AU2005270068B2 - C-Met modulators and method of use - Google Patents
C-Met modulators and method of use Download PDFInfo
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- AU2005270068B2 AU2005270068B2 AU2005270068A AU2005270068A AU2005270068B2 AU 2005270068 B2 AU2005270068 B2 AU 2005270068B2 AU 2005270068 A AU2005270068 A AU 2005270068A AU 2005270068 A AU2005270068 A AU 2005270068A AU 2005270068 B2 AU2005270068 B2 AU 2005270068B2
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- optionally substituted
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- alkyl
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/28—Oxygen atom
- C07D473/30—Oxygen atom attached in position 6, e.g. hypoxanthine
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- C07D473/32—Nitrogen atom
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- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US58497704P | 2004-07-02 | 2004-07-02 | |
| US60/584,977 | 2004-07-02 | ||
| PCT/US2005/023364 WO2006014325A2 (en) | 2004-07-02 | 2005-07-01 | C-met modulators and method of use |
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| Publication Number | Publication Date |
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| AU2005270068A1 AU2005270068A1 (en) | 2006-02-09 |
| AU2005270068B2 true AU2005270068B2 (en) | 2012-04-19 |
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| Application Number | Title | Priority Date | Filing Date |
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| AU2005270068A Ceased AU2005270068B2 (en) | 2004-07-02 | 2005-07-01 | C-Met modulators and method of use |
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| US (1) | US7977345B2 (https=) |
| EP (1) | EP1773826A4 (https=) |
| JP (1) | JP5368701B2 (https=) |
| AU (1) | AU2005270068B2 (https=) |
| CA (1) | CA2572331A1 (https=) |
| WO (1) | WO2006014325A2 (https=) |
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| LT4013412T (lt) | 2019-08-12 | 2026-03-25 | Deciphera Pharmaceuticals, Llc | Ripretinibas, skirtas virškinamojo trakto stromos navikų gydymui |
| HRP20231699T1 (hr) | 2019-12-30 | 2024-05-10 | Deciphera Pharmaceuticals, Llc | Formulacije inhibitora amorfne kinaze i postupci njihove primjene |
| CN115243681B (zh) | 2019-12-30 | 2024-08-16 | 德西费拉制药有限责任公司 | 1-(4-溴-5-(1-乙基-7-(甲氨基)-2-侧氧基-1,2-二氢-1,6-萘啶-3-基)-2-氟苯基)-3-苯基脲的组合物 |
| WO2021249913A1 (en) | 2020-06-09 | 2021-12-16 | Bayer Aktiengesellschaft | 2'-(quinolin-3-yl)-5',6'-dihydrospiro[azetidine-3,4'-pyrrolo[1,2-b]pyrazole]-1-carboxylate derivatives and related compounds as map4k1 (hpk1) inhibitors for the treatment of cancer |
| WO2022167627A1 (en) | 2021-02-05 | 2022-08-11 | Bayer Aktiengesellschaft | Map4k1 inhibitors |
| CN116836176B (zh) * | 2022-03-23 | 2026-02-24 | 中国科学院上海药物研究所 | 青蒿素类化合物、其制备方法和应用 |
| CN115160340B (zh) * | 2022-06-07 | 2023-07-21 | 四川大学华西医院 | 一种具有ack1抑制活性的小分子化合物及其应用 |
| US11779572B1 (en) | 2022-09-02 | 2023-10-10 | Deciphera Pharmaceuticals, Llc | Methods of treating gastrointestinal stromal tumors |
| US20260049059A1 (en) * | 2022-11-25 | 2026-02-19 | Synthon B.V. | A process for preparation of cabozantinib or tivozanib |
| TW202444365A (zh) | 2023-01-31 | 2024-11-16 | 漢達生技醫藥股份有限公司 | 改良之卡博替尼組合物及其使用方法 |
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- 2005-07-01 EP EP05763620A patent/EP1773826A4/en not_active Withdrawn
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Also Published As
| Publication number | Publication date |
|---|---|
| EP1773826A2 (en) | 2007-04-18 |
| WO2006014325A3 (en) | 2007-03-01 |
| US7977345B2 (en) | 2011-07-12 |
| AU2005270068A1 (en) | 2006-02-09 |
| CA2572331A1 (en) | 2006-02-09 |
| WO2006014325A2 (en) | 2006-02-09 |
| EP1773826A4 (en) | 2009-06-03 |
| JP2008505181A (ja) | 2008-02-21 |
| JP5368701B2 (ja) | 2013-12-18 |
| US20070179130A1 (en) | 2007-08-02 |
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