AU2016335287A1

AU2016335287A1 - Pharmaceutical formulations for the oral delivery of peptide drugs

Pharmaceutical formulations for the oral delivery of peptide drugs Download PDF

Info

Publication number: AU2016335287A1
Authority: AU; Australia
Prior art keywords: complex; salt; iron; sodium; copper
Prior art date: 2015-10-07
Legal status : Abandoned

Application number

AU2016335287A

Other languages

English (en)

Inventor

Florian Foger

Martin Werle

Current Assignee

Cyprumed GmbH

Original Assignee

Cyprumed GmbH

Priority date

2015-10-07

Filing date

2016-10-07

Publication date

2018-04-12

2016-10-07 Application filed by Cyprumed GmbH filed Critical Cyprumed GmbH

2018-04-12 Publication of AU2016335287A1 publication Critical patent/AU2016335287A1/en

Status Abandoned legal-status Critical Current

Links

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-1 copper salt Chemical class 0.000 claims abstract description 450
XEEYBQQBJWHFJM-UHFFFAOYSA-N iron Substances [Fe] XEEYBQQBJWHFJM-UHFFFAOYSA-N 0.000 claims abstract description 335
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239000010949 copper Substances 0.000 claims abstract description 175
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239000008139 complexing agent Substances 0.000 claims abstract description 128
239000011701 zinc Substances 0.000 claims abstract description 126
229910052725 zinc Inorganic materials 0.000 claims abstract description 126
239000011734 sodium Substances 0.000 claims description 140
229910052708 sodium Inorganic materials 0.000 claims description 140
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HCHKCACWOHOZIP-UHFFFAOYSA-N zinc Drugs [Zn] HCHKCACWOHOZIP-UHFFFAOYSA-N 0.000 claims description 137
DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 claims description 129
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