AU2017342156B2 - 1,3 di-substituted cyclobutane or azetidine derivatives as hematopoietic prostaglandin D synthase inhibitors - Google Patents

1,3 di-substituted cyclobutane or azetidine derivatives as hematopoietic prostaglandin D synthase inhibitors Download PDF

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Publication number
AU2017342156B2
AU2017342156B2 AU2017342156A AU2017342156A AU2017342156B2 AU 2017342156 B2 AU2017342156 B2 AU 2017342156B2 AU 2017342156 A AU2017342156 A AU 2017342156A AU 2017342156 A AU2017342156 A AU 2017342156A AU 2017342156 B2 AU2017342156 B2 AU 2017342156B2
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trans
muscle
mmol
substituted
thiazol
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AU2017342156A1 (en
Inventor
David Norman Deaton
Yu Guo
Ashley Paul Hancock
Christie SCHULTE
Barry George Shearer
Emilie Despagnet Smith
Eugene L. Stewart
Stephen Andrew Thomson
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GlaxoSmithKline Intellectual Property Development Ltd
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GlaxoSmithKline Intellectual Property Development Ltd
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    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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AU2017342156A 2016-10-13 2017-10-12 1,3 di-substituted cyclobutane or azetidine derivatives as hematopoietic prostaglandin D synthase inhibitors Ceased AU2017342156B2 (en)

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US201662407634P 2016-10-13 2016-10-13
US62/407,634 2016-10-13
PCT/IB2017/056320 WO2018069863A1 (en) 2016-10-13 2017-10-12 1,3 di-substituted cyclobutane or azetidine derivatives as hematopoietic prostaglandin d synthase inhibitors

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AU2017342156B2 true AU2017342156B2 (en) 2020-10-22

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EP (1) EP3526206A1 (OSRAM)
JP (1) JP6938628B2 (OSRAM)
KR (1) KR20190072565A (OSRAM)
CN (1) CN110072857A (OSRAM)
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AU (1) AU2017342156B2 (OSRAM)
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CA (1) CA3038756A1 (OSRAM)
CL (1) CL2019000986A1 (OSRAM)
CO (1) CO2019003482A2 (OSRAM)
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DO (1) DOP2019000087A (OSRAM)
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JOP20190072A1 (ar) 2016-10-13 2019-04-07 Glaxosmithkline Ip Dev Ltd مشتقات 1، 3 سيكلوبوتان ثنائي الاستبدال أو آزيتيدين كمثبطات للإنزيم المخلق للبروستاجلاندين d المكون للدم
EP3638672A1 (en) * 2017-06-13 2020-04-22 GlaxoSmithKline Intellectual Property Development Limited Chemical compounds as h-pgds inhibitors
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