AU2007309237B2 - Triazolo-pyridazine protein kinase modulators - Google Patents

Triazolo-pyridazine protein kinase modulators Download PDF

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Publication number
AU2007309237B2
AU2007309237B2 AU2007309237A AU2007309237A AU2007309237B2 AU 2007309237 B2 AU2007309237 B2 AU 2007309237B2 AU 2007309237 A AU2007309237 A AU 2007309237A AU 2007309237 A AU2007309237 A AU 2007309237A AU 2007309237 B2 AU2007309237 B2 AU 2007309237B2
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AU
Australia
Prior art keywords
substituted
unsubstituted
alkyl
compounds
pyridinyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2007309237A
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English (en)
Other versions
AU2007309237A1 (en
Inventor
Pierre-Yves Bounaud
Elizabeth Anne Jefferson
Patrick S. Lee
Christopher Ronald Smith
Eduardo Torres
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SGX Pharmaceuticals Inc
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SGX Pharmaceuticals Inc
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Publication of AU2007309237A1 publication Critical patent/AU2007309237A1/en
Application granted granted Critical
Publication of AU2007309237B2 publication Critical patent/AU2007309237B2/en
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AU2007309237A 2006-10-23 2007-10-18 Triazolo-pyridazine protein kinase modulators Ceased AU2007309237B2 (en)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US86255206P 2006-10-23 2006-10-23
US60/862,552 2006-10-23
US87138406P 2006-12-21 2006-12-21
US60/871,384 2006-12-21
US91375207P 2007-04-24 2007-04-24
US60/913,752 2007-04-24
US95283307P 2007-07-30 2007-07-30
US60/952,833 2007-07-30
PCT/US2007/081832 WO2008051805A2 (en) 2006-10-23 2007-10-18 Triazolo-pyridazine protein kinase modulators

Publications (2)

Publication Number Publication Date
AU2007309237A1 AU2007309237A1 (en) 2008-05-02
AU2007309237B2 true AU2007309237B2 (en) 2012-03-22

Family

ID=39031065

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2007309237A Ceased AU2007309237B2 (en) 2006-10-23 2007-10-18 Triazolo-pyridazine protein kinase modulators

Country Status (16)

Country Link
US (1) US8071581B2 (enExample)
EP (1) EP2081937B1 (enExample)
JP (1) JP2010507577A (enExample)
KR (1) KR101083177B1 (enExample)
AU (1) AU2007309237B2 (enExample)
BR (1) BRPI0717317A2 (enExample)
CA (1) CA2667453A1 (enExample)
DK (1) DK2081937T3 (enExample)
EA (1) EA016527B1 (enExample)
ES (1) ES2393132T3 (enExample)
MX (1) MX2009004060A (enExample)
PE (1) PE20081256A1 (enExample)
PL (1) PL2081937T3 (enExample)
PT (1) PT2081937E (enExample)
TW (1) TW200833692A (enExample)
WO (1) WO2008051805A2 (enExample)

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Also Published As

Publication number Publication date
PE20081256A1 (es) 2008-10-13
PL2081937T3 (pl) 2013-01-31
JP2010507577A (ja) 2010-03-11
US8071581B2 (en) 2011-12-06
CA2667453A1 (en) 2008-05-02
EP2081937A2 (en) 2009-07-29
MX2009004060A (es) 2009-06-19
WO2008051805A2 (en) 2008-05-02
PT2081937E (pt) 2012-10-15
KR20090069303A (ko) 2009-06-30
BRPI0717317A2 (pt) 2013-10-22
KR101083177B1 (ko) 2011-11-11
WO2008051805A3 (en) 2008-07-10
US20100120739A1 (en) 2010-05-13
EA016527B1 (ru) 2012-05-30
EA200970402A1 (ru) 2009-10-30
ES2393132T3 (es) 2012-12-18
EP2081937B1 (en) 2012-09-12
TW200833692A (en) 2008-08-16
AU2007309237A1 (en) 2008-05-02
DK2081937T3 (da) 2012-10-01

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