ES492566A0 - Procedimiento para la preparacion de nuevos derivados de en-cafalina - Google Patents

Procedimiento para la preparacion de nuevos derivados de en-cafalina

Info

Publication number
ES492566A0
ES492566A0 ES492566A ES492566A ES492566A0 ES 492566 A0 ES492566 A0 ES 492566A0 ES 492566 A ES492566 A ES 492566A ES 492566 A ES492566 A ES 492566A ES 492566 A0 ES492566 A0 ES 492566A0
Authority
ES
Spain
Prior art keywords
cafalina
procedure
preparation
new derivatives
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES492566A
Other languages
English (en)
Other versions
ES8105720A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richardson Vicks Inc
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of ES8105720A1 publication Critical patent/ES8105720A1/es
Publication of ES492566A0 publication Critical patent/ES492566A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1024Tetrapeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
ES492566A 1979-06-21 1980-06-18 Procedimiento para la preparacion de nuevos derivados de en-cafalina Granted ES492566A0 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5095079A 1979-06-21 1979-06-21
US06/130,431 US4341698A (en) 1979-06-21 1980-03-14 Enkaphalin derivatives
AU91877/82A AU559278B2 (en) 1979-06-21 1982-12-24 Piperazines

Publications (2)

Publication Number Publication Date
ES8105720A1 ES8105720A1 (es) 1981-06-16
ES492566A0 true ES492566A0 (es) 1981-06-16

Family

ID=36764304

Family Applications (1)

Application Number Title Priority Date Filing Date
ES492566A Granted ES492566A0 (es) 1979-06-21 1980-06-18 Procedimiento para la preparacion de nuevos derivados de en-cafalina

Country Status (17)

Country Link
US (1) US4341698A (es)
AU (1) AU559278B2 (es)
CA (1) CA1161838A (es)
CH (2) CH648835A5 (es)
DE (1) DE3022401A1 (es)
DK (1) DK265780A (es)
ES (1) ES492566A0 (es)
FR (2) FR2459236A1 (es)
GB (3) GB2051821B (es)
IE (1) IE49834B1 (es)
IL (1) IL60245A (es)
IT (1) IT1148277B (es)
NL (1) NL8003580A (es)
NO (1) NO801855L (es)
NZ (1) NZ193934A (es)
PH (1) PH19222A (es)
SE (3) SE447250B (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6063794A (en) 1996-10-11 2000-05-16 Cor Therapeutics Inc. Selective factor Xa inhibitors
US6262047B1 (en) 1996-10-11 2001-07-17 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6369080B2 (en) 1996-10-11 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6194435B1 (en) 1996-10-11 2001-02-27 Cor Therapeutics, Inc. Lactams as selective factor Xa inhibitors
US6133256A (en) * 1997-04-14 2000-10-17 Cor Therapeutics Inc Selective factor Xa inhibitors
JP2002514214A (ja) 1997-04-14 2002-05-14 シーオーアール セラピューティクス インコーポレイテッド 選択的Xa因子阻害剤
EP0977772A1 (en) 1997-04-14 2000-02-09 Cor Therapeutics, Inc. SELECTIVE FACTOR Xa INHIBITORS
US6228854B1 (en) 1997-08-11 2001-05-08 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6218382B1 (en) 1997-08-11 2001-04-17 Cor Therapeutics, Inc Selective factor Xa inhibitors
US6333321B1 (en) 1997-08-11 2001-12-25 Cor Therapeutics, Inc. Selective factor Xa inhibitors
AU2006227199A1 (en) 2005-03-22 2006-09-28 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids for treating premenstrual disorders
AU2006270039B2 (en) 2005-07-19 2013-07-04 Azevan Pharmaceuticals, Inc. Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists
US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
AU2007233123A1 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Linear natriuretic peptide constructs
US8114844B2 (en) * 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
CA2647143A1 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Cyclic natriuretic peptide constructs
JP5424867B2 (ja) * 2006-03-30 2014-02-26 パラティン・テクノロジーズ・インコーポレーテッド ペプチド構築物のためのアミノ酸代用物
US8580746B2 (en) 2006-03-30 2013-11-12 Palatin Technologies, Inc. Amide linkage cyclic natriuretic peptide constructs
ES2366980T3 (es) * 2006-12-19 2011-10-27 F. Hoffmann-La Roche Ag Derivados de heteroaril-pirrolidinil- y - piperidinil-cetona.
KR20110010783A (ko) * 2008-06-18 2011-02-07 에프. 호프만-라 로슈 아게 Mri로서의 아릴 케톤
EP2587919B1 (en) 2010-07-01 2017-12-13 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
NZ724718A (en) 2014-03-28 2023-04-28 Azevan Pharmaceuticals Inc Compositions and methods for treating neurodegenerative diseases
CN111295373A (zh) 2017-09-15 2020-06-16 阿泽凡药物公司 用于治疗脑损伤的组合物和方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604845A1 (de) * 1976-02-07 1977-08-18 Knoll Ag Neue piperazinderivate
US4254107A (en) * 1979-11-27 1981-03-03 Merck & Co., Inc. Long-lasting agonists of enkephalin

Also Published As

Publication number Publication date
SE447250B (sv) 1986-11-03
DE3022401A1 (de) 1981-01-08
IT1148277B (it) 1986-11-26
CA1161838A (en) 1984-02-07
FR2459236B1 (es) 1984-01-06
NZ193934A (en) 1983-02-15
NO801855L (no) 1980-12-22
SE8500878D0 (sv) 1985-02-22
FR2459236A1 (fr) 1981-01-09
SE460540B (sv) 1989-10-23
SE8500877D0 (sv) 1985-02-22
GB2106515B (en) 1983-11-23
SE8500877L (sv) 1985-02-22
NL8003580A (nl) 1980-12-23
SE8004254L (sv) 1980-12-22
ES8105720A1 (es) 1981-06-16
GB2051821A (en) 1981-01-21
AU9187782A (en) 1983-04-21
GB2051821B (en) 1983-04-27
FR2473042A1 (fr) 1981-07-10
GB2132605B (en) 1985-01-03
GB2132605A (en) 1984-07-11
CH645363A5 (de) 1984-09-28
IT8049032A0 (it) 1980-06-20
IE49834B1 (en) 1985-12-25
IE801152L (en) 1980-12-21
PH19222A (en) 1986-02-12
DK265780A (da) 1980-12-22
US4341698A (en) 1982-07-27
AU559278B2 (en) 1987-03-05
IL60245A (en) 1985-08-30
FR2473042B1 (es) 1983-07-01
SE460541B (sv) 1989-10-23
CH648835A5 (de) 1985-04-15
GB2106515A (en) 1983-04-13

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401