AU2020352037A1 - Granule having masked unpleasant taste and method for producing same - Google Patents

Granule having masked unpleasant taste and method for producing same Download PDF

Info

Publication number
AU2020352037A1
AU2020352037A1 AU2020352037A AU2020352037A AU2020352037A1 AU 2020352037 A1 AU2020352037 A1 AU 2020352037A1 AU 2020352037 A AU2020352037 A AU 2020352037A AU 2020352037 A AU2020352037 A AU 2020352037A AU 2020352037 A1 AU2020352037 A1 AU 2020352037A1
Authority
AU
Australia
Prior art keywords
active ingredient
particle
granule
unpleasant taste
ethylcellulose
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU2020352037A
Other languages
English (en)
Inventor
Tatsuo Nomura
Toru Yasuzawa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nobelpharma Co Ltd
Original Assignee
Nobelpharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nobelpharma Co Ltd filed Critical Nobelpharma Co Ltd
Publication of AU2020352037A1 publication Critical patent/AU2020352037A1/en
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/24—Heavy metals; Compounds thereof
    • A61K33/30—Zinc; Compounds thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5089—Processes

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AU2020352037A 2019-09-25 2020-09-24 Granule having masked unpleasant taste and method for producing same Pending AU2020352037A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2019-173744 2019-09-25
JP2019173744 2019-09-25
PCT/JP2020/035883 WO2021060304A1 (ja) 2019-09-25 2020-09-24 不快な味がマスクされた顆粒剤及びその製造方法

Publications (1)

Publication Number Publication Date
AU2020352037A1 true AU2020352037A1 (en) 2022-04-21

Family

ID=75164923

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2020352037A Pending AU2020352037A1 (en) 2019-09-25 2020-09-24 Granule having masked unpleasant taste and method for producing same

Country Status (8)

Country Link
US (1) US20230016901A1 (https=)
EP (1) EP4035733A4 (https=)
JP (3) JP6905781B1 (https=)
CN (1) CN114340601A (https=)
AU (1) AU2020352037A1 (https=)
CA (1) CA3153004A1 (https=)
TW (1) TWI865615B (https=)
WO (1) WO2021060304A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2020352037A1 (en) * 2019-09-25 2022-04-21 Nobelpharma Co., Ltd. Granule having masked unpleasant taste and method for producing same
TR2022010921A2 (tr) * 2022-07-01 2024-01-22 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Tadı maskelenmiş bir çinko katı bileşimi.

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2542122B2 (ja) * 1990-04-18 1996-10-09 旭化成工業株式会社 球状核、球形顆粒およびその製造方法
JP3985907B2 (ja) 1996-01-18 2007-10-03 旭化成ケミカルズ株式会社 フィルムコーティング粒剤の製造方法
JP2000053563A (ja) 1998-08-07 2000-02-22 Bayer Yakuhin Ltd 苦味がマスクされた速放性細粒剤
KR101168189B1 (ko) * 2003-10-29 2012-07-25 시오노기세이야쿠가부시키가이샤 불쾌미를 개선한 피복 제제의 제조 방법
CN102048734B (zh) * 2005-05-26 2013-11-20 大日本住友制药株式会社 药物组合物
JP2007031292A (ja) * 2005-07-22 2007-02-08 Hamari Chemicals Ltd 亜鉛化合物含有組成物およびその製造方法
JP5271081B2 (ja) * 2006-07-26 2013-08-21 旭化成ケミカルズ株式会社 球形素顆粒およびその製造方法
JP2008081448A (ja) * 2006-09-28 2008-04-10 Kowa Pharmaceutical Co Ltd 酒石酸ゾルピデムの苦味マスキング速放性粒子
EP2486917B1 (en) * 2009-10-09 2020-11-25 Asahi Kasei Kabushiki Kaisha Coating film, and granules and tablets each utilizing same
AU2010325746B2 (en) * 2009-12-02 2016-02-25 Adare Pharmaceuticals S.R.L. Fexofenadine microcapsules and compositions containing them
CN102018658B (zh) * 2010-07-16 2014-03-12 钟术光 一种控释制剂及其制备方法
JP5823401B2 (ja) * 2010-09-13 2015-11-25 大鵬薬品工業株式会社 不快な味が遮蔽された薬物含有膜被覆粒子
AU2020352037A1 (en) * 2019-09-25 2022-04-21 Nobelpharma Co., Ltd. Granule having masked unpleasant taste and method for producing same

Also Published As

Publication number Publication date
EP4035733A1 (en) 2022-08-03
CN114340601A (zh) 2022-04-12
TWI865615B (zh) 2024-12-11
JPWO2021060304A1 (ja) 2021-10-07
CA3153004A1 (en) 2021-04-01
JP6905781B1 (ja) 2021-07-21
WO2021060304A1 (ja) 2021-04-01
TW202128143A (zh) 2021-08-01
JP2025107467A (ja) 2025-07-17
US20230016901A1 (en) 2023-01-19
EP4035733A4 (en) 2024-01-10
JP2021138775A (ja) 2021-09-16
JP7715378B2 (ja) 2025-07-30

Similar Documents

Publication Publication Date Title
CA2539982C (en) Pantoprazole multiparticulate formulations
JP2000281564A (ja) 医薬製剤
JPH0237327B2 (https=)
EP3981390B1 (en) Lacosamide pharmaceutical composition and pharmaceutical preparation thereof
JP2025107467A (ja) 不快な味がマスクされた顆粒剤及びその製造方法
CN105982858A (zh) 一种阿奇霉素掩味的干混悬颗粒剂及其制备方法
BRPI0621397A2 (pt) tabletes de liberação prolongada de metoprolol succinato e seus processos de preparação
CA2823622C (en) Solid molecular dispersion of fesoterodine
JP3833314B2 (ja) 発泡性組成物およびその製造方法
CN103096880B (zh) 不愉快味道被掩蔽的含药膜包覆的颗粒
CN101754754B (zh) 含有包覆的含药物的颗粒的可分散药片及其制备方法
CN105919943A (zh) 一种盐酸可乐定控释颗粒及其制备方法
JPWO2002034268A1 (ja) ５−アセチル−４，６−ジメチル−２−［２−［４−（２−メトキシフェニル）ピペラジニル］エチルアミノ］ピリミジン・三塩酸塩を有効成分として含有する徐放性製剤
HK40068436A (en) Granule having masked unpleasant taste and method for producing same
JPH04103525A (ja) 難水溶性薬物の持続性製剤化方法
JPH09169645A (ja) イブジラスト含有持続性製剤およびその製法
KR20040079325A (ko) 메트포르민 및 글리부라이드의 고형 경구용 제형 및 이의제조 방법
JP2008050324A (ja) 苦味遮蔽組成物。
CN110664779A (zh) 一种头孢呋辛酯颗粒及其制备方法
JPH05163163A (ja) 有核製剤
HK1086766B (en) Pantoprazole multiparticulate formulations
JPH05271176A (ja) ４−エチル−２−ヒドロキシイミノ−５−ニトロ−３−ヘキセンアミドの安定化剤