ATE302604T1 - Thienylazolylalkoxyethanamine, deren herstellung und deren verwendung als medikamente - Google Patents

Thienylazolylalkoxyethanamine, deren herstellung und deren verwendung als medikamente

Info

Publication number
ATE302604T1
ATE302604T1 AT99913321T AT99913321T ATE302604T1 AT E302604 T1 ATE302604 T1 AT E302604T1 AT 99913321 T AT99913321 T AT 99913321T AT 99913321 T AT99913321 T AT 99913321T AT E302604 T1 ATE302604 T1 AT E302604T1
Authority
AT
Austria
Prior art keywords
thienylazolylalkoxyethanamines
medications
production
Prior art date
Application number
AT99913321T
Other languages
English (en)
Inventor
Ramon Merce-Vidal
Blas Andaluz-Mataro
Jordi Frigola-Constansa
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Application granted granted Critical
Publication of ATE302604T1 publication Critical patent/ATE302604T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
AT99913321T 1998-04-15 1999-04-15 Thienylazolylalkoxyethanamine, deren herstellung und deren verwendung als medikamente ATE302604T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009800793A ES2150353B1 (es) 1998-04-15 1998-04-15 Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos.
PCT/ES1999/000098 WO1999052525A1 (es) 1998-04-15 1999-04-15 Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos

Publications (1)

Publication Number Publication Date
ATE302604T1 true ATE302604T1 (de) 2005-09-15

Family

ID=8303465

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99913321T ATE302604T1 (de) 1998-04-15 1999-04-15 Thienylazolylalkoxyethanamine, deren herstellung und deren verwendung als medikamente

Country Status (31)

Country Link
US (3) US6410582B1 (de)
EP (1) EP1072266B8 (de)
JP (1) JP2002511412A (de)
KR (1) KR100523366B1 (de)
CN (1) CN1189170C (de)
AR (1) AR016210A1 (de)
AT (1) ATE302604T1 (de)
AU (1) AU754705B2 (de)
BG (1) BG64891B1 (de)
BR (1) BR9910124A (de)
CA (1) CA2328878A1 (de)
CO (1) CO5011045A1 (de)
CU (1) CU22960A3 (de)
CZ (1) CZ298222B6 (de)
EE (1) EE04739B1 (de)
ES (1) ES2150353B1 (de)
GE (1) GEP20032913B (de)
HU (1) HUP0102585A3 (de)
IS (1) IS5662A (de)
LT (1) LT4830B (de)
LV (1) LV12624B (de)
NO (1) NO320313B1 (de)
NZ (1) NZ507573A (de)
PL (1) PL343512A1 (de)
RO (1) RO121690B1 (de)
RU (1) RU2213743C2 (de)
SI (1) SI20473A (de)
SK (1) SK285039B6 (de)
TW (1) TW528756B (de)
UA (1) UA58589C2 (de)
WO (1) WO1999052525A1 (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2150353B1 (es) * 1998-04-15 2001-07-01 Esteve Labor Dr Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos.
ES2137136B1 (es) * 1998-05-18 2000-07-01 Esteve Labor Dr Empleo de derivados de aril (o heteroaril) azolilcarbinoles en la elaboracion de un medicamento para el tratamiento de la inflamacion neurogenica.
ES2150378B1 (es) * 1998-08-07 2001-07-01 Esteve Labor Dr Empleo de derivados de aril(o heteroaril)azolilcarbinoles en la elaboracion de un medicamento para el tratamiento de los trastornos mediados por un exceso de substancia p.
US6432954B1 (en) * 2000-07-14 2002-08-13 Targacept, Inc. Pharmaceutical compositions and methods for use
ES2174756B2 (es) * 2001-04-06 2003-11-16 Esteve Labor Dr Derivados de aril (o heteroaril) azolilcarbinoles para el tratamiento de enfermedades respiratorias.
US20040142929A1 (en) * 2001-07-06 2004-07-22 Ramon Merce-Vidal Derivatives of aryl (or heteroaryl) azolylcarbinoles for the treatment of urinary incontinence
ES2180449B1 (es) * 2001-07-06 2004-01-16 Esteve Labor Dr Derivados de aril (o heteroaril) azolilcarbinoles para el tratamiento de la incontinencia urinaria.
CL2004001034A1 (es) 2003-05-14 2005-03-28 Teijin Pharma Ltd Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r
TW200533657A (en) * 2004-02-17 2005-10-16 Esteve Labor Dr Substituted pyrazoline compounds, their preparation and use as medicaments
EP1584335A3 (de) * 2004-04-05 2006-02-22 Laboratorios Del Dr. Esteve, S.A. Zusammensetzung aus Aktiva mit einer Carbinolverbindung und einem Opioid
US20060040924A1 (en) * 2004-06-22 2006-02-23 Laboratorios Dr. Esteve S.A. Derivatives of aryl (or heteroaryl) azolylcarbinols for the treatment of renal colic
WO2006010627A1 (en) * 2004-07-30 2006-02-02 Laboratorios Del Dr. Esteve, S.A. Aryl (or heteroaryl) azolylcarbinols
EP1632227A1 (de) * 2004-09-07 2006-03-08 Laboratorios del Dr. Esteve S.A. Aryl- (oder Heteroaryl-) Azolcarbinole (insbesondere Cizolirtin Citrate) für die Behandlung von Opioid Abhängigkeit
EP1671968A1 (de) 2004-12-17 2006-06-21 Laboratorios Del Dr. Esteve, S.A. Verfahren zur Herstellung von Enantiomeren von Thienylazolylalkoxyethanamines
EP1828175A2 (de) * 2004-12-17 2007-09-05 Laboratorios Del Dr. Esteve, S.A. Verfahren zur gewinnung von enantiomeren von thienylazolylalkoxyethanaminen
EP1674465A1 (de) * 2004-12-27 2006-06-28 Laboratorios Del Dr. Esteve, S.A. Verfahren zur Gewinnung der Enatiomeren der Thienylazolylalkoxyethanaminen
ES2303795B1 (es) * 2004-12-27 2009-06-12 Laboratorios Del Dr. Esteve, S.A. Procedimiento para obtener enantiomeros de tienilazolilalcoxietanaminas.
WO2006069767A1 (en) * 2004-12-27 2006-07-06 Laboratorios Del Dr. Esteve, S.A. Process for obtaining enantiomers of thienylazolylalcoxyethanamines
EP1757587A1 (de) * 2005-07-15 2007-02-28 Laboratorios Del Dr. Esteve, S.A. Substituierte Pyrazolinderivate, ihre Herstellung und Verwendung als Arzneimittel
EP1743892A1 (de) * 2005-07-15 2007-01-17 Laboratorios del Dr. Esteve S.A. Substituierte Pyrazolin Verbindungen, deren Herstellung und Verwendung als Medikament
EP1743890A1 (de) * 2005-07-15 2007-01-17 Laboratorios Del Dr. Esteve, S.A. 4,5-Dihydro-1H-Pyrazol-Derivative, Verfahren zur Herstellung und ihre Verwendung als Medikamente.
US7897589B2 (en) * 2005-07-15 2011-03-01 Laboratorios Del Dr. Esteve, S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
US20070149590A1 (en) * 2005-08-05 2007-06-28 Garcia Francisco J L Controlled release dosage form of pirazole compounds
EP1820502A1 (de) 2006-02-10 2007-08-22 Laboratorios Del Dr. Esteve, S.A. Wirkstoffzusammensetzungen enthaltend Azolycarbinolderivate
EP2151234A1 (de) * 2008-07-28 2010-02-10 Laboratorios Del. Dr. Esteve, S.A. Pharmazeutische Formulierung mit einer CB1-Rezeptorverbindung in einer festen Lösung und/oder festen Dispersion
CN102432845B (zh) * 2011-08-22 2013-03-13 电子科技大学 聚3,4-双乙基羟基噻吩气敏材料及其制备方法
EP3233805B1 (de) * 2014-12-15 2019-02-06 Esteve Pharmaceuticals, S.A. Methyl-1h-pyrazol-alkylamin verbindungen mit einer multimodalen aktivität gegen schmerzen

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2613720B1 (fr) * 1987-04-10 1990-01-19 Esteve Labor Dr Derives d'aryl-heteroaryl carbinols avec activite analgesique
ES2150353B1 (es) 1998-04-15 2001-07-01 Esteve Labor Dr Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos.
ES2137136B1 (es) * 1998-05-18 2000-07-01 Esteve Labor Dr Empleo de derivados de aril (o heteroaril) azolilcarbinoles en la elaboracion de un medicamento para el tratamiento de la inflamacion neurogenica.

Also Published As

Publication number Publication date
CA2328878A1 (en) 1999-10-21
NZ507573A (en) 2002-07-26
RU2213743C2 (ru) 2003-10-10
GEP20032913B (en) 2003-03-25
CN1303283A (zh) 2001-07-11
LV12624B (lv) 2001-09-20
CO5011045A1 (es) 2001-02-28
SK15282000A3 (sk) 2001-12-03
RO121690B1 (ro) 2008-02-28
HUP0102585A2 (hu) 2001-12-28
EE04739B1 (et) 2006-12-15
EE200000596A (et) 2002-06-17
US20020188017A1 (en) 2002-12-12
IS5662A (is) 2000-10-13
EP1072266A1 (de) 2001-01-31
UA58589C2 (uk) 2003-08-15
SI20473A (sl) 2001-08-31
HUP0102585A3 (en) 2002-04-29
EP1072266B1 (de) 2005-08-24
JP2002511412A (ja) 2002-04-16
CU22960A3 (es) 2004-06-21
KR20010042739A (ko) 2001-05-25
LT2000097A (en) 2001-03-26
TW528756B (en) 2003-04-21
AU3148399A (en) 1999-11-01
US20040162324A1 (en) 2004-08-19
ES2150353A1 (es) 2000-11-16
CZ20003764A3 (en) 2001-05-16
BG104853A (en) 2001-04-30
NO20005146L (no) 2000-12-14
PL343512A1 (en) 2001-08-27
CN1189170C (zh) 2005-02-16
BG64891B1 (bg) 2006-08-31
KR100523366B1 (ko) 2005-10-20
CZ298222B6 (cs) 2007-07-25
SK285039B6 (sk) 2006-05-04
BR9910124A (pt) 2001-01-09
LT4830B (lt) 2001-08-27
AR016210A1 (es) 2001-06-20
ES2150353B1 (es) 2001-07-01
LV12624A (lv) 2001-03-20
WO1999052525A1 (es) 1999-10-21
EP1072266B8 (de) 2006-10-18
NO20005146D0 (no) 2000-10-13
US7129361B2 (en) 2006-10-31
US6410582B1 (en) 2002-06-25
AU754705B2 (en) 2002-11-21
NO320313B1 (no) 2005-11-21

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