AU672675B2 - Thiazolopyrimidine derivatives - Google Patents

Thiazolopyrimidine derivatives Download PDF

Info

Publication number
AU672675B2
AU672675B2 AU59252/94A AU5925294A AU672675B2 AU 672675 B2 AU672675 B2 AU 672675B2 AU 59252/94 A AU59252/94 A AU 59252/94A AU 5925294 A AU5925294 A AU 5925294A AU 672675 B2 AU672675 B2 AU 672675B2
Authority
AU
Australia
Prior art keywords
group
carbon atoms
compounds
pyrimidine
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU59252/94A
Other languages
English (en)
Other versions
AU5925294A (en
Inventor
Haruko Chatani
Michio Iwahana
Hiroo Matsumoto
Kiyoshi Nakayama
Noriko Tanaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Pharmaceutical Co Ltd
Original Assignee
Daiichi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Pharmaceutical Co Ltd filed Critical Daiichi Pharmaceutical Co Ltd
Publication of AU5925294A publication Critical patent/AU5925294A/en
Application granted granted Critical
Publication of AU672675B2 publication Critical patent/AU672675B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU59252/94A 1993-04-01 1994-03-31 Thiazolopyrimidine derivatives Ceased AU672675B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP11087793 1993-04-01
JP5-110877 1993-04-01

Publications (2)

Publication Number Publication Date
AU5925294A AU5925294A (en) 1994-10-06
AU672675B2 true AU672675B2 (en) 1996-10-10

Family

ID=14546967

Family Applications (1)

Application Number Title Priority Date Filing Date
AU59252/94A Ceased AU672675B2 (en) 1993-04-01 1994-03-31 Thiazolopyrimidine derivatives

Country Status (9)

Country Link
US (1) US5599813A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0618208A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1100425A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU672675B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2120395A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI941487A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO941135L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PH (1) PH31256A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
TW (1) TW272193B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997049679A1 (fr) * 1996-06-27 1997-12-31 Ono Pharmaceutical Co., Ltd. Derives d'aryle (sulfure, oxyde sulfonique et sulfone) et medicaments les contenant en tant que principe actif
NZ508950A (en) 1998-07-13 2003-10-31 Univ Texas Cancer treatment methods using antibodies to aminophospholipids
EP1234585A3 (en) 1998-09-04 2004-01-21 The Regents Of The University Of Michigan Methods and compositions for the prevention or treatment of cancer
US6930101B1 (en) 1999-05-17 2005-08-16 The Regents Of The University Of California Thiazolopyrimidines useful as TNFα inhibitors
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
CN104130327A (zh) 2002-07-15 2014-11-05 得克萨斯大学体系董事会 与阴离子磷脂和氨基磷脂结合的抗体及其治疗和成像用途
KR101372783B1 (ko) 2004-01-22 2014-03-11 유니버시티 오브 마이애미 국소용 코-엔자임 큐10 제형 및 그의 사용 방법
RU2403258C2 (ru) 2004-10-07 2010-11-10 Бёрингер Ингельхайм Интернациональ Гмбх Тиазолилдигидроиндазолы
KR20100102110A (ko) 2007-11-09 2010-09-20 페레그린 파마수티컬즈, 인크 항-ｖｅｇｆ 항체 조성물 및 방법
WO2010011347A2 (en) 2008-07-25 2010-01-28 The Regents Of The University Of Colorado Clip inhibitors and methods of modulating immune function
CN101899058B (zh) * 2010-05-24 2012-05-23 中国人民解放军第四军医大学 一种噻唑并嘧啶化合物及其制备方法和应用
CN103443107B (zh) * 2011-03-28 2016-04-20 弗·哈夫曼-拉罗切有限公司 噻唑并嘧啶化合物
WO2018145109A1 (en) 2017-02-06 2018-08-09 Massachusetts Institute Of Technology Methods and products related to glutaminase inhibitors

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0038731A2 (fr) * 1980-04-08 1981-10-28 Synthelabo Dérivés de thiazole, leur préparation et leur application en thérapeutique
EP0045251B1 (fr) * 1980-07-24 1983-11-30 Rhone-Poulenc Sante Nouveaux dérivés de la thiazolo (3,2-a) pyrimidine, leur préparation et les médicaments qui les contiennent
EP0404525A2 (en) * 1989-06-21 1990-12-27 Takeda Chemical Industries, Ltd. Sulfur-containing fused pyrimidine derivatives, their production and use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1556878A (en) * 1976-01-19 1979-11-28 Diamond Shamrock Corp Imidazothiazoles
US4347248A (en) * 1981-03-23 1982-08-31 American Cyanamid Company 2,3-Disubstituted-thiazolo[3,2-a]pyrimidines

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0038731A2 (fr) * 1980-04-08 1981-10-28 Synthelabo Dérivés de thiazole, leur préparation et leur application en thérapeutique
EP0045251B1 (fr) * 1980-07-24 1983-11-30 Rhone-Poulenc Sante Nouveaux dérivés de la thiazolo (3,2-a) pyrimidine, leur préparation et les médicaments qui les contiennent
EP0404525A2 (en) * 1989-06-21 1990-12-27 Takeda Chemical Industries, Ltd. Sulfur-containing fused pyrimidine derivatives, their production and use

Also Published As

Publication number Publication date
US5599813A (en) 1997-02-04
CN1100425A (zh) 1995-03-22
FI941487L (fi) 1994-10-02
FI941487A7 (fi) 1994-10-02
PH31256A (en) 1998-06-18
AU5925294A (en) 1994-10-06
EP0618208A1 (en) 1994-10-05
CA2120395A1 (en) 1994-10-02
NO941135D0 (no) 1994-03-28
TW272193B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1996-03-11
FI941487A0 (fi) 1994-03-30
NO941135L (no) 1994-10-03

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