AR231976A1 - Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento - Google Patents

Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento

Info

Publication number
AR231976A1
AR231976A1 AR290473A AR29047382A AR231976A1 AR 231976 A1 AR231976 A1 AR 231976A1 AR 290473 A AR290473 A AR 290473A AR 29047382 A AR29047382 A AR 29047382A AR 231976 A1 AR231976 A1 AR 231976A1
Authority
AR
Argentina
Prior art keywords
etil
hydroxi
amino
procedure
benzolinone
Prior art date
Application number
AR290473A
Other languages
English (en)
Spanish (es)
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Application granted granted Critical
Publication of AR231976A1 publication Critical patent/AR231976A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Feed For Specific Animals (AREA)
  • Fodder In General (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR290473A 1981-09-01 1982-08-30 Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento AR231976A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813134590 DE3134590A1 (de) 1981-09-01 1981-09-01 Neue benzo-heterocyclen

Publications (1)

Publication Number Publication Date
AR231976A1 true AR231976A1 (es) 1985-04-30

Family

ID=6140603

Family Applications (2)

Application Number Title Priority Date Filing Date
AR290473A AR231976A1 (es) 1981-09-01 1982-08-30 Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento
AR294856A AR231977A1 (es) 1981-09-01 1983-11-17 Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(44)-ona y de 7-(1-hidroxi-2-amino-etil)-2-benzoxazolinona

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR294856A AR231977A1 (es) 1981-09-01 1983-11-17 Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(44)-ona y de 7-(1-hidroxi-2-amino-etil)-2-benzoxazolinona

Country Status (25)

Country Link
EP (1) EP0073505B1 (cs)
JP (1) JPS5852278A (cs)
KR (1) KR890000380B1 (cs)
AR (2) AR231976A1 (cs)
AT (1) ATE16703T1 (cs)
AU (1) AU553589B2 (cs)
CA (1) CA1180012A (cs)
CS (1) CS236679B2 (cs)
DD (1) DD204477A5 (cs)
DE (2) DE3134590A1 (cs)
DK (1) DK158664C (cs)
ES (3) ES8308318A1 (cs)
FI (1) FI78475C (cs)
GB (1) GB2106105B (cs)
GR (1) GR77275B (cs)
HU (1) HU186112B (cs)
IE (1) IE53615B1 (cs)
IL (1) IL66683A0 (cs)
NO (1) NO157738C (cs)
NZ (1) NZ201777A (cs)
PL (1) PL139375B1 (cs)
PT (1) PT75478A (cs)
SU (1) SU1149876A3 (cs)
YU (1) YU42794B (cs)
ZA (1) ZA826349B (cs)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
DE3743265A1 (de) * 1987-12-19 1989-06-29 Boehringer Ingelheim Kg Neue ammoniumverbindungen, ihre herstellung und verwendung
TW372967B (en) * 1994-12-27 1999-11-01 Kanebo Ltd 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
DE10253282A1 (de) 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung
PE20040950A1 (es) 2003-02-14 2005-01-01 Theravance Inc DERIVADOS DE BIFENILO COMO AGONISTAS DE LOS RECEPTORES ADRENERGICOS ß2 Y COMO ANTAGONISTAS DE LOS RECEPTORES MUSCARINICOS
GB0307856D0 (en) * 2003-04-04 2003-05-14 Novartis Ag Organic compounds
JP4516064B2 (ja) * 2003-04-04 2010-08-04 ノバルティス アーゲー 気道疾患の処置のためのキノリン−２−オン誘導体
WO2005110990A1 (de) * 2004-05-13 2005-11-24 Boehringer Ingelheim International Gmbh Hydroxy-substituierte benzkondensierte heterozyklen als betaagonisten zur behandlung von atemwegserkrankungen
US7307076B2 (en) 2004-05-13 2007-12-11 Boehringer Ingelheim International Gmbh Beta agonists for the treatment of respiratory diseases
US7745621B2 (en) 2004-05-14 2010-06-29 Boehringer Ingelheim International Gmbh Long acting bronchodilators for the treatment of respiratory diseases
DE102004024452A1 (de) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Aerosolformulierung für die Inhalation von Betaagonisten
DE102004024451A1 (de) 2004-05-14 2005-12-22 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pulverformulierungen für die Inhalation, die Enantiomerenreine Betaagonisten enthalten
DE102004024454A1 (de) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
DE102004024453A1 (de) * 2004-05-14 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue langwirksame Bronchodilatoren zur Behandlung von Atemwegserkrankungen
MX2008001976A (es) 2005-08-15 2008-03-25 Boehringer Ingelheim Int Procedimiento para la preparacion de betamimeticos.
TWI389692B (zh) 2005-10-10 2013-03-21 Boehringer Ingelheim Int 用以吸入β-共效劑的氣溶膠調配物
GB0602778D0 (en) 2006-02-10 2006-03-22 Glaxo Group Ltd Novel compound
WO2008017638A1 (de) * 2006-08-07 2008-02-14 Boehringer Ingelheim International Gmbh Enantiomerenreine betaagonisten, verfahren zu deren herstellung und deren verwendung als arzneimittel
UY30543A1 (es) * 2006-08-18 2008-03-31 Boehringer Ingelheim Int Formulacion de aerosol para la inhalacion de beta- agonistas
MX2009005813A (es) * 2007-01-25 2009-06-16 Boehringer Ingelheim Int Procedimiento para la preparacion de betamimeticos.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035749A1 (cs) * 1969-02-06 1970-12-24 Bellon Labor Sa Roger
CA1041523A (en) * 1974-06-19 1978-10-31 Queen's University Preparation of 1-oxapenicillins and novel intermediates therefor

Also Published As

Publication number Publication date
PT75478A (en) 1982-09-01
CS236679B2 (en) 1985-05-15
DE3134590A1 (de) 1983-03-10
NO822932L (no) 1983-03-02
PL238077A1 (en) 1984-04-09
ES8402279A1 (es) 1984-01-16
DK389082A (da) 1983-03-02
ATE16703T1 (de) 1985-12-15
DE3267702D1 (en) 1986-01-09
NO157738B (no) 1988-02-01
GR77275B (cs) 1984-09-11
GB2106105B (en) 1985-07-10
HU186112B (en) 1985-06-28
IE822105L (en) 1983-03-01
KR890000380B1 (ko) 1989-03-15
NO157738C (no) 1988-05-11
ZA826349B (en) 1984-04-25
CA1180012A (en) 1984-12-27
ES515380A0 (es) 1983-08-16
ES8405778A1 (es) 1984-06-16
GB2106105A (en) 1983-04-07
SU1149876A3 (en) 1985-04-07
EP0073505A1 (de) 1983-03-09
FI78475C (fi) 1989-08-10
YU194982A (en) 1984-12-31
ES521871A0 (es) 1984-06-16
FI822985A0 (fi) 1982-08-30
PL139375B1 (en) 1987-01-31
IE53615B1 (en) 1988-12-21
KR840001560A (ko) 1984-05-07
ES8308318A1 (es) 1983-08-16
DK158664C (da) 1991-01-14
JPH035392B2 (cs) 1991-01-25
AU8787482A (en) 1983-03-10
DD204477A5 (de) 1983-11-30
EP0073505B1 (de) 1985-11-27
FI822985L (fi) 1983-03-02
ES521870A0 (es) 1984-01-16
YU42794B (en) 1988-12-31
IL66683A0 (en) 1982-12-31
NZ201777A (en) 1985-08-30
AR231977A1 (es) 1985-04-30
FI78475B (fi) 1989-04-28
AU553589B2 (en) 1986-07-24
DK158664B (da) 1990-07-02
JPS5852278A (ja) 1983-03-28

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