ZA200502341B - Novel piperidine derivatives for use in the tretment of chemokine mediated disease states. - Google Patents
Novel piperidine derivatives for use in the tretment of chemokine mediated disease states. Download PDFInfo
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- ZA200502341B ZA200502341B ZA200502341A ZA200502341A ZA200502341B ZA 200502341 B ZA200502341 B ZA 200502341B ZA 200502341 A ZA200502341 A ZA 200502341A ZA 200502341 A ZA200502341 A ZA 200502341A ZA 200502341 B ZA200502341 B ZA 200502341B
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
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| AR033517A1 (es) * | 2000-04-08 | 2003-12-26 | Astrazeneca Ab | Derivados de piperidina, proceso para su preparacion y uso de estos derivados en la fabricacion de medicamentos |
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| EP1937666B1 (de) | 2005-10-11 | 2012-02-22 | Schering Corporation | Substituierte heterocyclische verbindungen mit cxcr3-antagonistischer wirkung |
| TWI433838B (zh) * | 2008-06-25 | 2014-04-11 | 必治妥美雅史谷比公司 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
| GB0908394D0 (en) | 2009-05-15 | 2009-06-24 | Univ Leuven Kath | Novel viral replication inhibitors |
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| WO2012065963A2 (en) | 2010-11-15 | 2012-05-24 | Katholieke Universiteit Leuven | Novel antiviral compounds |
| ES2797123T3 (es) | 2011-12-21 | 2020-12-01 | Novira Therapeutics Inc | Agentes antivirales para la hepatitis B |
| NZ743463A (en) | 2012-08-28 | 2019-09-27 | Janssen Sciences Ireland Uc | Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b |
| SI2961732T1 (sl) | 2013-02-28 | 2017-07-31 | Janssen Sciences Ireland Uc | Sulfamoil-arilamidi in njihova uporaba kot zdravila za zdravljenje hepatitisa B |
| HUE033542T2 (en) | 2013-04-03 | 2017-12-28 | Janssen Sciences Ireland Uc | Their use as medicaments for the treatment of N-phenylcarboxamide derivatives and hepatitis B |
| JO3603B1 (ar) | 2013-05-17 | 2020-07-05 | Janssen Sciences Ireland Uc | مشتقات سلفامويل بيرولاميد واستخدامها كادوية لمعالجة التهاب الكبد نوع بي |
| LT2997019T (lt) | 2013-05-17 | 2018-11-26 | Janssen Sciences Ireland Uc | Sulfamoiltiofenamido dariniai ir jų panaudojimas kaip vaistų hepatito b gydymui |
| AP2015008968A0 (en) | 2013-07-25 | 2015-12-31 | Janssen Sciences Ireland Uc | Glyoxamide substituted pyrrolamide derivatives andthe use thereof as medicaments for the treatment of hepatitis b |
| DK3060547T3 (en) | 2013-10-23 | 2018-01-15 | Janssen Sciences Ireland Uc | CARBOXAMIDE DERIVATIVES AND USE THEREOF AS MEDICINES FOR TREATMENT OF HEPATITS B |
| US10392349B2 (en) | 2014-01-16 | 2019-08-27 | Novira Therapeutics, Inc. | Azepane derivatives and methods of treating hepatitis B infections |
| US9169212B2 (en) | 2014-01-16 | 2015-10-27 | Novira Therapeutics, Inc. | Azepane derivatives and methods of treating hepatitis B infections |
| KR20160128305A (ko) | 2014-02-05 | 2016-11-07 | 노비라 테라퓨틱스, 인코포레이티드 | Hbv 감염의 치료를 위한 병용 요법 |
| EA035848B1 (ru) | 2014-02-06 | 2020-08-20 | Янссен Сайенсиз Айрлэнд Юси | Производные сульфамоилпирроламида и их применение в качестве медикаментов для лечения гепатита b |
| JP2018510159A (ja) | 2015-03-19 | 2018-04-12 | ノヴィラ・セラピューティクス・インコーポレイテッド | アゾカン及びアゾナン誘導体及びｂ型肝炎感染症の治療法 |
| US10875876B2 (en) | 2015-07-02 | 2020-12-29 | Janssen Sciences Ireland Uc | Cyclized sulfamoylarylamide derivatives and the use thereof as medicaments for the treatment of hepatitis B |
| TW201718496A (zh) | 2015-09-29 | 2017-06-01 | 諾維拉治療公司 | B型肝炎抗病毒劑之晶型 |
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| KR20210130753A (ko) | 2019-02-22 | 2021-11-01 | 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 | Hbv 감염 또는 hbv-유발성 질환의 치료에 유용한 아미드 유도체 |
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| US4505915A (en) * | 1979-05-29 | 1985-03-19 | Merck & Co., Inc. | 6-N-Heterocyclyl penicillins |
| US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
| US4695575A (en) * | 1984-11-13 | 1987-09-22 | Janssen Pharmaceutica, N.V. | 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines |
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| WO1999055674A1 (fr) * | 1998-04-28 | 1999-11-04 | Dainippon Pharmaceutical Co., Ltd. | Derives de 1-[(1-substituee-4-piperidinyle)methyle]-4-piperidine, procede de production de ceux-ci, compositions medicinales contenant ces composes et intermediaires de ces composes |
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| DE69919171T2 (de) * | 1998-06-30 | 2005-08-04 | Schering Corp. | Muskarin-rezeptor antagonisten |
| EP1140834A1 (de) * | 1998-12-18 | 2001-10-10 | Du Pont Pharmaceuticals Company | Heterozyklische piperidine als modulatoren der aktivität der chemokinerezeptoren |
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-
2005
- 2005-03-18 ZA ZA200502341A patent/ZA200502341B/en unknown
- 2005-04-20 IS IS7813A patent/IS7813A/is unknown
- 2005-04-22 NO NO20051965A patent/NO20051965L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1684952A (zh) | 2005-10-19 |
| DE60315323T2 (de) | 2008-04-17 |
| EP1816123A1 (de) | 2007-08-08 |
| ATE368656T1 (de) | 2007-08-15 |
| US20060040984A1 (en) | 2006-02-23 |
| ES2289354T3 (es) | 2008-02-01 |
| KR20050052511A (ko) | 2005-06-02 |
| EP1546130A1 (de) | 2005-06-29 |
| PL376119A1 (en) | 2005-12-12 |
| NZ538527A (en) | 2006-10-27 |
| JP2006503066A (ja) | 2006-01-26 |
| NO20051965L (no) | 2005-06-23 |
| BR0314688A (pt) | 2005-08-02 |
| DE60315323D1 (de) | 2007-09-13 |
| RU2005105053A (ru) | 2005-12-10 |
| IS7813A (is) | 2005-04-20 |
| AU2003259004A1 (en) | 2004-04-19 |
| SE0202838D0 (sv) | 2002-09-24 |
| WO2004029041A1 (en) | 2004-04-08 |
| AU2003259004B2 (en) | 2007-02-08 |
| NO20051965D0 (no) | 2005-04-22 |
| MXPA05003007A (es) | 2005-06-22 |
| EP1546130B1 (de) | 2007-08-01 |
| CA2497280A1 (en) | 2004-04-08 |
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