AR222797A1 - Procedimiento para preparar compuestos de n-ciano-n'(2-(4-metil-5-imidazolil)-metiltio-etil)-n''alquilnilguanidinas y sus sales - Google Patents

Procedimiento para preparar compuestos de n-ciano-n'(2-(4-metil-5-imidazolil)-metiltio-etil)-n''alquilnilguanidinas y sus sales

Info

Publication number
AR222797A1
AR222797A1 AR272401A AR27240178A AR222797A1 AR 222797 A1 AR222797 A1 AR 222797A1 AR 272401 A AR272401 A AR 272401A AR 27240178 A AR27240178 A AR 27240178A AR 222797 A1 AR222797 A1 AR 222797A1
Authority
AR
Argentina
Prior art keywords
metithyl
alkyllnylguanidines
ciano
imidazolyl
salts
Prior art date
Application number
AR272401A
Other languages
English (en)
Spanish (es)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/848,959 external-priority patent/US4112234A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Application granted granted Critical
Publication of AR222797A1 publication Critical patent/AR222797A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/39Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
    • C07C323/43Y being a hetero atom
    • C07C323/44X or Y being nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR272401A 1977-06-03 1978-05-31 Procedimiento para preparar compuestos de n-ciano-n'(2-(4-metil-5-imidazolil)-metiltio-etil)-n''alquilnilguanidinas y sus sales AR222797A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US80300977A 1977-06-03 1977-06-03
US82679677A 1977-08-22 1977-08-22
US05/848,959 US4112234A (en) 1977-08-22 1977-11-07 Imidazolylmethylthioethyl alkynyl guanidines

Publications (1)

Publication Number Publication Date
AR222797A1 true AR222797A1 (es) 1981-06-30

Family

ID=27419995

Family Applications (2)

Application Number Title Priority Date Filing Date
AR272401A AR222797A1 (es) 1977-06-03 1978-05-31 Procedimiento para preparar compuestos de n-ciano-n'(2-(4-metil-5-imidazolil)-metiltio-etil)-n''alquilnilguanidinas y sus sales
AR278645A AR222503A1 (es) 1977-06-03 1979-10-26 Nuevos derivados de n-ciano-n'-alquinil(c3-c9)-iso ioureas s-sustituidas,utiles para preparar compuestos de n-ciano-n'-alquinil(c3-c9)-isotioureas lil)metiltio)-etil-n"-alquinil(c3-c9)-guanidinas y procedimientos para obtener dichas guanidinas y sus sales

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR278645A AR222503A1 (es) 1977-06-03 1979-10-26 Nuevos derivados de n-ciano-n'-alquinil(c3-c9)-iso ioureas s-sustituidas,utiles para preparar compuestos de n-ciano-n'-alquinil(c3-c9)-isotioureas lil)metiltio)-etil-n"-alquinil(c3-c9)-guanidinas y procedimientos para obtener dichas guanidinas y sus sales

Country Status (26)

Country Link
JP (1) JPS543067A (xx)
AR (2) AR222797A1 (xx)
CA (1) CA1110251A (xx)
CH (2) CH641167A5 (xx)
CY (3) CY1229A (xx)
DD (1) DD140038A5 (xx)
DE (1) DE2824066A1 (xx)
DK (1) DK243178A (xx)
ES (3) ES470474A1 (xx)
FI (1) FI69069C (xx)
FR (2) FR2401143A1 (xx)
GB (3) GB1598628A (xx)
GR (1) GR73860B (xx)
HK (3) HK38284A (xx)
HU (1) HU186766B (xx)
IE (1) IE47543B1 (xx)
IL (1) IL54819A (xx)
KE (1) KE3373A (xx)
LU (1) LU79725A1 (xx)
MY (3) MY8500452A (xx)
NL (1) NL7805935A (xx)
NO (3) NO152214C (xx)
NZ (1) NZ187376A (xx)
SE (3) SE443784B (xx)
SG (1) SG8584G (xx)
YU (4) YU129778A (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS568352A (en) * 1979-07-03 1981-01-28 Shionogi & Co Ltd Aminoalkylvenzene derivative
US4339439A (en) * 1981-01-19 1982-07-13 Bristol-Myers Company Pharmaceutical methods and compositions
JPS57134318A (en) * 1981-02-12 1982-08-19 Nissan Motor Co Ltd Air mixing construction of air conditioner
JPS5848516U (ja) * 1981-09-30 1983-04-01 日産車体株式会社 車両用空気調和装置
JPS6018010U (ja) * 1983-07-18 1985-02-07 日産自動車株式会社 車両用空気調和装置の温度調整機構
JPS60113211U (ja) * 1984-01-06 1985-07-31 松下電器産業株式会社 自動車用空気調和装置
ES2007948A6 (es) * 1988-07-06 1989-07-01 Vinas Lab Procedimiento para la obtencion de derivados propargilguanidicos.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4024271A (en) * 1971-03-09 1977-05-17 Smith Kline & French Laboratories Limited Pharmacologically active guanidine compounds
GB1338169A (en) * 1971-03-09 1973-11-21 Smith Kline French Lab Ureas thioureas and guanidines
GB1397436A (en) * 1972-09-05 1975-06-11 Smith Kline French Lab Heterocyclic n-cyanoguinidines
GB1531221A (en) * 1974-09-02 1978-11-08 Smith Kline French Lab Process for preparing guanidine derivatives
GB1533380A (en) * 1974-09-02 1978-11-22 Smith Kline French Lab Process for the preparation of heterocyclic substituted thioureas and h-cyanoguanidines
GB1531231A (en) * 1974-09-02 1978-11-08 Smith Kline French Lab Process for the production of cyanoguanidine derivatives

Also Published As

Publication number Publication date
CA1110251A (en) 1981-10-06
YU215582A (en) 1983-02-28
SG8584G (en) 1985-02-08
LU79725A1 (fr) 1979-02-02
IL54819A (en) 1983-03-31
DK243178A (da) 1978-12-04
DE2824066A1 (de) 1978-12-14
CY1231A (en) 1984-06-29
NO791637L (no) 1978-12-05
HK38084A (en) 1984-05-11
YU215482A (en) 1983-02-28
SE8401492L (sv) 1984-03-16
DD140038A5 (de) 1980-02-06
NL7805935A (nl) 1978-12-05
FI69069B (fi) 1985-08-30
MY8500451A (en) 1985-12-31
NO152214B (no) 1985-05-13
KE3373A (en) 1984-03-23
IE47543B1 (en) 1984-04-18
SE7806525A (sv) 1978-12-04
CY1229A (en) 1984-06-29
SE7806525L (sv) 1978-12-04
SE8401492D0 (sv) 1984-03-16
ES478202A1 (es) 1979-06-01
SE8401491L (sv) 1984-03-16
JPS5639313B2 (xx) 1981-09-11
HK38284A (en) 1984-05-11
IL54819A0 (en) 1978-07-31
MY8500453A (en) 1985-12-31
GB1598628A (en) 1981-09-23
YU41620B (en) 1987-12-31
YU53079A (en) 1983-09-30
YU40625B (en) 1986-02-28
CH641167A5 (en) 1984-02-15
FI781737A (fi) 1978-12-04
NO151824C (no) 1985-06-12
NO152214C (no) 1985-08-28
JPS543067A (en) 1979-01-11
YU129778A (en) 1983-02-28
GR73860B (xx) 1984-05-08
HU186766B (en) 1985-09-30
NO781928L (no) 1978-12-05
IE781112L (en) 1978-12-03
NZ187376A (en) 1981-05-29
ES470474A1 (es) 1979-09-01
MY8500452A (en) 1985-12-31
CH644591A5 (en) 1984-08-15
NO151824B (no) 1985-03-04
FR2436138A1 (fr) 1980-04-11
FR2401143A1 (fr) 1979-03-23
HK38184A (en) 1984-05-11
YU40624B (en) 1986-02-28
AR222503A1 (es) 1981-05-29
FR2436138B1 (xx) 1982-12-03
SE443784B (sv) 1986-03-10
FI69069C (fi) 1985-12-10
ES478203A1 (es) 1979-06-01
NO833255L (no) 1978-12-05
GB1598629A (en) 1981-09-23
GB1598630A (en) 1981-09-23
CY1230A (en) 1984-06-29
FR2401143B1 (xx) 1981-12-11
SE8401491D0 (sv) 1984-03-16

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