|
MX2008012945A
(es)
|
2006-04-07 |
2009-01-15 |
Vertex Pharma |
Moduladores de transportadores de cartucho de union a adenosina-trifosfato celular (atp).
|
|
US7645789B2
(en)
|
2006-04-07 |
2010-01-12 |
Vertex Pharmaceuticals Incorporated |
Indole derivatives as CFTR modulators
|
|
USRE50453E1
(en)
|
2006-04-07 |
2025-06-10 |
Vertex Pharmaceuticals Incorporated |
Indole derivatives as CFTR modulators
|
|
US10022352B2
(en)
|
2006-04-07 |
2018-07-17 |
Vertex Pharmaceuticals Incorporated |
Modulators of ATP-binding cassette transporters
|
|
US8217177B2
(en)
|
2006-07-14 |
2012-07-10 |
Amgen Inc. |
Fused heterocyclic derivatives and methods of use
|
|
PE20121506A1
(es)
|
2006-07-14 |
2012-11-26 |
Amgen Inc |
Compuestos triazolopiridinas como inhibidores de c-met
|
|
US8198448B2
(en)
|
2006-07-14 |
2012-06-12 |
Amgen Inc. |
Fused heterocyclic derivatives and methods of use
|
|
WO2008021781A1
(en)
|
2006-08-07 |
2008-02-21 |
Incyte Corporation |
Triazolotriazines as kinase inhibitors
|
|
US8563573B2
(en)
|
2007-11-02 |
2013-10-22 |
Vertex Pharmaceuticals Incorporated |
Azaindole derivatives as CFTR modulators
|
|
CA2669991C
(en)
|
2006-11-22 |
2016-01-26 |
Incyte Corporation |
Imidazotriazines and imidazopyrimidines as kinase inhibitors
|
|
KR20100128305A
(ko)
|
2008-02-28 |
2010-12-07 |
노파르티스 아게 |
C-met 티로신 키나제 매개 질환의 치료를 위한 이미다조[1,2-b]피리다진 유도체
|
|
CA2724742C
(en)
*
|
2008-05-21 |
2016-07-19 |
Incyte Corporation |
Salts of 2-fluoro-n-methyl-4-[7-(quinolin-6-yl-methyl)- imidazo[1,2-b][1,2,4]triazin-2-yl]benzamide and processes related to preparing the same
|
|
DE102008028905A1
(de)
*
|
2008-06-18 |
2009-12-24 |
Merck Patent Gmbh |
3-(3-Pyrimidin-2-yl-benzyl)-[1,2,4]triazolo[4,3-b]pyridazinderivate
|
|
DE102008037790A1
(de)
|
2008-08-14 |
2010-02-18 |
Merck Patent Gmbh |
Bicyclische Triazolderivate
|
|
DE102008038221A1
(de)
|
2008-08-18 |
2010-02-25 |
Merck Patent Gmbh |
7-Azaindolderivate
|
|
DE102008038222A1
(de)
|
2008-08-18 |
2010-02-25 |
Merck Patent Gmbh |
Indazol-5-carbonsäurehydrazid-derivate
|
|
DE102008038220A1
(de)
|
2008-08-18 |
2010-02-25 |
Merck Patent Gmbh |
Oxadiazolderivate
|
|
EP2356116A1
(en)
*
|
2008-11-20 |
2011-08-17 |
OSI Pharmaceuticals, Inc. |
Substituted pyrroloý2,3-b¨-pyridines and-pyrazines
|
|
CA2744563A1
(en)
*
|
2008-12-12 |
2010-06-17 |
Ariad Pharmaceuticals, Inc. |
Azaindole derivatives as kinase inhibitors
|
|
DE102008063667A1
(de)
*
|
2008-12-18 |
2010-07-01 |
Merck Patent Gmbh |
3-(3-Pyrimidin-2-yl-benzyl)-°[1,2,4]triazolo[4,3-b]pyrimidin-derivate
|
|
DE102008062825A1
(de)
|
2008-12-23 |
2010-06-24 |
Merck Patent Gmbh |
3-(3-Pyrimidin-2-yl-benzyl)-[1,2,4]triazolo [4,3-b]pyridazin-derivate
|
|
SG172986A1
(en)
*
|
2009-02-10 |
2011-08-29 |
Astrazeneca Ab |
Triazolo [4,3-b] pyridazine derivatives and their uses for prostate cancer
|
|
EP2406264A4
(en)
|
2009-03-09 |
2012-08-08 |
Univ California |
SUBSTITUTED HETEROCYCLES AND THEIR USE AS ALLOSTERIC MODULATORS OF NICOTINE AND GABAA RECEPTORS
|
|
US8389526B2
(en)
|
2009-08-07 |
2013-03-05 |
Novartis Ag |
3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
|
|
EA201200260A1
(ru)
|
2009-08-12 |
2012-09-28 |
Новартис Аг |
Гетероциклические гидразоны и их применение для лечения рака и воспаления
|
|
KR20120089463A
(ko)
|
2009-08-20 |
2012-08-10 |
노파르티스 아게 |
헤테로시클릭 옥심 화합물
|
|
BR112012016129B1
(pt)
*
|
2009-12-31 |
2020-11-03 |
Hutchison Medipharma Limited |
composto, composição e uso dos ditos compostos
|
|
ES2608329T3
(es)
|
2010-02-03 |
2017-04-07 |
Incyte Holdings Corporation |
Imidazo[1,2-b][1,2,4]triazinas como inhibidores de c-Met
|
|
US8802868B2
(en)
|
2010-03-25 |
2014-08-12 |
Vertex Pharmaceuticals Incorporated |
Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide
|
|
MX342288B
(es)
|
2010-04-22 |
2016-09-23 |
Vertex Pharma |
Proceso para producir compuestos de cicloalquilcarboxamido-indol.
|
|
AR081039A1
(es)
|
2010-05-14 |
2012-05-30 |
Osi Pharmaceuticals Llc |
Inhibidores biciclicos fusionados de quinasa
|
|
EP2569315A1
(en)
|
2010-05-14 |
2013-03-20 |
OSI Pharmaceuticals, LLC |
Fused bicyclic kinase inhibitors
|
|
JP5960688B2
(ja)
|
2010-05-17 |
2016-08-02 |
インコゼン セラピューティクス プライベート リミテッド |
プロテインキナーゼ調節物質としての新規3,5−二置換−3h−[1,2,3]トリアゾロ[4,5−b]ピリジン化合物
|
|
US10414760B2
(en)
|
2016-11-29 |
2019-09-17 |
Angion Biomedica Corp. |
Cytochrome P450 inhibitors and uses thereof
|
|
WO2011153192A2
(en)
*
|
2010-06-01 |
2011-12-08 |
Angion Biomedica Corp. |
Cytochrome p450 inhibitors and uses thereof
|
|
AR085183A1
(es)
|
2010-07-30 |
2013-09-18 |
Lilly Co Eli |
Compuesto 6-(1-metil-1h-pirazol-4-il)-3-(2-metil-2h-indazol-5-iltio)-[1,2,4]triazol[4,3-b]piridazina, composicion farmaceutica que lo comprende y uso para preparar un medicamento util para tratar cancer
|
|
US20130324526A1
(en)
|
2011-02-10 |
2013-12-05 |
Novartis Ag |
[1,2,4] triazolo [4,3-b] pyridazine compounds as inhibitors of the c-met tyrosine kinase
|
|
EP2710003A1
(en)
|
2011-05-16 |
2014-03-26 |
OSI Pharmaceuticals, LLC |
Fused bicyclic kinase inhibitors
|
|
AU2012310168B2
(en)
|
2011-09-15 |
2015-07-16 |
Novartis Ag |
6 - substituted 3 - (quinolin- 6 - ylthio) - [1,2,4] triazolo [4, 3 -a] pyradines as tyrosine kinase
|
|
CA2848518C
(en)
|
2011-09-27 |
2019-06-18 |
Genfit |
Derivatives of 6-substituted triazolopyridazines as rev-erb agonists
|
|
KR101869534B1
(ko)
*
|
2012-03-05 |
2018-06-20 |
한국화학연구원 |
신규한 트리아졸로 피리다진 유도체 및 그의 용도
|
|
BR112014024251A8
(pt)
|
2012-03-30 |
2018-01-23 |
Rhizen Pharmaceuticals S A |
novos compostos piridina 3,5-dissubstituída-3h-imidazo [4,5-b] e piridina 3,5-dissubstituída -3h-[1,2,3]triazolo[4,5-b] como moduladores de quinases de proteína c-met
|
|
US9012496B2
(en)
|
2012-07-16 |
2015-04-21 |
Vertex Pharmaceuticals Incorporated |
Pharmaceutical compositions of (R)-1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide and administration thereof
|
|
CN103122000B
(zh)
*
|
2012-09-03 |
2013-12-25 |
中美冠科生物技术(太仓)有限公司 |
用作抗肿瘤药物的高选择性的c-Met激酶抑制剂
|
|
ME02794B
(me)
|
2012-10-16 |
2018-01-20 |
Janssen Pharmaceutica Nv |
Metilen vezani hinolinil modulatori ror-gama-t
|
|
AU2013331493A1
(en)
|
2012-10-16 |
2015-04-09 |
Janssen Pharmaceutica Nv |
Heteroaryl linked quinolinyl modulators of RORyt
|
|
EP2909193B1
(en)
|
2012-10-16 |
2017-04-19 |
Janssen Pharmaceutica NV |
Phenyl linked quinolinyl modulators of ror-gamma-t
|
|
US9846345B2
(en)
|
2013-02-28 |
2017-12-19 |
Empire Technology Development Llc |
Colored pigment particles for electrophoretic displays
|
|
BR112015020716A2
(pt)
*
|
2013-03-13 |
2017-07-18 |
Hoffmann La Roche |
processo para a preparação de (2-(4-(2-(1-isopropil-3-metil-1h-1,2,4-triazol-5-il)-5,6-diidrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-il)-1h-pirazol-1-il)-2-metilpropanamida (i) e composto
|
|
US20140303121A1
(en)
*
|
2013-03-15 |
2014-10-09 |
Plexxikon Inc. |
Heterocyclic compounds and uses thereof
|
|
NZ630875A
(en)
*
|
2013-03-15 |
2017-12-22 |
Plexxikon Inc |
Heterocyclic compounds and uses thereof
|
|
AU2014334619A1
(en)
|
2013-10-15 |
2016-04-21 |
Janssen Pharmaceutica Nv |
Alkyl linked quinolinyl modulators of RORyt
|
|
US9328095B2
(en)
|
2013-10-15 |
2016-05-03 |
Janssen Pharmaceutica Nv |
Heteroaryl linked quinolinyl modulators of RORgammat
|
|
US9221804B2
(en)
|
2013-10-15 |
2015-12-29 |
Janssen Pharmaceutica Nv |
Secondary alcohol quinolinyl modulators of RORγt
|
|
US10555941B2
(en)
|
2013-10-15 |
2020-02-11 |
Janssen Pharmaceutica Nv |
Alkyl linked quinolinyl modulators of RORγt
|
|
EP3057422B1
(en)
|
2013-10-15 |
2019-05-15 |
Janssen Pharmaceutica NV |
Quinolinyl modulators of ror(gamma)t
|
|
US9284308B2
(en)
|
2013-10-15 |
2016-03-15 |
Janssen Pharmaceutica Nv |
Methylene linked quinolinyl modulators of RORγt
|
|
US9403816B2
(en)
|
2013-10-15 |
2016-08-02 |
Janssen Pharmaceutica Nv |
Phenyl linked quinolinyl modulators of RORγt
|
|
GB201321745D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
|
WO2015134854A2
(en)
*
|
2014-03-06 |
2015-09-11 |
Oyagen, Inc. |
Small molecule vif dimerization antagonists as anti-hiv agents and for use as hiv/aids therapeutics
|
|
KR102447581B1
(ko)
|
2014-04-15 |
2022-09-28 |
버텍스 파마슈티칼스 인코포레이티드 |
낭포성 섬유증 막전도 조절자 매개 질환 치료용 약제학적 조성물
|
|
JP6578349B2
(ja)
|
2014-08-11 |
2019-09-18 |
アンジオン バイオメディカ コーポレーション |
チトクロームp450阻害剤およびその使用
|
|
CN107531631B
(zh)
|
2014-12-31 |
2021-09-03 |
安吉昂生物医药公司 |
用于治疗疾病的方法和药剂
|
|
HUE053903T2
(hu)
*
|
2015-04-13 |
2021-07-28 |
Five Prime Therapeutics Inc |
Kombinációs terápia rák ellen
|
|
CR20180109A
(es)
|
2015-07-20 |
2018-05-03 |
Genzyme Corp |
Inhibidores de receptor del factor estimulador de colonias 1 (csf-1r)
|
|
AU2018348241B2
(en)
|
2017-10-13 |
2023-01-12 |
Opna Bio SA |
Solid forms of a compound for modulating kinases
|
|
GB201905721D0
(en)
|
2019-04-24 |
2019-06-05 |
Univ Dundee |
Compounds
|
|
CN113861198B
(zh)
*
|
2020-06-30 |
2024-08-02 |
上海医药集团股份有限公司 |
咪唑并[4,5-b]吡嗪类化合物、其制备方法及应用
|
|
EP4267573A1
(en)
|
2020-12-23 |
2023-11-01 |
Genzyme Corporation |
Deuterated colony stimulating factor-1 receptor (csf-1r) inhibitors
|