FR2860792B1 - Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique - Google Patents
Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2860792B1 FR2860792B1 FR0311861A FR0311861A FR2860792B1 FR 2860792 B1 FR2860792 B1 FR 2860792B1 FR 0311861 A FR0311861 A FR 0311861A FR 0311861 A FR0311861 A FR 0311861A FR 2860792 B1 FR2860792 B1 FR 2860792B1
- Authority
- FR
- France
- Prior art keywords
- thiophene
- preparation
- therapeutic use
- carboxamide derivatives
- carboxamide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Pulmonology (AREA)
- Reproductive Health (AREA)
- Ophthalmology & Optometry (AREA)
- Gastroenterology & Hepatology (AREA)
Priority Applications (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0311861A FR2860792B1 (fr) | 2003-10-10 | 2003-10-10 | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique |
ARP040103632A AR046056A1 (es) | 2003-10-10 | 2004-10-07 | Derivados de tiofeno-2-carboxamida y su uso como antagonistas de los receptores canabinoides cb1 |
TW093130467A TW200526647A (en) | 2003-10-10 | 2004-10-08 | Thiophene-2-carboxamide derivatives, their preparation and their therapeutic application |
EP04791498A EP1678159A2 (fr) | 2003-10-10 | 2004-10-08 | Derives de thiophene-2-carboxamide et leurs utilisation comme antagonistes des recepteurs cb1 des cannabinoides |
JP2006530423A JP2007508279A (ja) | 2003-10-10 | 2004-10-08 | チオフェン−2−カルボキサミド誘導体、それらの製造、および治療適用 |
PCT/FR2004/002546 WO2005035488A2 (fr) | 2003-10-10 | 2004-10-08 | Derives de thiophene-2-carboxamide et leurs utilisation comme antagonistes des recepteurs cb1 des cannabinoides |
US11/400,702 US7462631B2 (en) | 2003-10-10 | 2006-04-07 | Thiophene-2-carboxamide derivatives, preparation and therapeutic application thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0311861A FR2860792B1 (fr) | 2003-10-10 | 2003-10-10 | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2860792A1 FR2860792A1 (fr) | 2005-04-15 |
FR2860792B1 true FR2860792B1 (fr) | 2006-02-24 |
Family
ID=34355379
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0311861A Expired - Fee Related FR2860792B1 (fr) | 2003-10-10 | 2003-10-10 | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique |
Country Status (7)
Country | Link |
---|---|
US (1) | US7462631B2 (fr) |
EP (1) | EP1678159A2 (fr) |
JP (1) | JP2007508279A (fr) |
AR (1) | AR046056A1 (fr) |
FR (1) | FR2860792B1 (fr) |
TW (1) | TW200526647A (fr) |
WO (1) | WO2005035488A2 (fr) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2880023B1 (fr) * | 2004-12-23 | 2007-02-23 | Sanofi Aventis Sa | Derives de n-[(4,5-diphenyl-3-alkyl-2-thienyl) methyl] amine leur preparation et leur application en therapeutique |
FR2880890B1 (fr) * | 2005-01-19 | 2007-03-30 | Sanofi Aventis Sa | Derives de n-[(4,5-diphenyl-2-thienyl)methyl]sulfonamide, leur preparation et leur application en therapeutique |
FR2881744B1 (fr) | 2005-02-09 | 2007-04-27 | Sanofi Aventis Sa | Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique |
DE102008015032A1 (de) | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte Pyrazolamide und ihre Verwendung |
DE102008015033A1 (de) | 2008-03-17 | 2009-09-24 | Aicuris Gmbh & Co. Kg | Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung |
FR2934594B1 (fr) * | 2008-08-01 | 2010-09-10 | Sanofi Aventis | Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique. |
DE102008062863A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte (Thiophenyl-carbonyl)imidazolidinone und ihre Verwendung |
DE102008062878A1 (de) | 2008-12-17 | 2010-06-24 | Aicuris Gmbh & Co. Kg | Substituierte Furancarboxamide und ihre Verwendung |
FR2943672B1 (fr) * | 2009-03-27 | 2011-03-25 | Sanofi Aventis | Derives de 3-alcoxy-4,5-diarylthiophene-2-carboxamide,leur preparation et leur application en therapeutique. |
MX2019004214A (es) * | 2016-10-12 | 2019-06-10 | Res Triangle Inst | Agonistas heterociclicos del receptor de apelina (apj) y usos de los mismos. |
US11306067B2 (en) | 2018-03-05 | 2022-04-19 | Denovamed Inc. | Diphenyl substituted thiophene-2-amide derivatives and pharmaceutical compositions thereof useful as antimicrobial |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0753716B2 (ja) * | 1986-07-02 | 1995-06-07 | 吉富製薬株式会社 | イミダゾ−ルカルボキサミド誘導体 |
GB9012936D0 (en) * | 1990-06-11 | 1990-08-01 | Fujisawa Pharmaceutical Co | Thiophene derivatives,processes for preparation thereof and pharmaceutical composition comprising the same |
US5474995A (en) * | 1993-06-24 | 1995-12-12 | Merck Frosst Canada, Inc. | Phenyl heterocycles as cox-2 inhibitors |
FR2730996B1 (fr) * | 1995-02-23 | 1997-06-20 | Adir | Nouveaux composes du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant |
AU2002319627A1 (en) * | 2001-07-20 | 2003-03-03 | Merck And Co., Inc. | Substituted imidazoles as cannabinoid receptor modulators |
EP1412347B1 (fr) * | 2001-08-01 | 2006-01-11 | Basell Polyolefine GmbH | Procede de preparation de derives heterocycliques de pentalene |
WO2003037886A2 (fr) * | 2001-10-30 | 2003-05-08 | Pharmacia Corporation | Derives de carboxamide heteroaromatique destines au traitement des inflammations |
AR038966A1 (es) * | 2002-03-18 | 2005-02-02 | Solvay Pharm Bv | Derivados de tiazol que tienen actividad antagonista, agonista o agonista parcial de cb1 |
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2003
- 2003-10-10 FR FR0311861A patent/FR2860792B1/fr not_active Expired - Fee Related
-
2004
- 2004-10-07 AR ARP040103632A patent/AR046056A1/es not_active Application Discontinuation
- 2004-10-08 EP EP04791498A patent/EP1678159A2/fr not_active Withdrawn
- 2004-10-08 TW TW093130467A patent/TW200526647A/zh unknown
- 2004-10-08 JP JP2006530423A patent/JP2007508279A/ja active Pending
- 2004-10-08 WO PCT/FR2004/002546 patent/WO2005035488A2/fr active Application Filing
-
2006
- 2006-04-07 US US11/400,702 patent/US7462631B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
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WO2005035488A2 (fr) | 2005-04-21 |
US7462631B2 (en) | 2008-12-09 |
US20060264470A1 (en) | 2006-11-23 |
JP2007508279A (ja) | 2007-04-05 |
FR2860792A1 (fr) | 2005-04-15 |
TW200526647A (en) | 2005-08-16 |
WO2005035488A3 (fr) | 2005-06-23 |
EP1678159A2 (fr) | 2006-07-12 |
AR046056A1 (es) | 2005-11-23 |
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