AR241185A1 - Procedimiento para la preparacion de derivados de acilaminometil-3-imidazo¡1,2-a¿piridinas. - Google Patents

Procedimiento para la preparacion de derivados de acilaminometil-3-imidazo¡1,2-a¿piridinas.

Info

Publication number
AR241185A1
AR241185A1 AR85301203A AR30120385A AR241185A1 AR 241185 A1 AR241185 A1 AR 241185A1 AR 85301203 A AR85301203 A AR 85301203A AR 30120385 A AR30120385 A AR 30120385A AR 241185 A1 AR241185 A1 AR 241185A1
Authority
AR
Argentina
Prior art keywords
formula
methyl
phenyl
alkyl
pyridines
Prior art date
Application number
AR85301203A
Other languages
English (en)
Spanish (es)
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Application granted granted Critical
Publication of AR241185A1 publication Critical patent/AR241185A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR85301203A 1984-08-07 1985-08-06 Procedimiento para la preparacion de derivados de acilaminometil-3-imidazo¡1,2-a¿piridinas. AR241185A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8412447A FR2568880B1 (fr) 1984-08-07 1984-08-07 Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
AR241185A1 true AR241185A1 (es) 1992-01-31

Family

ID=9306856

Family Applications (1)

Application Number Title Priority Date Filing Date
AR85301203A AR241185A1 (es) 1984-08-07 1985-08-06 Procedimiento para la preparacion de derivados de acilaminometil-3-imidazo¡1,2-a¿piridinas.

Country Status (23)

Country Link
US (1) US4650796A (enExample)
EP (1) EP0172096B1 (enExample)
JP (1) JPS6147485A (enExample)
KR (1) KR910004450B1 (enExample)
AR (1) AR241185A1 (enExample)
AT (1) ATE40365T1 (enExample)
AU (1) AU575190B2 (enExample)
CA (1) CA1261830A (enExample)
CZ (1) CZ357691A3 (enExample)
DE (1) DE3567867D1 (enExample)
DK (1) DK163923C (enExample)
ES (1) ES8604592A1 (enExample)
FI (1) FI80696C (enExample)
FR (1) FR2568880B1 (enExample)
GR (1) GR851928B (enExample)
HU (1) HU193799B (enExample)
IE (1) IE58347B1 (enExample)
IL (1) IL76020A (enExample)
MX (1) MX160845A (enExample)
NO (1) NO162189C (enExample)
NZ (1) NZ213013A (enExample)
PT (1) PT80921B (enExample)
ZA (1) ZA855939B (enExample)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE62687T1 (de) * 1986-01-22 1991-05-15 Synthelabo Acylaminomethylimidazo(1,2-a>pyrimidinderivate, ihre herstellung und therapeutische verwendung.
FR2593180B1 (fr) * 1986-01-22 1990-10-26 Synthelabo Derives d'acylaminomethyl-1 imidazo (1,2-a)quinoleines, leur preparation et leur application en therapeutique
FR2593818B1 (fr) * 1986-02-05 1988-04-29 Synthelabo Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
US4990506A (en) * 1986-02-05 1991-02-05 Synthelabo 3-(acylaminomethyl)imidazo[1,2-a]pyridine derivatives and their application in therapy
FR2606409B1 (fr) * 1986-11-07 1989-05-05 Synthelabo Derives d'imidazopyridine, leur preparation et leur application en therapeutique
DE3865073D1 (de) * 1987-03-27 1991-10-31 Synthelabo Imidazopyridinderivate, ihre herstellung und therapeutische verwendung.
FR2615513B1 (fr) * 1987-05-21 1989-07-13 Synthelabo Derives d'acylaminomethyl-3 tetrahydro-5,6,7,8 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
FR2654933B1 (fr) * 1989-11-30 1994-06-10 Synthelabo Utilisation d'une imidazopyridine pour la fabrication de medicaments anesthesiques.
KR910011852A (ko) * 1989-12-04 1991-08-07 폴 디. 매튜카이티스 신경독 장해 치료용 이미다조[1,2-a]피리디닐알킬 화합물
US5716964A (en) * 1989-12-04 1998-02-10 G.D. Searle & Co. Tetrazolyl substituted imidazo 1,2-a!pyridinylalkyl compounds for treatment of neurotoxic injury
IE904346A1 (en) * 1989-12-04 1991-06-05 Searle & Co IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF¹NEUROTOXIC INJURY
US5464843A (en) * 1992-06-23 1995-11-07 G.D. Searle & Co. Imidazo[1,2-a]pyridinyldiacid compounds for cognitive enhancement and for treatment of cognitive disorders and neutrotoxic injury
AUPP278498A0 (en) * 1998-04-03 1998-04-30 Australian Nuclear Science & Technology Organisation Peripheral benzodiazepine receptor binding agents
DE10019714A1 (de) * 2000-04-20 2002-01-10 Gruenenthal Gmbh Salze von bicyclischen, N-acylierten Imidazo-3-aminen und Imidazo-5-aminen
US6552037B2 (en) 2000-06-30 2003-04-22 Neurogen Corporation 2-Substituted imidazo[1,2-A]pyridine derivatives
US6596731B2 (en) 2001-03-27 2003-07-22 Hoffmann-La Roche Inc. Substituted imidazo[1,2-A] pyridine derivatives
DE10247269A1 (de) 2002-10-10 2004-04-22 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yl-methylamine
US7723324B2 (en) * 2003-10-28 2010-05-25 Sepracor, Inc. Imidazo[1,2-A]pyridine anxiolytics
WO2005081749A2 (en) * 2004-01-23 2005-09-09 Avanir Pharmaceuticals, Inc. Neutralizing human antibodies to anthraxtoxin
FR2874611B1 (fr) * 2004-08-31 2006-11-17 Servier Lab Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
MX2007005611A (es) * 2004-11-11 2007-07-11 Ferrer Int Compuestos de imidazo[1,2-a]piridina, composiciones, usos y metodos relacionados.
US8178533B2 (en) 2005-06-01 2012-05-15 Ucb Pharma, S.A. 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
EP2152262A2 (en) * 2007-04-27 2010-02-17 UCB Pharma, S.A. New heterocyclic derivatives useful for the treatment of cns disorders
AU2009249186B2 (en) 2008-05-19 2014-05-22 Sunovion Pharmaceuticals Inc. Imidazo [1, 2-a] pyridine compounds as GABA-A receptor modulators
ES2403633T3 (es) * 2008-12-04 2013-05-20 Proximagen Limited Compuestos de imidazopiridina
WO2014187922A1 (en) 2013-05-24 2014-11-27 Iomet Pharma Ltd. Slc2a transporter inhibitors
US12282014B2 (en) 2015-11-19 2025-04-22 Dana-Farber Cancer Institute, Inc. Methods of identifying compounds that interfere with ERG-driven misguidance of BAF complexes in TMPRSS2-ERG driven prostate cancers
EP3746124A4 (en) 2018-01-30 2021-10-27 Foghorn Therapeutics Inc. COMPOUNDS AND THEIR USES
US12473334B2 (en) 2018-10-17 2025-11-18 Dana-Farber Cancer Institute, Inc. SWI/SNF family chromatin remodeling complexes and uses thereof
KR102797127B1 (ko) * 2018-12-29 2025-04-21 우한 크리에이터나 사이언스 앤드 테크놀로지 컴퍼니, 리미티드 헤테로고리계 화합물, 중간체, 이의 제조 방법 및 용도
US12509453B2 (en) 2019-01-29 2025-12-30 Foghorn Therapeutics Inc. BRM/BRG1 inhibitors and uses thereof
US12384776B2 (en) 2019-01-29 2025-08-12 Foghorn Therapeutics Inc. Compounds and uses thereof
WO2021155262A1 (en) 2020-01-29 2021-08-05 Foghorn Therapeutics Inc. Compounds and uses thereof
WO2021155264A1 (en) * 2020-01-29 2021-08-05 Foghorn Therapeutics Inc. Compounds and uses thereof
US12383555B2 (en) 2020-05-20 2025-08-12 Foghorn Therapeutics Inc. Methods of treating cancers
US12606553B2 (en) 2021-03-09 2026-04-21 Foghorn Therapeutics Inc. Crystalline forms, compositions containing same, and methods of their use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB991589A (en) * 1963-04-30 1965-05-12 Selvi & C Lab Bioterapico Novel [1,2-ª‡]imidazopyridines and a process for the manufacture thereof
GB1076089A (en) * 1965-11-09 1967-07-19 Selvi & C Lab Bioterapico New derivatives of imidazo [1,2-a]-pyridine and a process for the manufacture thereof

Also Published As

Publication number Publication date
HUT38637A (en) 1986-06-30
IE58347B1 (en) 1993-09-08
KR910004450B1 (ko) 1991-06-29
FI80696B (fi) 1990-03-30
DK163923B (da) 1992-04-21
DK356885D0 (da) 1985-08-06
GR851928B (enExample) 1985-12-09
JPH0523267B2 (enExample) 1993-04-02
IL76020A (en) 1989-01-31
DK163923C (da) 1992-09-14
CA1261830A (en) 1989-09-26
EP0172096B1 (fr) 1989-01-25
IL76020A0 (en) 1985-12-31
FI853026L (fi) 1986-02-08
NO853100L (no) 1986-02-10
ES545928A0 (es) 1986-02-01
CZ357691A3 (en) 1993-06-16
NO162189C (no) 1989-11-29
DE3567867D1 (en) 1989-03-02
JPS6147485A (ja) 1986-03-07
FR2568880A1 (fr) 1986-02-14
FR2568880B1 (fr) 1986-12-12
ES8604592A1 (es) 1986-02-01
AU4580985A (en) 1986-02-13
PT80921B (pt) 1987-12-30
FI853026A0 (fi) 1985-08-06
KR860001809A (ko) 1986-03-22
AU575190B2 (en) 1988-07-21
US4650796A (en) 1987-03-17
ZA855939B (en) 1986-03-26
PT80921A (fr) 1985-09-01
FI80696C (fi) 1990-07-10
IE851937L (en) 1986-02-07
ATE40365T1 (de) 1989-02-15
MX160845A (es) 1990-05-31
NZ213013A (en) 1988-05-30
NO162189B (no) 1989-08-14
HU193799B (en) 1987-11-30
EP0172096A1 (fr) 1986-02-19
DK356885A (da) 1986-02-08

Similar Documents

Publication Publication Date Title
ES8702400A1 (es) Procedimiento para la obtencion de acidos 7-amino-1-ciclopropil-6,8-dihalogeno-1,4-dihidro-4-oxo-3-quinolincarboxilico
DK157543C (da) Pyrazolanaloge af mevalonolacton og derivater deraf samt deres anvendelse
AR240794A2 (es) Derivados de 2-(2'-nitrobenzoil)-1,3-ciclohexanodiona composicion herbicida que los comprende y procedimiento para prepararlos.
ES2033423T3 (es) Procedimientos para preparar derivados de 2-fenilpurinona.
ATE116303T1 (de) Aryl-heteroaryl-karbinol-derivate mit analgetischer aktivität.
AR240916A2 (es) "un procedimiento para la preparacion de nuevos derivados de n(fenil)amino)carbonil) bencensulfonamida".
ES8606304A1 (es) Un procedimiento para preparar derivados de tiazina
FI884132A0 (fi) 1-/ (2-pyrimidinyl) -aminoalkyl/-piperidiner, deras framstaellning och anvaendning i terapi.
DK71780A (da) Fremgangsmaade til fremstilling af difenylhydantoinderivater
DK138982A (da) Fremgangsmaade til fremstilling af bispidinderivater
ES8301220A1 (es) Procedimiento para la preparacion de derivados de imidazol
ES2028042T3 (es) Procedimiento para la obtencion de derivados de 1,8-naftiridina y fungidas que les contienen.
NO177995C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 1,3-dioksanderivater
ATE57184T1 (de) Gamma-carboline.
ES493527A0 (es) Procedimiento para la obtencion de derivados de triazo- lil-alquenos de efecto fungicida
DK247888D0 (da) Aminosyrederivater af 4-benzyl-1-(2h)-phthalazinon
DK624586A (da) 10beta-alkynyloestrenderivater og fremgangsmaade til fremstilling deraf
DK1582A (da) Substituerede thienotricycler fremgangsmaade til fremstilling deraf og anvendelse af saadanne forbindelser
ES8705421A1 (es) Un procedimiento para la preparacion de 4-amino-2-fenil-quinolinas
DE3672352D1 (de) Aminoacrylsaeure-derivate.
SE8700914D0 (sv) Anvendning av adenosinderivat
ES2038684T3 (es) Procedimiento de preparacion de derivados de octahidroindol y de compuestos intermedios de su preparacion.
ES2059550T3 (es) Derivados de la bencimidazola, su preparacion y su aplicacion en terapeutica.
ES519005A0 (es) Procedimiento para preparar 3-(1h-tetrazol-5-il)-4 (3 h)-quinazolinonas.
DE3661833D1 (de) Steroidic aromatase inhibitors