AU2006224842B2 - The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases - Google Patents
The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases Download PDFInfo
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- AU2006224842B2 AU2006224842B2 AU2006224842A AU2006224842A AU2006224842B2 AU 2006224842 B2 AU2006224842 B2 AU 2006224842B2 AU 2006224842 A AU2006224842 A AU 2006224842A AU 2006224842 A AU2006224842 A AU 2006224842A AU 2006224842 B2 AU2006224842 B2 AU 2006224842B2
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- glycopyrrolate
- pharmaceutical
- montelukast
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- combination
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Medicinal Preparation (AREA)
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| US20050048614A1 (en) * | 2000-06-13 | 2005-03-03 | Children's Medical Center Corporation | Biosynthetic oncolytic molecules and uses therefor |
| DE602004016002D1 (de) * | 2003-07-28 | 2008-10-02 | Janssen Pharmaceutica Nv | Benzimidazol-, benzothiazol- und benzoxazolderivate und deren verwendung als lta4h-modulatoren |
| ES2614090T3 (es) | 2005-12-29 | 2017-05-29 | Celtaxsys, Inc. | Derivados de diamina como inhibidores de leucotrieno A4 hidrolasa |
| TW200906396A (en) * | 2007-02-14 | 2009-02-16 | Janssen Pharmaceutica Nv | LTA4H modulators and uses thereof |
| EP2200550B1 (en) | 2007-10-18 | 2018-04-18 | Rose U, LLC | Topical glycopyrrolate formulations |
| AU2008316283A1 (en) * | 2007-10-25 | 2009-04-30 | Merck Frosst Canada Ltd | Inhalation compositions comprising montelukast acid and a PDE-4 inhibitor or an inhaled corticosteroid |
| CA2764867C (en) * | 2009-06-09 | 2016-05-17 | Elevation Pharmaceuticals, Inc. | Treatment of chronic obstructive pulmonary disease with nebulized beta 2-agonist or combined nebulized beta 2-agonist and anticholinergic administration |
| US9378456B2 (en) * | 2012-11-19 | 2016-06-28 | Microsoft Technology Licensing, Llc | Task completion |
| US9006462B2 (en) | 2013-02-28 | 2015-04-14 | Dermira, Inc. | Glycopyrrolate salts |
| EP2961734B1 (en) | 2013-02-28 | 2018-09-26 | Dermira, Inc. | Glycopyrrolate salts |
| US8558008B2 (en) | 2013-02-28 | 2013-10-15 | Dermira, Inc. | Crystalline glycopyrrolate tosylate |
| WO2014164658A1 (en) * | 2013-03-12 | 2014-10-09 | Celtaxsys, Inc. | Methods of inhibiting leukotriene a4 hydrolase |
| KR20150127245A (ko) | 2013-03-14 | 2015-11-16 | 켈탁시스, 인코퍼레이티드 | 류코트라이엔 a4 가수분해효소의 저해제 |
| SG10202000496XA (en) * | 2014-01-10 | 2020-03-30 | Afimmune Ltd | Pharmaceutical compositions comprising 15-hepe and methods of treating asthma and lung disorders using same |
| CA3102077A1 (en) | 2018-05-31 | 2019-12-05 | Sanjeev AHUJA | Method of reducing pulmonary exacerbations in respiratory disease patients |
| TW202042813A (zh) * | 2019-01-10 | 2020-12-01 | 大陸商江陰貝瑞森製藥有限公司 | 含有白三烯受體拮抗劑的新穎調配物 |
| AU2021215849B2 (en) * | 2020-02-03 | 2023-08-03 | Taro Pharmaceutical Industries Ltd. | Topical montelukast formulations |
| CN115792229B (zh) * | 2022-01-28 | 2024-06-18 | 华中科技大学同济医学院附属同济医院 | 鼻分泌物中tPA在制备鼻息肉及其预后检测剂中的应用 |
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| CZ290266B6 (cs) * | 1993-07-02 | 2002-06-12 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituované benzamidy, způsob jejich výroby a farmaceutické prostředky s jejich obsahem |
| EP0932401A1 (en) | 1996-07-01 | 1999-08-04 | Sepracor, Inc. | Methods and compositions for treating urinary incontinence using enantiomerically enriched (r,r)-glycopyrrolate |
| DK0937041T3 (da) * | 1996-11-11 | 2003-08-11 | Christian R Noe | Anvendelse af et farmaceutisk egnet salt af (3R,2'R)-3-[(cyclopentil-hydroxyphenylacetyl)oxyl]-1,1-dimethyl-pyrrolidinium til fremstilling af et lægemiddel |
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| AU7455498A (en) * | 1998-05-29 | 1999-12-20 | Citizen Watch Co. Ltd. | Method of subjecting ink jet printer to preuse treatment |
| DK1102579T3 (da) * | 1998-08-04 | 2003-07-14 | Jago Res Ag | Medicinske aerosolformuleringer |
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| DE19921693A1 (de) * | 1999-05-12 | 2000-11-16 | Boehringer Ingelheim Pharma | Neuartige Arzneimittelkompositionen auf der Basis von anticholinergisch wirksamen Verbindungen und ß-Mimetika |
| US6086914A (en) * | 1999-03-12 | 2000-07-11 | Weinstein; Robert E. | Nonsedating formulations for allergic rhinitis which possess antihistaminic and anticholinergic activity |
| US20040002548A1 (en) * | 1999-05-12 | 2004-01-01 | Boehringer Ingelheim Pharma Kg | Medicament compositions containing anticholinergically-effective compounds and betamimetics |
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| GB0008660D0 (en) | 2000-04-07 | 2000-05-31 | Arakis Ltd | The treatment of respiratory diseases |
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| AU2002221741B2 (en) * | 2000-10-31 | 2007-04-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Inhalative solution formulation containing a tiotropium salt |
| DE10110772A1 (de) | 2001-03-07 | 2002-09-12 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren |
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| DE50211045D1 (de) | 2001-03-30 | 2007-11-22 | Jagotec Ag | Medizinische aerosolformulierungen |
| US6667344B2 (en) * | 2001-04-17 | 2003-12-23 | Dey, L.P. | Bronchodilating compositions and methods |
| JP2004530705A (ja) | 2001-05-25 | 2004-10-07 | ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | 閉塞性気道疾患及びその他の炎症性疾患を治療するためのｐｄｅ４インヒビター及びチオトロピウム又はその誘導体の組み合わせ |
| OA12610A (en) | 2001-05-25 | 2006-06-09 | Pfizer | A PDE 4 inhbitor and an anti-cholinergic agent in combination for treating obstructive airways diseases. |
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| WO2005055999A1 (ja) | 2003-12-08 | 2005-06-23 | Nippon Shinyaku Co., Ltd. | 抗コリン作用剤 |
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Patent Citations (1)
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|---|---|---|---|---|
| AU2005244439A1 (en) * | 2004-05-18 | 2005-11-24 | Novartis Ag | Combinations of glycopyrrolate and beta2 adrenoceptor agonists |
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| Tzelepis et al. European Respiratory Journal (1996) vol. 9, no. 8, pages 100-103 * |
Also Published As
| Publication number | Publication date |
|---|---|
| CY1117571T1 (el) | 2017-04-26 |
| MX2007011273A (es) | 2007-11-08 |
| JP4991693B2 (ja) | 2012-08-01 |
| CN101128196A (zh) | 2008-02-20 |
| US8268864B2 (en) | 2012-09-18 |
| ES2570332T3 (es) | 2016-05-17 |
| CA2595791A1 (en) | 2006-09-21 |
| WO2006097250A1 (en) | 2006-09-21 |
| EP1863476B1 (en) | 2016-02-03 |
| CA2595791C (en) | 2013-10-08 |
| DK1863476T3 (en) | 2016-05-17 |
| US20060211729A1 (en) | 2006-09-21 |
| SI1863476T1 (sl) | 2016-05-31 |
| RU2007138270A (ru) | 2009-04-27 |
| HRP20160373T1 (hr) | 2016-05-06 |
| NO340405B1 (no) | 2017-04-18 |
| AU2006224842A1 (en) | 2006-09-21 |
| HUE027076T2 (en) | 2016-08-29 |
| NO20075287L (no) | 2007-12-05 |
| RU2420285C2 (ru) | 2011-06-10 |
| JP2008533072A (ja) | 2008-08-21 |
| HK1114013A1 (en) | 2008-10-24 |
| CN101128196B (zh) | 2013-01-02 |
| EP1863476A1 (en) | 2007-12-12 |
| PL1863476T3 (pl) | 2016-07-29 |
| NZ560206A (en) | 2009-09-25 |
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| DA3 | Amendments made section 104 |
Free format text: THE NATURE OF THE AMENDMENT IS: AMEND THE INVENTION TITLE TO READ THE COMBINATION OF ANTICHOLINERGICS AND LEUKOTRIENE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY DISEASES |
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| FGA | Letters patent sealed or granted (standard patent) | ||
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |