AU2002234588B2 - Organic compounds - Google Patents

Organic compounds Download PDF

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Publication number
AU2002234588B2
AU2002234588B2 AU2002234588A AU2002234588A AU2002234588B2 AU 2002234588 B2 AU2002234588 B2 AU 2002234588B2 AU 2002234588 A AU2002234588 A AU 2002234588A AU 2002234588 A AU2002234588 A AU 2002234588A AU 2002234588 B2 AU2002234588 B2 AU 2002234588B2
Authority
AU
Australia
Prior art keywords
alkyl
halogen
formula
compounds
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU2002234588A
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English (en)
Other versions
AU2002234588A1 (en
Inventor
Jacques Bouvier
Pierre Ducray
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Elanco Tiergesundheit AG
Original Assignee
Elanco Tiergesundheit AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elanco Tiergesundheit AG filed Critical Elanco Tiergesundheit AG
Publication of AU2002234588A1 publication Critical patent/AU2002234588A1/en
Application granted granted Critical
Publication of AU2002234588B2 publication Critical patent/AU2002234588B2/en
Assigned to NOVARTIS AG, ELANCO TIERGESUNDHEIT AG reassignment NOVARTIS AG Request to Amend Deed and Register Assignors: NOVARTIS AG, Novartis Tiergensunheit AG
Assigned to NOVARTIS TIERGESUNDHEIT AG reassignment NOVARTIS TIERGESUNDHEIT AG Request for Assignment Assignors: NOVARTIS AG
Assigned to ELANCO TIERGESUNDHEIT AG reassignment ELANCO TIERGESUNDHEIT AG Request to Amend Deed and Register Assignors: NOVARTIS TIERGESUNDHEIT AG
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/275—Nitriles; Isonitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/275—Nitriles; Isonitriles
    • A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Paper (AREA)
AU2002234588A 2000-12-20 2001-12-18 Organic compounds Expired AU2002234588B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH2489/00 2000-12-20
CH24892000 2000-12-20
PCT/EP2001/014926 WO2002049641A2 (en) 2000-12-20 2001-12-18 Anti-endoparasitic amidoacetonitrils

Publications (2)

Publication Number Publication Date
AU2002234588A1 AU2002234588A1 (en) 2002-09-05
AU2002234588B2 true AU2002234588B2 (en) 2005-03-24

Family

ID=4569596

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2002234588A Expired AU2002234588B2 (en) 2000-12-20 2001-12-18 Organic compounds
AU3458802A Pending AU3458802A (en) 2000-12-20 2001-12-18 Organic compounds

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU3458802A Pending AU3458802A (en) 2000-12-20 2001-12-18 Organic compounds

Country Status (21)

Country Link
US (1) US7700656B2 (enExample)
EP (1) EP1392281B1 (enExample)
JP (1) JP2004521097A (enExample)
KR (1) KR100850252B1 (enExample)
CN (1) CN1531426A (enExample)
AR (1) AR035523A1 (enExample)
AT (1) ATE354360T1 (enExample)
AU (2) AU2002234588B2 (enExample)
BR (1) BR0116326A (enExample)
CA (1) CA2432388C (enExample)
CY (1) CY1106509T1 (enExample)
DE (1) DE60126838T2 (enExample)
DK (1) DK1392281T3 (enExample)
ES (1) ES2281453T3 (enExample)
MX (1) MXPA03005701A (enExample)
NZ (1) NZ526538A (enExample)
PT (1) PT1392281E (enExample)
RU (1) RU2286775C2 (enExample)
TW (1) TWI292712B (enExample)
WO (1) WO2002049641A2 (enExample)
ZA (1) ZA200304331B (enExample)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
TWI261053B (en) 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
TW200409760A (en) 2002-09-11 2004-06-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
AU2005303993B2 (en) * 2004-11-09 2009-10-29 Elanco Tiergesundheit Ag Process for the preparation of enantiomers of amidoacetonitrile compounds from their racemates
JP2009502834A (ja) * 2005-07-25 2009-01-29 ノバルティス アクチエンゲゼルシャフト アミドニトリル化合物
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
ES2435191T3 (es) 2007-02-09 2013-12-16 Pfizer Limited Agentes antiparasitarios
BRPI0807354A2 (pt) * 2007-02-21 2014-05-06 Pfizer Ltd Agentes antiparasíticos
ME03373B (me) 2007-05-15 2020-01-20 Merial Inc Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene
BRPI0920145B8 (pt) 2008-10-21 2021-05-25 Merial Ltd compostos de tioamida, método de produção e método de uso dos mesmos
PT3050874T (pt) 2008-11-14 2019-05-09 Boehringer Ingelheim Animal Health Usa Inc Compostos parasiticidas de ariloazol-2-il-cianoetilamino enantiomericamente enriquecidos
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
KR101856577B1 (ko) * 2011-03-02 2018-05-10 고쿠리츠다이가쿠호우진 도쿄다이가쿠 내부 기생충 방제제
MX349802B (es) * 2011-11-25 2017-08-14 Bayer Ip Gmbh Uso de aril- y hetarilcarboxamidas como endoparasiticidas.
WO2013122041A1 (ja) * 2012-02-14 2013-08-22 日本曹達株式会社 アリールオキシ酢酸アミド化合物および有害生物防除剤
US9790176B2 (en) * 2012-08-06 2017-10-17 Pitney Pharmaceuticals Pty Limited Compounds for the treatment of mTOR pathway related diseases
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
JP6556700B2 (ja) * 2013-09-13 2019-08-07 ピットニー ファーマシューティカル ピーティーワイ リミテッド アミノアセトニトリル化合物を有効成分として含有する抗癌剤
JP2018513835A (ja) * 2015-02-24 2018-05-31 ピットニー ファーマシューティカル ピーティーワイ リミテッド アミノアセトニトリル化合物を有効成分とする抗癌剤
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) * 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
EP0580374A1 (en) * 1992-07-23 1994-01-26 Ishihara Sangyo Kaisha, Ltd. Pyridine amides and their salts, processes for their production and pesticidal compositions containing them
EP0953565A2 (en) * 1998-05-01 1999-11-03 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative, agricultural and horticultural insecticide containing the same, and use thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
KR100628842B1 (ko) 2001-05-15 2006-09-29 노파르티스 아게 벤즈아미도아세토니트릴 및 이의 항기생충제로서의 용도
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) * 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
EP0580374A1 (en) * 1992-07-23 1994-01-26 Ishihara Sangyo Kaisha, Ltd. Pyridine amides and their salts, processes for their production and pesticidal compositions containing them
EP0953565A2 (en) * 1998-05-01 1999-11-03 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative, agricultural and horticultural insecticide containing the same, and use thereof

Also Published As

Publication number Publication date
KR20030061414A (ko) 2003-07-18
US20040082624A1 (en) 2004-04-29
BR0116326A (pt) 2004-07-06
CA2432388A1 (en) 2002-06-27
ATE354360T1 (de) 2007-03-15
CA2432388C (en) 2010-06-08
US7700656B2 (en) 2010-04-20
JP2004521097A (ja) 2004-07-15
TWI292712B (en) 2008-01-21
AU3458802A (en) 2002-07-01
CY1106509T1 (el) 2012-01-25
NZ526538A (en) 2005-12-23
DE60126838T2 (de) 2007-11-08
DE60126838D1 (de) 2007-04-05
WO2002049641A3 (en) 2003-12-04
AR035523A1 (es) 2004-06-02
RU2003122196A (ru) 2005-03-20
RU2286775C2 (ru) 2006-11-10
WO2002049641A2 (en) 2002-06-27
EP1392281B1 (en) 2007-02-21
ES2281453T3 (es) 2007-10-01
PT1392281E (pt) 2007-05-31
ZA200304331B (en) 2004-04-28
CN1531426A (zh) 2004-09-22
MXPA03005701A (es) 2003-10-06
DK1392281T3 (da) 2007-06-11
KR100850252B1 (ko) 2008-08-04
EP1392281A2 (en) 2004-03-03

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Owner name: NOVARTIS AG

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Owner name: ELANCO TIERGESUNDHEIT AG

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PC Assignment registered

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HB Alteration of name in register

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MK14 Patent ceased section 143(a) (annual fees not paid) or expired