ATE368656T1 - Piperidinderivate zur verwendung bei der behandlung von durch chemokins vermittelten leiden - Google Patents

Piperidinderivate zur verwendung bei der behandlung von durch chemokins vermittelten leiden

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Publication number
ATE368656T1
ATE368656T1 AT03798620T AT03798620T ATE368656T1 AT E368656 T1 ATE368656 T1 AT E368656T1 AT 03798620 T AT03798620 T AT 03798620T AT 03798620 T AT03798620 T AT 03798620T AT E368656 T1 ATE368656 T1 AT E368656T1
Authority
AT
Austria
Prior art keywords
chemokine
treatment
piperidine derivatives
mediated conditions
formula
Prior art date
Application number
AT03798620T
Other languages
English (en)
Inventor
Christopher Luckhurst
Matthew Perry
Brian Springthorpe
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of ATE368656T1 publication Critical patent/ATE368656T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • AIDS & HIV (AREA)
AT03798620T 2002-09-24 2003-09-12 Piperidinderivate zur verwendung bei der behandlung von durch chemokins vermittelten leiden ATE368656T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0202838A SE0202838D0 (sv) 2002-09-24 2002-09-24 Chemical compounds

Publications (1)

Publication Number Publication Date
ATE368656T1 true ATE368656T1 (de) 2007-08-15

Family

ID=20289093

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03798620T ATE368656T1 (de) 2002-09-24 2003-09-12 Piperidinderivate zur verwendung bei der behandlung von durch chemokins vermittelten leiden

Country Status (20)

Country Link
US (1) US20060040984A1 (de)
EP (2) EP1546130B1 (de)
JP (1) JP2006503066A (de)
KR (1) KR20050052511A (de)
CN (1) CN1684952A (de)
AT (1) ATE368656T1 (de)
AU (1) AU2003259004B2 (de)
BR (1) BR0314688A (de)
CA (1) CA2497280A1 (de)
DE (1) DE60315323T2 (de)
ES (1) ES2289354T3 (de)
IS (1) IS7813A (de)
MX (1) MXPA05003007A (de)
NO (1) NO20051965L (de)
NZ (1) NZ538527A (de)
PL (1) PL376119A1 (de)
RU (1) RU2005105053A (de)
SE (1) SE0202838D0 (de)
WO (1) WO2004029041A1 (de)
ZA (1) ZA200502341B (de)

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GB0120461D0 (en) 2001-08-22 2001-10-17 Astrazeneca Ab Novel compounds
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SE0300957D0 (sv) * 2003-04-01 2003-04-01 Astrazeneca Ab Chemical compounds
SE0301368D0 (sv) * 2003-05-09 2003-05-09 Astrazeneca Ab Chemical compounds
SE0400925D0 (sv) * 2004-04-06 2004-04-06 Astrazeneca Ab Chemical compounds
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WO2006126948A1 (en) * 2005-05-27 2006-11-30 Astrazeneca Ab Piperidines for the treatment of chemokine mediated diseases
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HRP20181863T1 (hr) 2013-05-17 2018-12-28 Janssen Sciences Ireland Uc Derivati sulfamoiltiofenamida i njihova uporaba kao lijekova za liječenje hepatitisa b
JO3583B1 (ar) 2013-05-17 2020-07-05 Janssen Sciences Ireland Uc مشتقات سلفامويل بيرولاميد واستخدامها كادوية لمعالجة التهاب الكبد نوع بي
NO3024819T3 (de) 2013-07-25 2018-07-21
MX368158B (es) 2013-10-23 2019-09-20 Janssen Sciences Ireland Uc Derivados de carboxamida y su uso como medicamentos para el tratamiento de la hepatitis b.
US10392349B2 (en) 2014-01-16 2019-08-27 Novira Therapeutics, Inc. Azepane derivatives and methods of treating hepatitis B infections
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JP2021515769A (ja) 2018-03-14 2021-06-24 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー カプシド集合調節剤の投薬レジメン
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DE60315323T2 (de) 2008-04-17
EP1546130A1 (de) 2005-06-29
RU2005105053A (ru) 2005-12-10
KR20050052511A (ko) 2005-06-02
ZA200502341B (en) 2005-09-19
EP1546130B1 (de) 2007-08-01
ES2289354T3 (es) 2008-02-01
SE0202838D0 (sv) 2002-09-24
DE60315323D1 (de) 2007-09-13
AU2003259004B2 (en) 2007-02-08
IS7813A (is) 2005-04-20
JP2006503066A (ja) 2006-01-26
CN1684952A (zh) 2005-10-19
NO20051965L (no) 2005-06-23
AU2003259004A1 (en) 2004-04-19
MXPA05003007A (es) 2005-06-22
NZ538527A (en) 2006-10-27
EP1816123A1 (de) 2007-08-08
BR0314688A (pt) 2005-08-02
PL376119A1 (en) 2005-12-12
US20060040984A1 (en) 2006-02-23
CA2497280A1 (en) 2004-04-08
NO20051965D0 (no) 2005-04-22
WO2004029041A1 (en) 2004-04-08

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