SE8500878D0 - Nya enkafalinderivat - Google Patents

Nya enkafalinderivat

Info

Publication number
SE8500878D0
SE8500878D0 SE8500878A SE8500878A SE8500878D0 SE 8500878 D0 SE8500878 D0 SE 8500878D0 SE 8500878 A SE8500878 A SE 8500878A SE 8500878 A SE8500878 A SE 8500878A SE 8500878 D0 SE8500878 D0 SE 8500878D0
Authority
SE
Sweden
Prior art keywords
hydrogen
image
hydroxy
carbon atoms
group
Prior art date
Application number
SE8500878A
Other languages
English (en)
Other versions
SE460541B (sv
Inventor
A A Carr
R A Farr
J M Kane
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of SE8500878D0 publication Critical patent/SE8500878D0/sv
Publication of SE460541B publication Critical patent/SE460541B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
SE8500878A 1979-06-21 1985-02-22 Nya 6-oxo-2-piperazinkarboxylsyraestrar samt foerfarande foer framstaellning daerav SE460541B (sv)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5095079A 1979-06-21 1979-06-21
US06/130,431 US4341698A (en) 1979-06-21 1980-03-14 Enkaphalin derivatives
AU91877/82A AU559278B2 (en) 1979-06-21 1982-12-24 Piperazines

Publications (2)

Publication Number Publication Date
SE8500878D0 true SE8500878D0 (sv) 1985-02-22
SE460541B SE460541B (sv) 1989-10-23

Family

ID=36764304

Family Applications (3)

Application Number Title Priority Date Filing Date
SE8004254A SE447250B (sv) 1979-06-21 1980-06-06 Nya enkafalinderivat
SE8500877A SE460540B (sv) 1979-06-21 1985-02-22 Nya 2-oxopiperazinfoereningar samt foerfarande foer framstaellning daerav
SE8500878A SE460541B (sv) 1979-06-21 1985-02-22 Nya 6-oxo-2-piperazinkarboxylsyraestrar samt foerfarande foer framstaellning daerav

Family Applications Before (2)

Application Number Title Priority Date Filing Date
SE8004254A SE447250B (sv) 1979-06-21 1980-06-06 Nya enkafalinderivat
SE8500877A SE460540B (sv) 1979-06-21 1985-02-22 Nya 2-oxopiperazinfoereningar samt foerfarande foer framstaellning daerav

Country Status (17)

Country Link
US (1) US4341698A (sv)
AU (1) AU559278B2 (sv)
CA (1) CA1161838A (sv)
CH (2) CH645363A5 (sv)
DE (1) DE3022401A1 (sv)
DK (1) DK265780A (sv)
ES (1) ES492566A0 (sv)
FR (2) FR2459236A1 (sv)
GB (3) GB2051821B (sv)
IE (1) IE49834B1 (sv)
IL (1) IL60245A (sv)
IT (1) IT1148277B (sv)
NL (1) NL8003580A (sv)
NO (1) NO801855L (sv)
NZ (1) NZ193934A (sv)
PH (1) PH19222A (sv)
SE (3) SE447250B (sv)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6262047B1 (en) 1996-10-11 2001-07-17 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6063794A (en) 1996-10-11 2000-05-16 Cor Therapeutics Inc. Selective factor Xa inhibitors
US6369080B2 (en) 1996-10-11 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6194435B1 (en) 1996-10-11 2001-02-27 Cor Therapeutics, Inc. Lactams as selective factor Xa inhibitors
NZ500353A (en) 1997-04-14 2002-02-01 Cor Therapeutics Inc Cyclic diaza compounds that are selective inhibitors of factor Xa
EP0977773A1 (en) 1997-04-14 2000-02-09 Cor Therapeutics, Inc. SELECTIVE FACTOR Xa INHIBITORS
US6133256A (en) * 1997-04-14 2000-10-17 Cor Therapeutics Inc Selective factor Xa inhibitors
US6333321B1 (en) 1997-08-11 2001-12-25 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6218382B1 (en) 1997-08-11 2001-04-17 Cor Therapeutics, Inc Selective factor Xa inhibitors
US6228854B1 (en) 1997-08-11 2001-05-08 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US9597314B2 (en) 2005-03-22 2017-03-21 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids for treating premenstrual disorders
AU2006270039B2 (en) 2005-07-19 2013-07-04 Azevan Pharmaceuticals, Inc. Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists
US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
DK2001518T3 (da) * 2006-03-30 2013-10-07 Palatin Technologies Inc Cykliske natriuretiske peptidfremstillinger
US8580746B2 (en) 2006-03-30 2013-11-12 Palatin Technologies, Inc. Amide linkage cyclic natriuretic peptide constructs
US8114844B2 (en) * 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
AU2007233105B2 (en) * 2006-03-30 2013-05-16 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
AU2007233123A1 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Linear natriuretic peptide constructs
CN101563319B (zh) * 2006-12-19 2012-09-05 弗·哈夫曼-拉罗切有限公司 杂芳基吡咯烷基和哌啶基甲酮衍生物
BRPI0914160A2 (pt) * 2008-06-18 2019-09-24 Hoffmann La Roche aril cetona como mri
CN103269584B (zh) 2010-07-01 2017-05-03 阿泽凡药物公司 用于治疗创伤后应激障碍的方法
MX2016012645A (es) 2014-03-28 2017-01-11 Azevan Pharmaceuticals Inc Composiciones y metodos para tratar enfermedades neurodegenerativas.
WO2019055913A1 (en) 2017-09-15 2019-03-21 Azevan Pharmaceuticals, Inc. COMPOSITIONS AND METHODS FOR TREATMENT OF BRAIN INJURY

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604845A1 (de) * 1976-02-07 1977-08-18 Knoll Ag Neue piperazinderivate
US4254107A (en) * 1979-11-27 1981-03-03 Merck & Co., Inc. Long-lasting agonists of enkephalin

Also Published As

Publication number Publication date
GB2051821A (en) 1981-01-21
SE8500877D0 (sv) 1985-02-22
FR2473042A1 (fr) 1981-07-10
FR2459236A1 (fr) 1981-01-09
AU9187782A (en) 1983-04-21
US4341698A (en) 1982-07-27
FR2473042B1 (sv) 1983-07-01
GB2132605A (en) 1984-07-11
CH648835A5 (de) 1985-04-15
SE8500877L (sv) 1985-02-22
PH19222A (en) 1986-02-12
SE460541B (sv) 1989-10-23
IT8049032A0 (it) 1980-06-20
CA1161838A (en) 1984-02-07
GB2106515A (en) 1983-04-13
IT1148277B (it) 1986-11-26
IE801152L (en) 1980-12-21
NL8003580A (nl) 1980-12-23
GB2132605B (en) 1985-01-03
GB2106515B (en) 1983-11-23
AU559278B2 (en) 1987-03-05
ES8105720A1 (es) 1981-06-16
IE49834B1 (en) 1985-12-25
GB2051821B (en) 1983-04-27
NO801855L (no) 1980-12-22
CH645363A5 (de) 1984-09-28
SE8004254L (sv) 1980-12-22
FR2459236B1 (sv) 1984-01-06
ES492566A0 (es) 1981-06-16
SE447250B (sv) 1986-11-03
DK265780A (da) 1980-12-22
IL60245A (en) 1985-08-30
SE460540B (sv) 1989-10-23
NZ193934A (en) 1983-02-15
DE3022401A1 (de) 1981-01-08

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