MX2012007367A - Compuestos substituidos de imidazopiridinilo-aminopiridina. - Google Patents

Compuestos substituidos de imidazopiridinilo-aminopiridina.

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Publication number
MX2012007367A
MX2012007367A MX2012007367A MX2012007367A MX2012007367A MX 2012007367 A MX2012007367 A MX 2012007367A MX 2012007367 A MX2012007367 A MX 2012007367A MX 2012007367 A MX2012007367 A MX 2012007367A MX 2012007367 A MX2012007367 A MX 2012007367A
Authority
MX
Mexico
Prior art keywords
compounds
substituted imidazopyridinyl
aminopyridine compounds
aminopyridine
methods
Prior art date
Application number
MX2012007367A
Other languages
English (en)
Inventor
Shin Iimura
Yanbin Liu
Jason Hill
Rocio Palma
Jean-Marc Lapierre
Manish Tandon
David Vensel
Nivedita Namdev
Mark A Ashwell
Chris Brassard
Anton Filikov
Steffi Koerner
Robert Nicewonger
Akihisa Matsuda
Yuko Yamamoto
Original Assignee
Arqule Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arqule Inc filed Critical Arqule Inc
Publication of MX2012007367A publication Critical patent/MX2012007367A/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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Abstract

La presente invención se relaciona con compuestos sustituidos de imidazopiridinilo-aminopiridina y métodos para sintetizar estos compuestos. La presente invención también se relaciona con composiciones farmacéuticas que contienen compuestos sustituidos de imidazopiridinilo-aminopiridina y métodos para el tratamiento de trastornos celulares proliferativos, tales como cáncer, mediante la administración de estos compuestos y composiciones farmacéuticas a sujetos en necesidad de los mismos.
MX2012007367A 2009-12-30 2010-12-29 Compuestos substituidos de imidazopiridinilo-aminopiridina. MX2012007367A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29092309P 2009-12-30 2009-12-30
PCT/US2010/062440 WO2011082270A2 (en) 2009-12-30 2010-12-29 Substituted imidazopyridinyl-aminopyridine compounds

Publications (1)

Publication Number Publication Date
MX2012007367A true MX2012007367A (es) 2013-04-03

Family

ID=44227150

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012007367A MX2012007367A (es) 2009-12-30 2010-12-29 Compuestos substituidos de imidazopiridinilo-aminopiridina.

Country Status (20)

Country Link
US (1) US8501770B2 (es)
EP (1) EP2519522B1 (es)
JP (1) JP5774602B2 (es)
KR (1) KR101689421B1 (es)
CN (1) CN102781940B (es)
AU (1) AU2010339533B2 (es)
BR (1) BR112012016398B1 (es)
CA (1) CA2785536C (es)
CO (1) CO6511271A2 (es)
DK (1) DK2519522T3 (es)
ES (1) ES2531109T3 (es)
IL (1) IL220571A (es)
MX (1) MX2012007367A (es)
MY (1) MY157124A (es)
NZ (1) NZ600801A (es)
PH (1) PH12012501323A1 (es)
RU (1) RU2619463C2 (es)
SG (1) SG181947A1 (es)
TW (1) TWI585086B (es)
WO (1) WO2011082270A2 (es)

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