AU2006224842B2 - The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases - Google Patents
The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases Download PDFInfo
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- AU2006224842B2 AU2006224842B2 AU2006224842A AU2006224842A AU2006224842B2 AU 2006224842 B2 AU2006224842 B2 AU 2006224842B2 AU 2006224842 A AU2006224842 A AU 2006224842A AU 2006224842 A AU2006224842 A AU 2006224842A AU 2006224842 B2 AU2006224842 B2 AU 2006224842B2
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- glycopyrrolate
- pharmaceutical
- montelukast
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- combination
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
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- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Chemical Kinetics & Catalysis (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US20050048614A1 (en) * | 2000-06-13 | 2005-03-03 | Children's Medical Center Corporation | Biosynthetic oncolytic molecules and uses therefor |
| AU2004261610B2 (en) * | 2003-07-28 | 2010-05-20 | Janssen Pharmaceutica N.V. | Benzimidazole, benzthiazole and benzoxazole derivatives and their use as LTA4H modulators |
| US7737145B2 (en) | 2005-12-29 | 2010-06-15 | Estrellita Pharmaceuticals, Llc | Diamine derivatives as inhibitors of leukotriene A4 hydrolase |
| CL2008000468A1 (es) * | 2007-02-14 | 2008-08-22 | Janssen Pharmaceutica Nv | Uso de compuestos derivados de heterociclos, inhibidores de leucotrina a4 hidrolasa (lta4h), utiles para tratar o prevenir la dermatitis, acne, infarto al miocardio, dolor, picazon, gingivitis, cancer, artritis, entre otras. |
| US8618160B2 (en) * | 2007-10-18 | 2013-12-31 | Rose U | Topical glycopyrrolate formulations |
| KR20100072295A (ko) * | 2007-10-25 | 2010-06-30 | 머크 프로스트 캐나다 리미티드 | 병용 요법 |
| AU2010258751A1 (en) * | 2009-06-09 | 2012-02-02 | Sunovion Respiratory Development Inc. | Treatment of chronic obstructive pulmonary disease with nebulized beta 2-agonist or combined nebulized beta 2-agonist and anticholinergic administration |
| US9378456B2 (en) * | 2012-11-19 | 2016-06-28 | Microsoft Technology Licensing, Llc | Task completion |
| US8558008B2 (en) | 2013-02-28 | 2013-10-15 | Dermira, Inc. | Crystalline glycopyrrolate tosylate |
| US9006462B2 (en) | 2013-02-28 | 2015-04-14 | Dermira, Inc. | Glycopyrrolate salts |
| JP6114841B2 (ja) | 2013-02-28 | 2017-04-12 | ダーミラ， インク．Ｄｅｒｍｉｒａ， Ｉｎｃ． | グリコピロレート塩 |
| CA2905340C (en) | 2013-03-12 | 2022-05-31 | Celtaxsys, Inc. | Low dose oral formulations of acebilustat |
| MX2015011677A (es) | 2013-03-14 | 2016-07-08 | Celtaxsys Inc | Inhibidores de leucotrieno a4 hidrolasa. |
| MX2016008953A (es) * | 2014-01-10 | 2017-02-02 | Dignity Sciences Ltd | Composiciones farmaceuticas que comprenden i5-hidroxi-eicosa- 5,8,11,13,17-pentaenoico ( 15-hepe ) y metodos para tratar el asma y trastornos pulmonares que usan las mismas. |
| WO2019232306A1 (en) | 2018-05-31 | 2019-12-05 | Celtaxsys, Inc. | Method of reducing pulmonary exacerbations in respiratory disease patients |
| KR20210114962A (ko) * | 2019-01-10 | 2021-09-24 | 장인 무코케어 파마슈티컬 컴퍼니 리미티드 | 류코트리엔 수용체 길항제를 함유하는 신규 제제 |
| BR112022015199A2 (pt) * | 2020-02-03 | 2022-10-11 | Taro Pharma Ind | Formulações tópicas de montelucaste |
| CN115792229B (zh) * | 2022-01-28 | 2024-06-18 | 华中科技大学同济医学院附属同济医院 | 鼻分泌物中tPA在制备鼻息肉及其预后检测剂中的应用 |
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| AU2005244439A1 (en) * | 2004-05-18 | 2005-11-24 | Novartis Ag | Combinations of glycopyrrolate and beta2 adrenoceptor agonists |
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| DE59709927D1 (de) * | 1996-11-11 | 2003-05-28 | Noe Christian | Verwendung eines pharmazeutisch geeigneten Salzes von (3R,2'R)-3-[(Cyclopentyl-hydroxyphenylacetyl)oxy]-1,1-dimethyl-pyrrolidinium zur Herstellung eines Arzneimittels |
| IL131492A0 (en) * | 1997-04-30 | 2001-01-28 | Warner Lambert Co | Topical nasal antiinflammatory compositions |
| US6384038B1 (en) * | 1998-04-14 | 2002-05-07 | Sepracor Inc. | Methods and compositions using cetirizine in combination with leukotriene inhibitors or decongestants |
| WO1999062720A1 (fr) * | 1998-05-29 | 1999-12-09 | Citizen Watch Co., Ltd. | Procede permettant de soumettre une imprimante a jet d'encre a un traitement de pre-utilisation |
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| DK1131059T3 (da) * | 1998-11-13 | 2003-06-30 | Jago Res Ag | Tørpulver til inhalation |
| US6086914A (en) * | 1999-03-12 | 2000-07-11 | Weinstein; Robert E. | Nonsedating formulations for allergic rhinitis which possess antihistaminic and anticholinergic activity |
| DE19921693A1 (de) * | 1999-05-12 | 2000-11-16 | Boehringer Ingelheim Pharma | Neuartige Arzneimittelkompositionen auf der Basis von anticholinergisch wirksamen Verbindungen und ß-Mimetika |
| US20040002548A1 (en) * | 1999-05-12 | 2004-01-01 | Boehringer Ingelheim Pharma Kg | Medicament compositions containing anticholinergically-effective compounds and betamimetics |
| SE9903995D0 (sv) * | 1999-11-03 | 1999-11-03 | Astra Ab | New combination |
| DE19961300A1 (de) * | 1999-12-18 | 2001-06-21 | Asta Medica Ag | Vorratssystem für Arzneimittel in Pulverform und damit ausgestatteter Inhalator |
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| DE10110772A1 (de) | 2001-03-07 | 2002-09-12 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren |
| GB0029903D0 (en) * | 2000-12-07 | 2001-01-24 | Arakis Ltd | Use of anti-muscarinic agents |
| DE50211045D1 (de) | 2001-03-30 | 2007-11-22 | Jagotec Ag | Medizinische aerosolformulierungen |
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| EP1452179A1 (en) * | 2003-02-27 | 2004-09-01 | CHIESI FARMACEUTICI S.p.A. | Novel medicament combination of a highly potent long-lasting beta2-agonist and a corticosteroid |
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| WO2005055999A1 (ja) | 2003-12-08 | 2005-06-23 | Nippon Shinyaku Co., Ltd. | 抗コリン作用剤 |
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2005244439A1 (en) * | 2004-05-18 | 2005-11-24 | Novartis Ag | Combinations of glycopyrrolate and beta2 adrenoceptor agonists |
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| Tzelepis et al. European Respiratory Journal (1996) vol. 9, no. 8, pages 100-103 * |
Also Published As
| Publication number | Publication date |
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| HRP20160373T1 (hr) | 2016-05-06 |
| CA2595791C (en) | 2013-10-08 |
| ES2570332T3 (es) | 2016-05-17 |
| HK1114013A1 (en) | 2008-10-24 |
| US20060211729A1 (en) | 2006-09-21 |
| CN101128196A (zh) | 2008-02-20 |
| SI1863476T1 (sl) | 2016-05-31 |
| EP1863476B1 (en) | 2016-02-03 |
| MX2007011273A (es) | 2007-11-08 |
| JP4991693B2 (ja) | 2012-08-01 |
| NO20075287L (no) | 2007-12-05 |
| PL1863476T3 (pl) | 2016-07-29 |
| HUE027076T2 (en) | 2016-08-29 |
| NZ560206A (en) | 2009-09-25 |
| CN101128196B (zh) | 2013-01-02 |
| RU2420285C2 (ru) | 2011-06-10 |
| CA2595791A1 (en) | 2006-09-21 |
| DK1863476T3 (en) | 2016-05-17 |
| NO340405B1 (no) | 2017-04-18 |
| AU2006224842A1 (en) | 2006-09-21 |
| JP2008533072A (ja) | 2008-08-21 |
| CY1117571T1 (el) | 2017-04-26 |
| EP1863476A1 (en) | 2007-12-12 |
| RU2007138270A (ru) | 2009-04-27 |
| WO2006097250A1 (en) | 2006-09-21 |
| US8268864B2 (en) | 2012-09-18 |
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Free format text: THE NATURE OF THE AMENDMENT IS: AMEND THE INVENTION TITLE TO READ THE COMBINATION OF ANTICHOLINERGICS AND LEUKOTRIENE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY DISEASES |
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| FGA | Letters patent sealed or granted (standard patent) | ||
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