ATE349459T1 - Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters - Google Patents

Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters

Info

Publication number
ATE349459T1
ATE349459T1 AT03766325T AT03766325T ATE349459T1 AT E349459 T1 ATE349459 T1 AT E349459T1 AT 03766325 T AT03766325 T AT 03766325T AT 03766325 T AT03766325 T AT 03766325T AT E349459 T1 ATE349459 T1 AT E349459T1
Authority
AT
Austria
Prior art keywords
ntrenyl
dodecahydrocyclopenta
polymorpho
phen
ester
Prior art date
Application number
AT03766325T
Other languages
German (de)
English (en)
Inventor
Guido Jordine
Michael Mutz
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE349459T1 publication Critical patent/ATE349459T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J33/00Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J33/00Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
AT03766325T 2002-07-29 2003-07-28 Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters ATE349459T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0217504.0A GB0217504D0 (en) 2002-07-29 2002-07-29 Organic compounds

Publications (1)

Publication Number Publication Date
ATE349459T1 true ATE349459T1 (de) 2007-01-15

Family

ID=9941275

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03766325T ATE349459T1 (de) 2002-07-29 2003-07-28 Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters

Country Status (30)

Country Link
US (1) US7683048B2 (enExample)
EP (2) EP1554303B1 (enExample)
JP (1) JP2006501207A (enExample)
KR (1) KR100688371B1 (enExample)
CN (1) CN1305892C (enExample)
AR (1) AR040692A1 (enExample)
AT (1) ATE349459T1 (enExample)
AU (1) AU2003251651B2 (enExample)
BR (1) BR0313044A (enExample)
CA (1) CA2493330C (enExample)
CY (1) CY1106406T1 (enExample)
DE (1) DE60310747T2 (enExample)
DK (1) DK1554303T3 (enExample)
EC (1) ECSP055579A (enExample)
ES (1) ES2279970T3 (enExample)
GB (1) GB0217504D0 (enExample)
HK (1) HK1080484B (enExample)
IL (2) IL166287A0 (enExample)
MX (1) MXPA05001173A (enExample)
MY (1) MY136407A (enExample)
NO (1) NO20050806L (enExample)
NZ (2) NZ537868A (enExample)
PE (1) PE20040722A1 (enExample)
PL (1) PL209409B1 (enExample)
PT (1) PT1554303E (enExample)
RU (2) RU2348646C1 (enExample)
SI (1) SI1554303T1 (enExample)
TW (1) TWI309164B (enExample)
WO (1) WO2004013156A1 (enExample)
ZA (1) ZA200500370B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0019172D0 (en) 2000-08-05 2000-09-27 Glaxo Group Ltd Novel compounds
AU7576001A (en) 2000-08-05 2002-02-18 Glaxo Group Ltd 6.alpha., 9.alpha.-difluoro-17.alpha.-`(2-furanylcarboxyl) oxy]-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4,-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent
US6858596B2 (en) 2000-08-05 2005-02-22 Smithkline Beecham Corporation Formulation containing anti-inflammatory androstane derivative
US6777399B2 (en) 2000-08-05 2004-08-17 Smithkline Beecham Corporation Anti-inflammatory androstane derivative compositions
WO2002088167A1 (en) 2001-04-30 2002-11-07 Glaxo Group Limited Anti-inflammatory 17.beta.-carbothioate ester derivatives of androstane with a cyclic ester group in position 17.alpha
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
GB0523654D0 (en) * 2005-11-21 2005-12-28 Novartis Ag Organic compounds
GB0523656D0 (en) * 2005-11-21 2005-12-28 Novartis Ag Organic compounds
GB0603783D0 (en) * 2006-02-24 2006-04-05 Novartis Ag Organic compounds
CN103622962A (zh) * 2008-03-14 2014-03-12 大塚制药株式会社 制剂组合物在制备治疗以mmp-2及/或mmp-9为起因的纤维症的药物中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU550939A1 (ru) * 1975-05-19 1994-07-15 Институт химии древесины АН ЛатвССР 1,2,3,4,4а,4в,5,6,10,10а -декагидро -6- хлорацетоксиметил -1,4а-диметил -7- (1-метилэтил) -1- фенантренкарбоновая кислота или ее соли
JPH08291073A (ja) * 1995-04-22 1996-11-05 Kissei Pharmaceut Co Ltd 医薬品組成物及びその製造方法
GB0015876D0 (en) * 2000-06-28 2000-08-23 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
TWI309164B (en) 2009-05-01
CN1671731A (zh) 2005-09-21
HK1080484A1 (en) 2006-04-28
EP1554303B1 (en) 2006-12-27
PL209409B1 (pl) 2011-08-31
RU2330043C2 (ru) 2008-07-27
NZ537868A (en) 2006-11-30
PE20040722A1 (es) 2004-11-29
US7683048B2 (en) 2010-03-23
PT1554303E (pt) 2007-03-30
MXPA05001173A (es) 2005-05-16
IL184848A0 (en) 2007-12-03
JP2006501207A (ja) 2006-01-12
ES2279970T3 (es) 2007-09-01
GB0217504D0 (en) 2002-09-04
DK1554303T3 (da) 2007-04-30
ZA200500370B (en) 2006-07-26
NO20050806L (no) 2005-02-15
CA2493330A1 (en) 2004-02-12
DE60310747D1 (en) 2007-02-08
CY1106406T1 (el) 2011-10-12
CA2493330C (en) 2011-08-23
AR040692A1 (es) 2005-04-13
NZ549713A (en) 2008-04-30
EP1554303A1 (en) 2005-07-20
IL166287A0 (en) 2006-01-15
HK1080484B (en) 2007-08-03
DE60310747T2 (de) 2007-10-11
ECSP055579A (es) 2005-04-18
KR100688371B1 (ko) 2007-03-02
BR0313044A (pt) 2005-06-14
CN1305892C (zh) 2007-03-21
WO2004013156A1 (en) 2004-02-12
MY136407A (en) 2008-09-30
EP1676854A1 (en) 2006-07-05
AU2003251651B2 (en) 2007-07-12
AU2003251651A1 (en) 2004-02-23
TW200401633A (en) 2004-02-01
RU2007143025A (ru) 2009-01-20
RU2005105688A (ru) 2005-10-10
US20060166954A1 (en) 2006-07-27
PL373140A1 (en) 2005-08-22
KR20050033632A (ko) 2005-04-12
SI1554303T1 (sl) 2007-06-30
RU2348646C1 (ru) 2009-03-10

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