AU597159B2 - Process for the preparation of nitroethene derivatives - Google Patents

Process for the preparation of nitroethene derivatives Download PDF

Info

Publication number
AU597159B2
AU597159B2 AU13134/88A AU1313488A AU597159B2 AU 597159 B2 AU597159 B2 AU 597159B2 AU 13134/88 A AU13134/88 A AU 13134/88A AU 1313488 A AU1313488 A AU 1313488A AU 597159 B2 AU597159 B2 AU 597159B2
Authority
AU
Australia
Prior art keywords
general formula
compound corresponding
compound
process according
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU13134/88A
Other languages
English (en)
Other versions
AU1313488A (en
Inventor
Kurt Henning Dr Ahrens
Peter Dr. Morsdorf
Helmut Dr. Schickaneder
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Heumann Pharma GmbH and Co
Original Assignee
Heumann Pharma GmbH and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Heumann Pharma GmbH and Co filed Critical Heumann Pharma GmbH and Co
Publication of AU1313488A publication Critical patent/AU1313488A/en
Application granted granted Critical
Publication of AU597159B2 publication Critical patent/AU597159B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28—Radicals substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Furan Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU13134/88A 1987-04-06 1988-03-15 Process for the preparation of nitroethene derivatives Ceased AU597159B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP87105064A EP0285681B1 (de) 1987-04-06 1987-04-06 Verfahren zur Herstellung von Nitroethenderivaten
EP87105064 1987-04-06

Publications (2)

Publication Number Publication Date
AU1313488A AU1313488A (en) 1988-10-06
AU597159B2 true AU597159B2 (en) 1990-05-24

Family

ID=8196897

Family Applications (1)

Application Number Title Priority Date Filing Date
AU13134/88A Ceased AU597159B2 (en) 1987-04-06 1988-03-15 Process for the preparation of nitroethene derivatives

Country Status (17)

Country Link
US (1) US4968808A (enExample)
EP (1) EP0285681B1 (enExample)
JP (1) JP2755385B2 (enExample)
KR (1) KR940010179B1 (enExample)
AR (1) AR245116A1 (enExample)
AT (1) ATE86619T1 (enExample)
AU (1) AU597159B2 (enExample)
CA (1) CA1321594C (enExample)
DE (1) DE3784698D1 (enExample)
DK (1) DK155488A (enExample)
ES (1) ES2053462T3 (enExample)
GR (1) GR3007314T3 (enExample)
HU (1) HU200760B (enExample)
IE (1) IE61744B1 (enExample)
IL (1) IL85706A (enExample)
NZ (1) NZ223844A (enExample)
PT (1) PT87116B (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9009437D0 (en) * 1990-04-26 1990-06-20 Glaxo Group Ltd Chemical compounds
IN181698B (enExample) * 1994-05-13 1998-09-05 Ranbaxy Lab Ltd
ES2119268T3 (es) * 1994-06-24 1998-10-01 Ranbaxy Lab Ltd Procedimiento para fabricar ranitidina base de calidad farmaceutica.
US5470865A (en) * 1994-08-30 1995-11-28 Eli Lilly And Company Pharmaceutical composition
TR199900532T2 (xx) * 1996-09-11 1999-05-21 Knoll Aktiengesellschaft Nizatidin haz�rlanmas� i�in y�ntem.
IT1299198B1 (it) * 1998-03-05 2000-02-29 Nicox Sa Sali nitrati di farmaci antiulcera
JP2002529503A (ja) 1998-11-17 2002-09-10 ニトロメッド，インク． ニトロソ化及びニトロシル化ｈ２リセプターアンタゴニスト化合物及び組成物並びにその利用方法
US6555139B2 (en) 1999-06-28 2003-04-29 Wockhardt Europe Limited Preparation of micron-size pharmaceutical particles by microfluidization
US9457011B2 (en) * 2014-02-25 2016-10-04 Muslim D. Shahid Compositions and methods for the treatment of acid-related gastrointestinal disorders containing a dithiolane compound and a gastric acid secretion inhibitor

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1254583A (en) * 1982-03-19 1983-09-22 Eli Lilly And Company N-thiazolylmethyl thioalkyl-n:-alkenyl (or alkynyl) and related compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1421792A (en) * 1973-05-17 1976-01-21 Smith Kline French Lab Heterocyclic substituted-1, 1-diamino-ethylene derivatives methods for their preparation and compositions containing them
GB1565966A (en) * 1976-08-04 1980-04-23 Allen & Hanburys Ltd Aminoalkyl furan derivatives
US4233302A (en) * 1977-12-23 1980-11-11 Glaxo Group Limited Amine derivatives and pharmaceutical compositions containing them
US4760075A (en) * 1980-10-02 1988-07-26 Eli Lilly And Company N-thiazolylmethylthioalkyl-N-alkyl-amidines and related compounds
US4375547A (en) 1980-10-02 1983-03-01 Eli Lilly And Company N-Methyl-N'-2-([(2-dimethylaminomethyl)-4-thiazolyl]methylthio)ethyl 2-nitro-1,1-ethenediamine
ES507180A0 (es) * 1981-11-16 1982-08-16 Pharmedical Sa Lab Procedimiento de preparacion de amino alcosi furanos o tio- fenos.
US4625025A (en) * 1983-08-25 1986-11-25 Ube Industries, Ltd. Process for producing a 2H-1,3-thiazolidine, 2H-tetrahydro-1,3-thiazine, or 2H-hexahydro-1,3-thiazepine derivative substituted at the 2 position by a nitromethylene group derivative
EP0224612A1 (de) * 1985-12-05 1987-06-10 HEUMANN PHARMA GMBH & CO Verfahren zur Herstellung von N-Cyano-N'-methyl-N"[2-[[(5-methyl-1H-imidazol-4-yl)methyl]thio]ethyl]guanidin
US4777260A (en) * 1985-12-18 1988-10-11 Eli Lilly And Company Synthesis of nizatidine intermediate

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1254583A (en) * 1982-03-19 1983-09-22 Eli Lilly And Company N-thiazolylmethyl thioalkyl-n:-alkenyl (or alkynyl) and related compounds

Also Published As

Publication number Publication date
DK155488D0 (da) 1988-03-22
AR245116A1 (es) 1993-12-30
EP0285681B1 (de) 1993-03-10
KR940010179B1 (ko) 1994-10-22
US4968808A (en) 1990-11-06
PT87116B (pt) 1992-07-31
DE3784698D1 (de) 1993-04-15
IL85706A0 (en) 1988-08-31
JPS63258861A (ja) 1988-10-26
AU1313488A (en) 1988-10-06
KR880012579A (ko) 1988-11-28
GR3007314T3 (enExample) 1993-07-30
DK155488A (da) 1988-10-07
IE61744B1 (en) 1994-11-30
EP0285681A1 (de) 1988-10-12
IE880977L (en) 1988-10-06
PT87116A (pt) 1988-04-01
IL85706A (en) 1992-06-21
JP2755385B2 (ja) 1998-05-20
HU200760B (en) 1990-08-28
ATE86619T1 (de) 1993-03-15
CA1321594C (en) 1993-08-24
NZ223844A (en) 1989-12-21
ES2053462T3 (es) 1994-08-01

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired