en)
|
2005-12-09 |
2006-01-18 |
Xention Discovery Ltd |
Compounds
|
TWI417095B
(zh)
|
2006-03-15 |
2013-12-01 |
Janssen Pharmaceuticals Inc |
1,4-二取代之3-氰基-吡啶酮衍生物及其作為mGluR2-受體之正向異位性調節劑之用途
|
DK2024372T3
(da)
*
|
2006-04-26 |
2010-09-20 |
Hoffmann La Roche |
Thieno[3,2-d]pyrimidin-derivat, der er egnet som P13K inhibitor
|
EP2402347A1
(fr)
|
2006-04-26 |
2012-01-04 |
F. Hoffmann-La Roche AG |
Composés pharmaceutiques
|
AR060632A1
(es)
|
2006-04-26 |
2008-07-02 |
Genentech Inc |
Compuestos inhibidores de fosfoinositida 3- quinasa y metodos de uso
|
WO2007135029A1
(fr)
|
2006-05-22 |
2007-11-29 |
Basf Se |
Méthodes insecticides utilisant des composés de 4-amino-5-chloro-thiéno[2,3-d]-pyrimidine
|
NZ578162A
(en)
*
|
2006-12-07 |
2011-12-22 |
Genentech Inc |
Phosphoinositide 3-kinase inhibitor compounds and methods of use
|
KR101507182B1
(ko)
*
|
2006-12-07 |
2015-03-30 |
제넨테크, 인크. |
포스포이노시타이드 3-키나제 억제제 화합물 및 그의 사용 방법
|
TW200900065A
(en)
|
2007-03-07 |
2009-01-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
|
TW200845978A
(en)
*
|
2007-03-07 |
2008-12-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
|
US7928111B2
(en)
*
|
2007-06-08 |
2011-04-19 |
Senomyx, Inc. |
Compounds including substituted thienopyrimidinone derivatives as ligands for modulating chemosensory receptors
|
US8633186B2
(en)
|
2007-06-08 |
2014-01-21 |
Senomyx Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
US9603848B2
(en)
*
|
2007-06-08 |
2017-03-28 |
Senomyx, Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
CA2698929C
(fr)
*
|
2007-09-14 |
2016-01-19 |
Addex Pharma S.A. |
4-phenyle-1h-pyridine-2-ones 1,3-disubstituees
|
AU2008297876B2
(en)
|
2007-09-14 |
2011-07-07 |
Addex Pharma S.A. |
1,3-disubstituted 4-(aryl-x-phenyl)-1h-pyridin-2-ones
|
ATE496906T1
(de)
|
2007-09-14 |
2011-02-15 |
Ortho Mcneil Janssen Pharm |
1',3'-disubstituierte 4-phenyl-3,4,5,6-tetrahydro-2h,1'h-ä1,4'übipyri inyl-2'-one
|
CN101909631B
(zh)
|
2007-10-25 |
2012-09-12 |
健泰科生物技术公司 |
制备噻吩并嘧啶化合物的方法
|
GB0721095D0
(en)
*
|
2007-10-26 |
2007-12-05 |
Piramed Ltd |
Pharmaceutical compounds
|
CN101861316B
(zh)
*
|
2007-11-14 |
2013-08-21 |
奥梅-杨森制药有限公司 |
咪唑并[1,2-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途
|
US8609173B2
(en)
|
2008-07-31 |
2013-12-17 |
Senomyx Inc. |
Compositions comprising sweetness enhancers and methods of making them
|
EP2323997B1
(fr)
|
2008-07-31 |
2017-09-06 |
Senomyx, Inc. |
Procédés et intermédiaires pour la réalisation d`exhausteurs de goût sucré
|
CA2735764C
(fr)
|
2008-09-02 |
2016-06-14 |
Ortho-Mcneil-Janssen Pharmaceuticals, Inc. |
Derives de 3-azabicyclo[3.1.0]hexyle comme modulateurs des recepteurs metabotropiques du glutamate
|
AU2009304293B2
(en)
|
2008-10-16 |
2012-04-26 |
Addex Pharma S.A. |
Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
|
US8691813B2
(en)
|
2008-11-28 |
2014-04-08 |
Janssen Pharmaceuticals, Inc. |
Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
|
EP2445877B1
(fr)
*
|
2008-12-03 |
2014-07-23 |
Nanotherapeutics, Inc. |
Composés bicycliques et leurs procédés de fabrication et d'utilisation
|
CA2760259C
(fr)
|
2009-05-12 |
2018-05-01 |
Janssen Pharmaceuticals, Inc. |
Derives de la 1,2,4-triazolo [4,3-a] pyridine et leur utilisation en tant que modulateurs allosteriques positifs des recepteurs mglur2
|
MY153913A
(en)
|
2009-05-12 |
2015-04-15 |
Janssen Pharmaceuticals Inc |
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
|
RS53075B
(en)
|
2009-05-12 |
2014-04-30 |
Janssen Pharmaceuticals Inc. |
1,2,4-TRIAZOLO [4,3-A] PYRIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OR PREVENTION OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS
|
CA2761445A1
(fr)
*
|
2009-05-27 |
2010-12-02 |
Genentech, Inc. |
Composes pyrimidines bicycliques inhibiteurs de pi3k selectifs pour p110 delta, et procedes d'utilisation
|
US8158625B2
(en)
*
|
2009-05-27 |
2012-04-17 |
Genentech, Inc. |
Bicyclic indole-pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use
|
TWI485138B
(zh)
*
|
2009-07-16 |
2015-05-21 |
Sds Biotech Corp |
4- (3-butynyl) aminopyrimidine derivatives as a pest control agent for agricultural and horticulture
|
BR112012002164B1
(pt)
*
|
2009-07-30 |
2021-04-20 |
Merial, Inc |
compostos inseticidas de 4-amino-tieno[2,3-d]-pirimidina e métodos para seu uso
|
PE20121816A1
(es)
*
|
2009-10-12 |
2013-01-02 |
Hoffmann La Roche |
Combinaciones de un inhibidor de pi3k y un inhibidor de mek
|
WO2012012712A2
(fr)
*
|
2010-07-23 |
2012-01-26 |
President And Fellows Of Harvard College |
Composés renforçant l'activité protéasome tricyclique
|
BR112013003332B1
(pt)
|
2010-08-12 |
2018-11-13 |
Senomyx, Inc. |
método para melhorar a estabilidade de intensificador de doce e composição contendo intensificador de doce estabilizado
|
PL2649069T3
(pl)
|
2010-11-08 |
2016-01-29 |
Janssen Pharmaceuticals Inc |
Pochodne 1,2,4-triazolo[4,3-a]pirydyny i ich zastosowanie jako dodatnich allosterycznych modulatorów receptorów mGluR2
|
EP2661435B1
(fr)
|
2010-11-08 |
2015-08-19 |
Janssen Pharmaceuticals, Inc. |
Dérivés 1,2,4-triazolo[4,3-a]pyridine et leur utilisation en tant que modulateurs allostériques positifs des récepteurs mglur2
|
EP2643320B1
(fr)
|
2010-11-08 |
2015-03-04 |
Janssen Pharmaceuticals, Inc. |
Dérivés de la 1,2,4-triazolo [4,3-a] pyridine et leur utilisation en tant que modulateurs allostériques positifs des récepteurs mglur2
|
SI2651951T1
(sl)
|
2010-12-16 |
2015-01-30 |
F. Hoffmann-La Roche Ag |
Tricikliäśne p13k inhibitorske spojine in postopki uporabe
|
EP2664238A4
(fr)
*
|
2011-01-14 |
2014-09-17 |
Sds Biotech Corp |
Composition de lutte contre les organismes nuisibles contenant un dérivé de 4-(3-butynyl)aminopyrimidine pour utilisation agricole ou horticole
|
KR20130116358A
(ko)
*
|
2011-02-09 |
2013-10-23 |
에프. 호프만-라 로슈 아게 |
Pi3 키나아제 억제제로서 헤테로사이클릭 화합물
|
CN103946226A
(zh)
|
2011-07-19 |
2014-07-23 |
无限药品股份有限公司 |
杂环化合物及其应用
|
PE20191204A1
(es)
|
2012-08-06 |
2019-09-10 |
Firmenich Incorporated |
Modificador del sabor dulce
|
JO3155B1
(ar)
|
2013-02-19 |
2017-09-20 |
Senomyx Inc |
معدِّل نكهة حلوة
|
JO3368B1
(ar)
|
2013-06-04 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
|
JO3367B1
(ar)
|
2013-09-06 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
|
KR20200126026A
(ko)
|
2014-01-21 |
2020-11-05 |
얀센 파마슈티카 엔.브이. |
대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
|
CN109999033B
(zh)
|
2014-01-21 |
2022-12-23 |
詹森药业有限公司 |
包括代谢型谷氨酸能受体亚型2的正别构调节物或正位激动剂的组合及其用途
|
CN104725398B
(zh)
*
|
2015-01-29 |
2017-01-18 |
杨威 |
一种jak/stat3磷酸化抑制剂及其制备方法与用途
|
WO2017019537A1
(fr)
*
|
2015-07-24 |
2017-02-02 |
University Of Louisville Research Foundation, Inc. |
Composés, compositions, procédés pour le traitement de maladies et procédés pour la préparation de composés
|
WO2019018359A1
(fr)
*
|
2017-07-17 |
2019-01-24 |
Saint Louis University |
Thiéno[2,3-d]pyrimidines et benzofuro(3,2-d) pyrimidines utiles en tant qu'agents antimicrobiens
|
BR112021002261A2
(pt)
|
2018-08-07 |
2021-05-04 |
Firmenich Incorporated |
2,2-dióxidos de 4-amino-1h-benzo[c][1,2,6]tiadiazina 5-substituídos e formulações e usos dos mesmos
|