SE0100567D0
(sv)
*
|
2001-02-20 |
2001-02-20 |
Astrazeneca Ab |
Compounds
|
WO2003027276A2
(en)
*
|
2001-09-24 |
2003-04-03 |
University Of Aarhus |
Novel compositions and methods for diagnosis and treatment of lymphoma and leukemia
|
DE60215864T2
(de)
*
|
2001-11-30 |
2007-05-31 |
Qlt Inc., Vancouver |
Behandlung von okularen neovaskularen erkrankungen
|
WO2003074525A1
(fr)
*
|
2002-03-01 |
2003-09-12 |
Yamanouchi Pharmaceutical Co., Ltd. |
Compose heterocyclique azote
|
AU2003255845A1
(en)
*
|
2002-08-22 |
2004-03-11 |
Piramed Limited |
Phosphadidylinositol 3,5-biphosphate inhibitors as anti-viral agents
|
BRPI0414171A
(pt)
*
|
2003-09-04 |
2006-10-31 |
Warner Lambert Co |
benzo[b]tiofenos halossubstituìdos com atividade inibidora de pi3k como agentes terapêuticos
|
EA012328B1
(ru)
*
|
2004-01-12 |
2009-08-28 |
Лаборатуар Сероно Са |
Производные тиазола и их применение
|
EP1786811A2
(de)
*
|
2004-08-18 |
2007-05-23 |
Pharmacia & Upjohn Company LLC |
Triazolopyridinverbindungen
|
GB0420722D0
(en)
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
AU2005302279A1
(en)
*
|
2004-10-28 |
2006-05-11 |
Irm Llc |
Compounds and compositions as hedgehog pathway modulators
|
WO2006049339A1
(ja)
|
2004-11-08 |
2006-05-11 |
Banyu Pharmaceutical Co., Ltd. |
新規縮環イミダゾール誘導体
|
US7723336B2
(en)
|
2005-09-22 |
2010-05-25 |
Bristol-Myers Squibb Company |
Fused heterocyclic compounds useful as kinase modulators
|
TWI417095B
(zh)
|
2006-03-15 |
2013-12-01 |
Janssen Pharmaceuticals Inc |
1,4-二取代之3-氰基-吡啶酮衍生物及其作為mGluR2-受體之正向異位性調節劑之用途
|
CA2663528A1
(en)
*
|
2006-09-18 |
2008-03-27 |
Vertex Pharmaceuticals Incorporated |
Heterocyclic inhibitors of c-met and uses thereof
|
KR20090085591A
(ko)
*
|
2006-10-30 |
2009-08-07 |
노파르티스 아게 |
Pi3k 지질 키나제 억제제로서의 이미다조피리다진
|
EP1972631A1
(de)
*
|
2007-03-23 |
2008-09-24 |
Novartis AG |
Imidazopyridazine als PI3K-Lipidkinaseinhibitoren
|
CA2670636A1
(en)
|
2006-11-27 |
2008-06-05 |
H. Lundbeck A/S |
Heteroaryl amide derivatives
|
AR064106A1
(es)
*
|
2006-12-05 |
2009-03-11 |
Bayer Schering Pharma Ag |
Derivados de 2,3-dihidroimidazo [1,2-c] quinazolina sustituida utiles para el tratamiento de enfermedades y trastornos hiper-proliferativos asociados con la angiogenesis
|
CN101502484B
(zh)
*
|
2006-12-26 |
2011-04-20 |
济南康泉医药科技有限公司 |
同载糖皮质激素和化疗药物的抗癌缓释剂
|
TW200900065A
(en)
|
2007-03-07 |
2009-01-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
|
TW200845978A
(en)
|
2007-03-07 |
2008-12-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
|
SG182205A1
(en)
|
2007-03-15 |
2012-07-30 |
Novartis Ag |
Organic compounds and their uses
|
WO2008124323A1
(en)
|
2007-04-03 |
2008-10-16 |
Array Biopharma Inc. |
Imidazo[1,2-a]pyridine compounds as receptor tyrosine kinase inhibitors
|
MX2009010523A
(es)
|
2007-04-10 |
2009-12-15 |
Lundbeck & Co As H |
Análogos de amidas heteroarílicas como antagonistas de p2x7.
|
JP2010524953A
(ja)
*
|
2007-04-17 |
2010-07-22 |
ブリストル−マイヤーズ スクイブ カンパニー |
縮合ヘテロ環11−β−ヒドロキシステロイドデヒドロゲナーゼI型阻害剤
|
PE20090215A1
(es)
*
|
2007-05-09 |
2009-03-30 |
Novartis Ag |
Compuestos derivados de imidazopiridazinas como inhibidores de cinasa
|
WO2008141731A2
(en)
*
|
2007-05-18 |
2008-11-27 |
Bayer Healthcare Ag |
Inhibitors of hypoxia inducible factor (hif) useful for treating hyper-proliferative disorders and diseases associated with angiogenesis
|
EP2176259B1
(de)
|
2007-08-14 |
2011-03-30 |
Bayer Schering Pharma Aktiengesellschaft |
Kondensierte imidazole zur krebsbehandlung
|
EP2062893A1
(de)
*
|
2007-10-18 |
2009-05-27 |
Bayer Schering Pharma AG |
Fusionierte Imidazole zur Behandlung von Krebs
|
US9114138B2
(en)
|
2007-09-14 |
2015-08-25 |
Janssen Pharmaceuticals, Inc. |
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones
|
EA019085B1
(ru)
|
2007-09-14 |
2014-01-30 |
Янссен Фармасьютикалз, Инк. |
1',3-двузамещенные 4-(арил-х-фенил)-1н-пиридин-2-оны
|
EP2060565A1
(de)
|
2007-11-16 |
2009-05-20 |
4Sc Ag |
Neue bifunktionelle Verbindungen die Proteinkinasen und Histonedeacetylasen hemmen
|
UA102828C2
(en)
*
|
2007-11-27 |
2013-08-27 |
Целльзом Лимитед |
Amino triazoles as p13k inhibitors
|
US8389527B2
(en)
|
2008-02-06 |
2013-03-05 |
Bristol-Myers Squibb Company |
Substituted imidazopyridazines useful as kinase inhibitors
|
CA2717034A1
(en)
|
2008-02-28 |
2009-09-03 |
Pascal Furet |
Imidazo[1,2-b]pyridazine derivatives for the treatment of c-met tyrosine kinase mediated disease
|
US8394823B2
(en)
|
2008-04-11 |
2013-03-12 |
Bristol-Myers Squibb Company |
Triazolopyridine compounds useful as DGAT1 inhibitors
|
WO2009126624A1
(en)
|
2008-04-11 |
2009-10-15 |
Bristol-Myers Squibb Company |
Triazolo compounds useful as dgat1 inhibitors
|
NZ590320A
(en)
|
2008-07-14 |
2012-12-21 |
Gilead Sciences Inc |
Fused heterocyclyc inhibitors of histone deacetylase and/or cyclin-dependent kinases
|
US8344018B2
(en)
|
2008-07-14 |
2013-01-01 |
Gilead Sciences, Inc. |
Oxindolyl inhibitor compounds
|
NZ590283A
(en)
|
2008-07-14 |
2012-11-30 |
Gilead Sciences Inc |
Imidazolylpyrimidine compounds as hdac and / or cdk inhibitors
|
WO2010007099A1
(en)
*
|
2008-07-15 |
2010-01-21 |
Cellzome Limited |
2-aminoimidazo[1,2-b]pyridazine derivatives as pi3k inhibitors
|
US20100041663A1
(en)
|
2008-07-18 |
2010-02-18 |
Novartis Ag |
Organic Compounds as Smo Inhibitors
|
CN102123987A
(zh)
|
2008-07-28 |
2011-07-13 |
吉里德科学公司 |
亚环烷基和亚杂环烷基组蛋白脱乙酰酶抑制剂化合物
|
TWI496779B
(zh)
|
2008-08-19 |
2015-08-21 |
Array Biopharma Inc |
作為pim激酶抑制劑之三唑吡啶化合物
|
US8895550B2
(en)
|
2008-08-19 |
2014-11-25 |
Array Biopharma Inc. |
Triazolopyridine compounds as PIM kinase inhibitors
|
WO2010022081A1
(en)
*
|
2008-08-19 |
2010-02-25 |
Array Biopharma Inc. |
Triazolopyridine compounds as pim kinase inhibitors
|
US8987251B2
(en)
|
2008-08-19 |
2015-03-24 |
Array Biopharma Inc. |
Triazolopyridine compounds as PIM kinase inhibitors
|
WO2010025890A1
(en)
|
2008-09-02 |
2010-03-11 |
Ortho-Mcneil-Janssen Pharmaceuticals, Inc |
3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors
|
TWI491610B
(zh)
|
2008-10-09 |
2015-07-11 |
必治妥美雅史谷比公司 |
作為激酶抑制劑之咪唑并嗒腈
|
AU2009319387B2
(en)
|
2008-11-28 |
2012-05-10 |
Addex Pharma S.A. |
Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
|
WO2010074586A1
(en)
*
|
2008-12-23 |
2010-07-01 |
Pathway Therapeutics Limited |
Pyrazolo[1,5-a]pyridine and imidazo[1,2-a]pyridine derivatives and their use in cancer therapy
|
WO2010117926A1
(en)
|
2009-04-07 |
2010-10-14 |
Schering Corporation |
Substituted triazolopyridines and analogs thereof
|
CA2760259C
(en)
|
2009-05-12 |
2018-05-01 |
Janssen Pharmaceuticals, Inc. |
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
|
MY153913A
(en)
|
2009-05-12 |
2015-04-15 |
Janssen Pharmaceuticals Inc |
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
|
JP5634506B2
(ja)
|
2009-05-12 |
2014-12-03 |
ジャンセン ファーマシューティカルズ, インコーポレイテッド |
1,2,3−トリアゾロ[4,3−a]ピリジン誘導体ならびに神経障害および精神障害の治療または予防のためのその使用
|
JP2012529514A
(ja)
|
2009-06-08 |
2012-11-22 |
ギリアード サイエンシーズ, インコーポレイテッド |
シクロアルキルカルバメートベンズアミドアニリンhdac阻害剤化合物
|
WO2010144371A1
(en)
|
2009-06-08 |
2010-12-16 |
Gilead Colorado, Inc. |
Alkanoylamino benzamide aniline hdac inihibitor compounds
|
US8389526B2
(en)
|
2009-08-07 |
2013-03-05 |
Novartis Ag |
3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
|
CA2770873A1
(en)
|
2009-08-12 |
2011-02-17 |
Novartis Ag |
Heterocyclic hydrazone compounds and their uses to treat cancer and inflammation
|
EP2467383A1
(de)
|
2009-08-20 |
2012-06-27 |
Novartis AG |
Heterocyclische oximverbindungen
|
CN110483499A
(zh)
|
2009-11-05 |
2019-11-22 |
圣母大学 |
咪唑并[1,2-a]吡啶类化合物及其合成及使用方法
|
EP2496577A1
(de)
*
|
2009-11-06 |
2012-09-12 |
Piramal Life Sciences Limited |
Imidazopyridinderivate
|
MX2012007367A
(es)
*
|
2009-12-30 |
2013-04-03 |
Arqule Inc |
Compuestos substituidos de imidazopiridinilo-aminopiridina.
|
EP2563792B1
(de)
|
2010-04-28 |
2014-08-27 |
Bristol-Myers Squibb Company |
Imidazopyridazinylverbindungen und ihre verwendung für krebs
|
TWI541243B
(zh)
|
2010-09-10 |
2016-07-11 |
拜耳知識產權公司 |
經取代咪唑并嗒
|
JP5852666B2
(ja)
|
2010-11-08 |
2016-02-03 |
ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド |
1,2,4−トリアゾロ[4,3−a]ピリジン誘導体およびmGluR2受容体のポジティブアロステリックモジュレーターとしてのそれらの使用
|
ES2552455T3
(es)
|
2010-11-08 |
2015-11-30 |
Janssen Pharmaceuticals, Inc. |
Derivados de 1,2,4-triazolo[4,3-a]piridina y su uso como moduladores alostéricos positivos de receptores mGluR2
|
JP5852665B2
(ja)
|
2010-11-08 |
2016-02-03 |
ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド |
1,2,4−トリアゾロ[4,3−a]ピリジン誘導体およびmGluR2受容体のポジティブアロステリックモジュレーターとしてのそれらの使用
|
US20120129872A1
(en)
*
|
2010-11-18 |
2012-05-24 |
Kristi Anne Leonard |
Fused heteroaryl inhibitors of pro-matrix metalloproteinase activation
|
WO2012087833A1
(en)
|
2010-12-22 |
2012-06-28 |
Abbott Laboratories |
Hepatitis c inhibitors and uses thereof
|
CN102030752A
(zh)
*
|
2011-01-06 |
2011-04-27 |
贵阳中医学院 |
一种制备化合物2-(咪唑并[1,2-a]吡啶-3-基)乙腈的方法
|
CN103298468A
(zh)
|
2011-02-01 |
2013-09-11 |
协和发酵麒麟株式会社 |
稠环杂环衍生物
|
ME02365B
(de)
|
2011-02-25 |
2016-06-20 |
Array Biopharma Inc |
Triazolopyridinverbindungen als pim-kinase-hemmer
|
EA024890B1
(ru)
|
2011-04-07 |
2016-10-31 |
Байер Интеллектчуал Проперти Гмбх |
Имидазопиридазины в качестве ингибиторов akt киназы
|
WO2012156379A1
(en)
*
|
2011-05-13 |
2012-11-22 |
Universität Zürich |
PIK3/P110α INHIBITORS FOR PREVENTION OF RESTENOSIS BY APPLICATION AS AN IMPLANT COATING
|
KR101274986B1
(ko)
*
|
2011-07-27 |
2013-06-17 |
한국과학기술원 |
이미다조피리딘 유도체, 이를 포함하는 PI3K 및/또는 mTOR 저해제용 약학 조성물 및 PI3K 및/또는 mTOR과 연관된 질환 치료용 약학 조성물
|
WO2014021383A1
(ja)
|
2012-07-31 |
2014-02-06 |
協和発酵キリン株式会社 |
縮環複素環化合物
|
US8796305B2
(en)
|
2012-11-05 |
2014-08-05 |
Bayer Pharma Aktiengesellschaft |
Carboxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
US8778964B2
(en)
|
2012-11-05 |
2014-07-15 |
Bayer Pharma Aktiengesellschaft |
Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use
|
US9624214B2
(en)
|
2012-11-05 |
2017-04-18 |
Bayer Pharma Aktiengesellschaft |
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
US9126998B2
(en)
|
2012-11-05 |
2015-09-08 |
Bayer Pharma AG |
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
|
MX2015006856A
(es)
*
|
2012-11-30 |
2016-02-17 |
Astellas Pharma Inc |
Compuestos imidazopiridina.
|
PE20151332A1
(es)
|
2013-02-19 |
2015-09-20 |
Pfizer |
Compuestos de azabencimidazol
|
JO3368B1
(ar)
|
2013-06-04 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
|
CA2914100A1
(en)
*
|
2013-06-04 |
2014-12-11 |
Bayer Pharma Aktiengesellschaft |
3-aryl-substituted imidazo[1,2-a]pyridines and the use thereof
|
JO3367B1
(ar)
|
2013-09-06 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
|
LT3096790T
(lt)
|
2014-01-21 |
2019-10-10 |
Janssen Pharmaceutica, N.V. |
Deriniai, apimantys 2 potipio metabotropinio glutamaterginio receptoriaus teigiamus alosterinius moduliatorius arba ortosterinius agonistus, ir jų panaudojimas
|
WO2015110435A1
(en)
|
2014-01-21 |
2015-07-30 |
Janssen Pharmaceutica Nv |
Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use
|
SG11201606689VA
(en)
|
2014-02-13 |
2016-09-29 |
Incyte Corp |
Cyclopropylamines as lsd1 inhibitors
|
ES2672797T3
(es)
|
2014-02-13 |
2018-06-18 |
Incyte Corporation |
Ciclopropilaminas como inhibidores de LSD1
|
WO2015123437A1
(en)
|
2014-02-13 |
2015-08-20 |
Incyte Corporation |
Cyclopropylamines as lsd1 inhibitors
|
BR112016018555B1
(pt)
|
2014-02-13 |
2024-01-23 |
Incyte Holdings Corporation |
Ciclopropilaminas como inibidores de lsd1, seu uso, composição farmacêutica que os compreende e método de inibição de lsd1
|
CN106459090A
(zh)
|
2014-02-19 |
2017-02-22 |
拜耳制药股份公司 |
3‑(嘧啶‑2‑基)咪唑并[1,2‑a]吡啶
|
EP3119777A1
(de)
|
2014-03-21 |
2017-01-25 |
Bayer Pharma Aktiengesellschaft |
Cyano-substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung
|
WO2015148464A1
(en)
*
|
2014-03-24 |
2015-10-01 |
Arqule Inc. |
Process of preparing 3-(3-(4-(1-aminocyclobutyl)phenyl)-5-phenyl-3h-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine
|
WO2015164479A1
(en)
*
|
2014-04-22 |
2015-10-29 |
Arqule, Inc. |
Salts and polymorphs of a substituted imidazopyridinyl-aminopyridine compound
|
EP3137463A1
(de)
|
2014-05-02 |
2017-03-08 |
Bayer Pharma Aktiengesellschaft |
Enantiomere des n-(2-amino-5-fluor-2-methylpentyl)-8-[(2,6-difluorbenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-carboxamids sowie der di- and tri-fluor-derivate zur behandlung von kardiovaskulären erkrankungen
|
WO2016007727A1
(en)
|
2014-07-10 |
2016-01-14 |
Incyte Corporation |
Triazolopyridines and triazolopyrazines as lsd1 inhibitors
|
TW201613925A
(en)
|
2014-07-10 |
2016-04-16 |
Incyte Corp |
Imidazopyrazines as LSD1 inhibitors
|
WO2016007731A1
(en)
|
2014-07-10 |
2016-01-14 |
Incyte Corporation |
Imidazopyridines and imidazopyrazines as lsd1 inhibitors
|
US9695167B2
(en)
|
2014-07-10 |
2017-07-04 |
Incyte Corporation |
Substituted triazolo[1,5-a]pyridines and triazolo[1,5-a]pyrazines as LSD1 inhibitors
|
JP6713982B2
(ja)
|
2014-07-24 |
2020-06-24 |
ファイザー・インク |
ピラゾロピリミジン化合物
|
DK3177624T3
(da)
|
2014-08-06 |
2019-07-01 |
Pfizer |
Imidazopyridazinforbindelser
|
CN107001361A
(zh)
|
2014-12-02 |
2017-08-01 |
拜耳医药股份有限公司 |
杂芳基取代的咪唑并[1,2‑a]吡啶及其用途
|
US9944647B2
(en)
|
2015-04-03 |
2018-04-17 |
Incyte Corporation |
Heterocyclic compounds as LSD1 inhibitors
|
US10329255B2
(en)
|
2015-08-12 |
2019-06-25 |
Incyte Corporation |
Salts of an LSD1 inhibitor
|
PE20181352A1
(es)
|
2015-09-17 |
2018-08-22 |
Marvin J Miller |
Compuestos heterociclicos que contienen bencilamina y composiciones utiles contra infeccion por micobacterias
|
GB201602527D0
(en)
*
|
2016-02-12 |
2016-03-30 |
Glaxosmithkline Ip Dev Ltd |
Chemical compounds
|
CN107304202A
(zh)
*
|
2016-04-20 |
2017-10-31 |
苏州苏领生物医药有限公司 |
五元杂环类化合物及其制备方法、药物组合物和用途
|
WO2017181973A1
(zh)
*
|
2016-04-20 |
2017-10-26 |
苏州苏领生物医药有限公司 |
五元杂环类化合物及其制备方法、药物组合物和用途
|
AU2017252328B2
(en)
|
2016-04-22 |
2023-02-23 |
Incyte Corporation |
Formulations of an LSD1 inhibitor
|
EP3454852A4
(de)
|
2016-05-11 |
2020-02-26 |
Emory University |
Phosphotidylinositol-3-kinase-inhibitoren
|
US11352328B2
(en)
|
2016-07-12 |
2022-06-07 |
Arisan Therapeutics Inc. |
Heterocyclic compounds for the treatment of arenavirus
|
WO2018184976A1
(de)
|
2017-04-05 |
2018-10-11 |
Bayer Pharma Aktiengesellschaft |
Substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung
|
CN111225917A
(zh)
|
2017-10-24 |
2020-06-02 |
拜耳股份公司 |
取代咪唑并吡啶酰胺及其用途
|
WO2020047198A1
(en)
|
2018-08-31 |
2020-03-05 |
Incyte Corporation |
Salts of an lsd1 inhibitor and processes for preparing the same
|
US11560388B2
(en)
|
2019-03-19 |
2023-01-24 |
Boehringer Ingelheim Vetmedica Gmbh |
Anthelmintic aza-benzothiophene and aza-benzofuran compounds
|
WO2020216669A1
(de)
|
2019-04-23 |
2020-10-29 |
Bayer Aktiengesellschaft |
Phenylsubstituierte imidazopyridinamide und ihre verwendung
|
TW202206407A
(zh)
*
|
2020-04-27 |
2022-02-16 |
南韓商奧士擇破利悟股份有限公司 |
用於ubr盒結構域配體之化合物、組成物以及醫藥組成物
|
WO2021242581A1
(en)
|
2020-05-29 |
2021-12-02 |
Boehringer Ingelheim Animal Health USA Inc. |
Anthelmintic heterocyclic compounds
|
CN113135913B
(zh)
*
|
2021-04-28 |
2022-05-24 |
沈阳药科大学 |
3-取代基-6-吡啶类取代基-六元并五元杂环类衍生物及其制法与用途
|
CA3236894A1
(en)
|
2021-11-01 |
2023-05-04 |
Boehringer Ingelheim Vetmedica Gmbh |
Anthelmintic pyrrolopyridazine compounds
|