AR080271A2 - Proceso para la preparacion de derivados de fenilpropargileter - Google Patents

Proceso para la preparacion de derivados de fenilpropargileter

Info

Publication number
AR080271A2
AR080271A2 ARP100102586A ARP100102586A AR080271A2 AR 080271 A2 AR080271 A2 AR 080271A2 AR P100102586 A ARP100102586 A AR P100102586A AR P100102586 A ARP100102586 A AR P100102586A AR 080271 A2 AR080271 A2 AR 080271A2
Authority
AR
Argentina
Prior art keywords
carbon atoms
compound
formula
halogen
group
Prior art date
Application number
ARP100102586A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35098316&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR080271(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR080271A2 publication Critical patent/AR080271A2/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/02Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/12Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/02Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/34Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/02Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups
    • C07C251/04Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/10Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • C07C251/16Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/01Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/37Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by etherified hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00Preparation of sulfones; Preparation of sulfoxides
    • C07C315/04Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C07C319/20Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/46Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/58Unsaturated compounds containing ether groups, groups, groups, or groups
    • C07C59/64Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
    • C07C59/66Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings
    • C07C59/68Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
    • C07C59/70Ethers of hydroxy-acetic acid, e.g. substitutes on the ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/734Ethers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se revela un proceso para la preparacion de un compuesto de formula (1) donde R es un grupo alquinilo; R1 es alquilo, alquenilo, alquinilo, cicloalquilo, cicloalquilo-alquilo, fenilo y fenilalquilo, siendo posible a su vez para todos los grupos anteriores portar uno o más de átomos de halogeno iguales o diferentes; alcoxi; alqueniloxi; alquiniloxi; alcoxialquilo; haloalcoxi; alquiltio; haloalquiltio; alquilsulfonilo; formilo; alcanoílo; hidroxi; halogeno; ciano; nitro; amino; alquilamino; dialquilamino; carboxilo; alcoxicarbonilo; alqueniloxicarbonilo; o alquiniloxicarbonilo; y n es un entero de 0 a 3, dicho proceso que comprende: (i) la reaccion de un compuesto de formula (3) donde R, R1 y n son segun se definio en la presente anteriormente; m y m' son independientemente 0 o 1; cuando m y m' son ambos 0, A es un grupo alquilo, alquenilo o alquinilo (que tiene convenientemente hasta ocho átomos de carbono), opcionalmente sustituido con uno o más grupos independientemente seleccionados de halogeno, hidroxi, alcoxi, dialquilamino C1-4 o ciano; cuando uno de m y m' es 0 y el otro es 1, A es un grupo alcanodiílo, alquenodiílo o alquinodiílo que contiene al menos dos átomos de carbono (y tiene convenientemente hasta ocho átomos de carbono), opcionalmente sustituido con uno o más grupos independientemente seleccionados de halogeno, hidroxi, alcoxi, dialquilamino C1-4 o ciano; cuando m y m' son ambos 1, A es un grupo alcanotriílo, alquenotriílo o alquinotriílo que contiene al menos tres átomos de carbono (y tiene convenientemente hasta ocho átomos de carbono), opcionalmente sustituido con uno o más grupos independientemente seleccionados de halogeno, hidroxi, alcoxi, dialquilamino C1-4 o ciano; y donde si el grupo A contiene tres o más átomos de carbono, uno o más de los átomos de carbono puede estar cada uno de ellos opcionalmente reemplazado con un átomo de oxígeno, siempre que exista al menos un átomo de carbono entre cualquiera de los átomos de oxígeno en la molécula, con un compuesto de formula (4) para dar un compuesto de formula (2) donde R, R1 y n son segun se definio en la presente anteriormente, y (ii) la reaccion de un compuesto de formula (2) L--s, con donde L es un grupo saliente, para dar el compuesto de formula (1) segun se definio en la presente anteriormente.
ARP100102586A 2005-08-15 2010-07-15 Proceso para la preparacion de derivados de fenilpropargileter AR080271A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0516705.1A GB0516705D0 (en) 2005-08-15 2005-08-15 Process

Publications (1)

Publication Number Publication Date
AR080271A2 true AR080271A2 (es) 2012-03-28

Family

ID=35098316

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP060103483A AR057741A1 (es) 2005-08-15 2006-08-09 Proceso para la preparacion de derivados de fenilpropargileter
ARP100102586A AR080271A2 (es) 2005-08-15 2010-07-15 Proceso para la preparacion de derivados de fenilpropargileter

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP060103483A AR057741A1 (es) 2005-08-15 2006-08-09 Proceso para la preparacion de derivados de fenilpropargileter

Country Status (26)

Country Link
US (1) US8129560B2 (es)
EP (1) EP1919857B1 (es)
JP (1) JP5350790B2 (es)
KR (1) KR101305928B1 (es)
CN (1) CN101243040B (es)
AR (2) AR057741A1 (es)
AU (1) AU2006281293B2 (es)
BR (1) BRPI0616593B1 (es)
CA (1) CA2619435C (es)
CR (1) CR9710A (es)
EC (1) ECSP088183A (es)
ES (1) ES2572137T3 (es)
GB (1) GB0516705D0 (es)
GT (1) GT200600369A (es)
HN (1) HN2006029142A (es)
HU (1) HUE028929T2 (es)
IL (3) IL188919A (es)
MX (1) MX2008001794A (es)
MY (1) MY150654A (es)
NZ (1) NZ574781A (es)
PL (1) PL1919857T3 (es)
RU (1) RU2470914C9 (es)
TW (2) TWI428314B (es)
UA (1) UA90810C2 (es)
WO (1) WO2007020381A2 (es)
ZA (1) ZA200800691B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0808764D0 (en) * 2008-05-14 2008-06-18 Syngenta Ltd Process
JP5747625B2 (ja) 2011-04-12 2015-07-15 住友化学株式会社 マンデロニトリル化合物の製造方法
WO2013113776A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
AU2013214353A1 (en) 2012-02-03 2014-08-21 Basf Se Fungicidal pyrimidine compounds
WO2013113716A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113778A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113720A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013113773A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
EA201491472A1 (ru) 2012-02-03 2015-01-30 Басф Се Фунгицидные соединения пиримидина
WO2013113791A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
CN110204556B (zh) * 2019-07-16 2020-09-18 重庆医药高等专科学校 (rs)-甲氧基头孢西丁的制备方法
WO2023044364A1 (en) 2021-09-15 2023-03-23 Enko Chem, Inc. Protoporphyrinogen oxidase inhibitors
JP2025541336A (ja) 2022-12-16 2025-12-18 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト 改良された殺有害生物組成物

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GB1030756A (en) * 1963-04-01 1966-05-25 Boots Pure Drug Co Ltd Anti-inflammatory compositions comprising biphenylyl-alkane derivatives
US3393192A (en) 1965-04-26 1968-07-16 Schering Corp Novel benzazepines
DK133742B (da) 1970-10-30 1976-07-12 Merck & Co Inc Fremgangsmåde til fremstilling af 2-acetamidoethyl-(3-trifluormethylphenoxy)-(4-chlorphenyl)-acetat.
FR2120246A5 (es) * 1970-12-03 1972-08-18 Micsunescu Francine
FR2131802A7 (en) * 1971-03-11 1972-11-17 Micsunescu Francine Galvanizing bath brigenting agents - produced by reacting aromatic aldehydes or ketones with acetylenic alcohols
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GT199800109A (es) * 1997-08-06 2000-01-13 Derivados de n-sulfonilglicinalquiniloxifenetilamida microbicidas.
GB9804265D0 (en) * 1998-02-27 1998-04-22 Ciba Geigy Ag Organic compounds
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GB0011944D0 (en) * 2000-05-17 2000-07-05 Novartis Ag Organic compounds
GB0108339D0 (en) * 2001-04-03 2001-05-23 Syngenta Participations Ag Organics compounds
GB0127554D0 (en) * 2001-11-16 2002-01-09 Syngenta Participations Ag Organic compounds
GB0127559D0 (en) * 2001-11-16 2002-01-09 Syngenta Participations Ag Organic compounds
AU2003255004A1 (en) * 2002-08-19 2004-03-03 Sumitomo Chemical Company, Limited Phenylpyridine compound and bactericidal composition containing the same
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Also Published As

Publication number Publication date
MX2008001794A (es) 2008-04-07
IL188919A0 (en) 2008-08-07
CN101243040A (zh) 2008-08-13
BRPI0616593A2 (pt) 2011-06-28
US20090118532A1 (en) 2009-05-07
TW201332944A (zh) 2013-08-16
ES2572137T3 (es) 2016-05-30
HN2006029142A (es) 2010-08-19
WO2007020381A3 (en) 2007-05-03
IL226403A0 (en) 2013-06-27
TWI399363B (zh) 2013-06-21
GB0516705D0 (en) 2005-09-21
KR101305928B1 (ko) 2013-09-12
PL1919857T3 (pl) 2016-10-31
MY150654A (en) 2014-02-14
CR9710A (es) 2008-04-16
TWI428314B (zh) 2014-03-01
HUE028929T2 (en) 2017-01-30
NZ574781A (en) 2011-06-30
CA2619435A1 (en) 2007-02-22
CA2619435C (en) 2014-02-18
ZA200800691B (en) 2011-12-28
RU2008110063A (ru) 2009-09-27
EP1919857B1 (en) 2016-03-09
EP1919857A2 (en) 2008-05-14
RU2470914C9 (ru) 2016-05-20
TW200720230A (en) 2007-06-01
KR20080034934A (ko) 2008-04-22
JP5350790B2 (ja) 2013-11-27
JP2009504715A (ja) 2009-02-05
IL226404A0 (en) 2013-06-27
IL188919A (en) 2015-04-30
AU2006281293A1 (en) 2007-02-22
ECSP088183A (es) 2008-03-26
WO2007020381A2 (en) 2007-02-22
US8129560B2 (en) 2012-03-06
CN101243040B (zh) 2012-12-05
AR057741A1 (es) 2007-12-12
AU2006281293B2 (en) 2011-04-28
GT200600369A (es) 2007-09-19
RU2470914C2 (ru) 2012-12-27
UA90810C2 (ru) 2010-05-25
BRPI0616593B1 (pt) 2017-06-27

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