AU697832B2 - New thiophene compounds, process for their preparation and pharmaceutical compositions containing them - Google Patents
New thiophene compounds, process for their preparation and pharmaceutical compositions containing them Download PDFInfo
- Publication number
- AU697832B2 AU697832B2 AU45675/96A AU4567596A AU697832B2 AU 697832 B2 AU697832 B2 AU 697832B2 AU 45675/96 A AU45675/96 A AU 45675/96A AU 4567596 A AU4567596 A AU 4567596A AU 697832 B2 AU697832 B2 AU 697832B2
- Authority
- AU
- Australia
- Prior art keywords
- formula
- compound
- och
- compounds
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9502061A FR2730996B1 (fr) | 1995-02-23 | 1995-02-23 | Nouveaux composes du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant |
| FR9502061 | 1995-02-23 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU4567596A AU4567596A (en) | 1996-08-29 |
| AU697832B2 true AU697832B2 (en) | 1998-10-15 |
Family
ID=9476411
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU45675/96A Ceased AU697832B2 (en) | 1995-02-23 | 1996-02-21 | New thiophene compounds, process for their preparation and pharmaceutical compositions containing them |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US5705525A (el) |
| EP (1) | EP0728755B1 (el) |
| JP (1) | JPH08253470A (el) |
| CN (1) | CN1058965C (el) |
| AT (1) | ATE200488T1 (el) |
| AU (1) | AU697832B2 (el) |
| CA (1) | CA2170097C (el) |
| CY (1) | CY2262B1 (el) |
| DE (1) | DE69612416T2 (el) |
| DK (1) | DK0728755T3 (el) |
| ES (1) | ES2158255T3 (el) |
| FI (1) | FI960795A (el) |
| FR (1) | FR2730996B1 (el) |
| GR (1) | GR3036192T3 (el) |
| NO (1) | NO314997B1 (el) |
| NZ (1) | NZ286045A (el) |
| PT (1) | PT728755E (el) |
| ZA (1) | ZA961472B (el) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999018099A1 (en) * | 1997-10-03 | 1999-04-15 | Merck Frosst Canada & Co. | Aryl thiophene derivatives as pde iv inhibitors |
| AUPR283801A0 (en) * | 2001-02-01 | 2001-03-01 | Australian National University, The | Chemical compounds and methods |
| FR2860792B1 (fr) * | 2003-10-10 | 2006-02-24 | Sanofi Synthelabo | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique |
| KR20220100607A (ko) * | 2019-10-28 | 2022-07-15 | 상하이 인스티튜트 오브 마테리아 메디카 차이니즈 아카데미 오브 싸이언시즈 | 5원 헤테로사이클릭 옥소카르복실산 화합물 및 이의 의약 용도 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0055471A1 (en) * | 1980-12-29 | 1982-07-07 | E.I. Du Pont De Nemours And Company | Antiinflammatory 4,5-diaryl-alpha,alpha-bis(polyhalomethyl)-2-thiophenemethanamines |
| GB8525716D0 (en) * | 1985-10-18 | 1985-11-20 | Roussel Lab Ltd | Chemical compounds |
| FR2655043B1 (fr) * | 1989-11-24 | 1992-02-07 | Adir | Nouveaux derives du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant. |
| GB9012936D0 (en) * | 1990-06-11 | 1990-08-01 | Fujisawa Pharmaceutical Co | Thiophene derivatives,processes for preparation thereof and pharmaceutical composition comprising the same |
| US5571810A (en) * | 1990-06-11 | 1996-11-05 | Fujisawa Pharmaceutical Co., Ltd. | Thiophene derivatives |
-
1995
- 1995-02-23 FR FR9502061A patent/FR2730996B1/fr not_active Expired - Fee Related
-
1996
- 1996-02-17 CN CN96106004A patent/CN1058965C/zh not_active Expired - Fee Related
- 1996-02-21 FI FI960795A patent/FI960795A/fi not_active IP Right Cessation
- 1996-02-21 AU AU45675/96A patent/AU697832B2/en not_active Ceased
- 1996-02-22 US US08/605,537 patent/US5705525A/en not_active Ceased
- 1996-02-22 AT AT96400359T patent/ATE200488T1/de not_active IP Right Cessation
- 1996-02-22 PT PT96400359T patent/PT728755E/pt unknown
- 1996-02-22 DK DK96400359T patent/DK0728755T3/da active
- 1996-02-22 CA CA002170097A patent/CA2170097C/fr not_active Expired - Fee Related
- 1996-02-22 EP EP96400359A patent/EP0728755B1/fr not_active Expired - Lifetime
- 1996-02-22 JP JP8035131A patent/JPH08253470A/ja active Pending
- 1996-02-22 NO NO19960706A patent/NO314997B1/no unknown
- 1996-02-22 ES ES96400359T patent/ES2158255T3/es not_active Expired - Lifetime
- 1996-02-22 NZ NZ286045A patent/NZ286045A/en unknown
- 1996-02-22 DE DE69612416T patent/DE69612416T2/de not_active Expired - Fee Related
- 1996-02-23 ZA ZA961472A patent/ZA961472B/xx unknown
-
1999
- 1999-08-03 US US09/368,343 patent/USRE37078E1/en not_active Expired - Fee Related
-
2001
- 2001-07-09 GR GR20010401040T patent/GR3036192T3/el not_active IP Right Cessation
-
2002
- 2002-03-27 CY CY0200012A patent/CY2262B1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ286045A (en) | 1996-10-28 |
| CA2170097C (fr) | 2002-02-26 |
| CA2170097A1 (fr) | 1996-08-24 |
| NO960706D0 (no) | 1996-02-22 |
| NO960706L (no) | 1996-08-26 |
| AU4567596A (en) | 1996-08-29 |
| FR2730996B1 (fr) | 1997-06-20 |
| FI960795A0 (fi) | 1996-02-21 |
| JPH08253470A (ja) | 1996-10-01 |
| US5705525A (en) | 1998-01-06 |
| NO314997B1 (no) | 2003-06-23 |
| GR3036192T3 (en) | 2001-10-31 |
| CN1142496A (zh) | 1997-02-12 |
| DK0728755T3 (da) | 2001-07-30 |
| ZA961472B (en) | 1996-08-28 |
| EP0728755A1 (fr) | 1996-08-28 |
| CY2262B1 (en) | 2003-07-04 |
| FI960795A (fi) | 1996-08-24 |
| FR2730996A1 (fr) | 1996-08-30 |
| PT728755E (pt) | 2001-09-28 |
| EP0728755B1 (fr) | 2001-04-11 |
| ES2158255T3 (es) | 2001-09-01 |
| DE69612416T2 (de) | 2001-11-22 |
| ATE200488T1 (de) | 2001-04-15 |
| USRE37078E1 (en) | 2001-02-27 |
| CN1058965C (zh) | 2000-11-29 |
| DE69612416D1 (de) | 2001-05-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Assignment registered |
Owner name: LES LABORATOIRES SERVIER Free format text: FORMER OWNER WAS: ADIR ET COMPAGNIE |