AU2004268941A1 - Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases - Google Patents

Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases Download PDF

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Publication number
AU2004268941A1
AU2004268941A1 AU2004268941A AU2004268941A AU2004268941A1 AU 2004268941 A1 AU2004268941 A1 AU 2004268941A1 AU 2004268941 A AU2004268941 A AU 2004268941A AU 2004268941 A AU2004268941 A AU 2004268941A AU 2004268941 A1 AU2004268941 A1 AU 2004268941A1
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Prior art keywords
substituted
compound
group
formula
heterocycle
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AU2004268941A
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Inventor
Timothy James Davis
Sunil K.C. Kumar
Jagadish Sircar
Wenbin Ying
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Avanir Pharmaceuticals Inc
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Avanir Pharmaceuticals Inc
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Application filed by Avanir Pharmaceuticals Inc filed Critical Avanir Pharmaceuticals Inc
Publication of AU2004268941A1 publication Critical patent/AU2004268941A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61P37/02—Immunomodulators
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P7/06—Antianaemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Virology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
AU2004268941A 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases Abandoned AU2004268941A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US49744303P 2003-08-22 2003-08-22
US60/497,443 2003-08-22
PCT/US2004/025683 WO2005021546A1 (en) 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases

Publications (1)

Publication Number Publication Date
AU2004268941A1 true AU2004268941A1 (en) 2005-03-10

Family

ID=34272569

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AU2004268941A Abandoned AU2004268941A1 (en) 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases

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Country Link
US (2) US20050124604A1 (enExample)
EP (1) EP1656376A1 (enExample)
JP (1) JP2007503388A (enExample)
CN (1) CN1839133A (enExample)
AR (1) AR045471A1 (enExample)
AU (1) AU2004268941A1 (enExample)
BR (1) BRPI0413695A (enExample)
CA (1) CA2531506A1 (enExample)
MX (1) MXJL06000006A (enExample)
PE (1) PE20051112A1 (enExample)
TW (1) TW200524928A (enExample)
UY (1) UY28483A1 (enExample)
WO (1) WO2005021546A1 (enExample)

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JP7377679B2 (ja) 2018-11-19 2023-11-10 アムジエン・インコーポレーテツド がん治療のためのｋｒａｓｇ１２ｃ阻害剤及び１種以上の薬学的に活性な追加の薬剤を含む併用療法
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US20070191388A1 (en) 2007-08-16
CN1839133A (zh) 2006-09-27
US20050124604A1 (en) 2005-06-09
AR045471A1 (es) 2005-10-26
EP1656376A1 (en) 2006-05-17
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CA2531506A1 (en) 2005-03-10
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UY28483A1 (es) 2005-03-31
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