AU2012318580A1 - Novel quinoxaline inhibitors of PI3K - Google Patents

Novel quinoxaline inhibitors of PI3K Download PDF

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Publication number
AU2012318580A1
AU2012318580A1 AU2012318580A AU2012318580A AU2012318580A1 AU 2012318580 A1 AU2012318580 A1 AU 2012318580A1 AU 2012318580 A AU2012318580 A AU 2012318580A AU 2012318580 A AU2012318580 A AU 2012318580A AU 2012318580 A1 AU2012318580 A1 AU 2012318580A1
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Jerry B. Evarts
Thomas Judge
Edward A. Kesicki
Kamal D. Puri
Roger G. Ulrich
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Gilead Calistoga LLC
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Gilead Calistoga LLC
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine
    • AHUMAN NECESSITIES
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/24Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one nitrogen and one sulfur atom

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  • Health & Medical Sciences (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Rheumatology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2012318580A 2011-10-04 2012-10-04 Novel quinoxaline inhibitors of PI3K Abandoned AU2012318580A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161543176P 2011-10-04 2011-10-04
US61/543,176 2011-10-04
PCT/US2012/058800 WO2013052699A2 (en) 2011-10-04 2012-10-04 Novel quinoxaline inhibitors of pi3k

Publications (1)

Publication Number Publication Date
AU2012318580A1 true AU2012318580A1 (en) 2014-05-22

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AU2012318580A Abandoned AU2012318580A1 (en) 2011-10-04 2012-10-04 Novel quinoxaline inhibitors of PI3K

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US (1) US20140235643A1 (enExample)
EP (1) EP2763994A4 (enExample)
JP (1) JP2014528451A (enExample)
CN (1) CN104024257A (enExample)
AU (1) AU2012318580A1 (enExample)
CA (1) CA2850763A1 (enExample)
HK (1) HK1201065A1 (enExample)
WO (1) WO2013052699A2 (enExample)

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