AR079536A1 - Granulos para preparaciones farmaceuticas, metodo y aparato para su produccion - Google Patents

Granulos para preparaciones farmaceuticas, metodo y aparato para su produccion

Info

Publication number
AR079536A1
AR079536A1 ARP100104755A ARP100104755A AR079536A1 AR 079536 A1 AR079536 A1 AR 079536A1 AR P100104755 A ARP100104755 A AR P100104755A AR P100104755 A ARP100104755 A AR P100104755A AR 079536 A1 AR079536 A1 AR 079536A1
Authority
AR
Argentina
Prior art keywords
granules
pharmaceutical
pharmaceutical preparation
active ingredient
ingredient
Prior art date
Application number
ARP100104755A
Other languages
English (en)
Original Assignee
Ferring Int Ct Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42110308&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR079536(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ferring Int Ct Sa filed Critical Ferring Int Ct Sa
Publication of AR079536A1 publication Critical patent/AR079536A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • A61K31/609Amides, e.g. salicylamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1694Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Reivindicacion 1: Una preparacion farmacéutica que comprende gránulos de los cuales cada uno tiene un ingrediente activo farmacéutico y de los cuales cada uno tiene un eje predeterminado y el mismo perfil transversal predeterminado, en donde por lo menos 80% en cantidad de estos gránulos tienen una proporcion de aspecto menor de 2.2. Reivindicacion 8: La preparacion farmacéutica de cualquier reivindicacion precedente, en donde el ingrediente activo farmacéutico comprende un ingrediente anti-inflamatorio. Reivindicacion 9: La preparacion farmacéutica de cualquier reivindicacion precedente, en donde el ingrediente activo farmacéutico es 5-ácido aminosalicílico. Reivindicacion 20: El uso de un separador de longitud en un método para producir una preparacion farmacéutica, en donde el uso ocurre durante la seleccion de gránulos de los cuales cada uno tiene un eje predeterminado y el mismo perfil transversal predeterminado y del cual por lo menos una cantidad tiene un ingrediente activo farmacéutico.
ARP100104755A 2009-12-18 2010-12-20 Granulos para preparaciones farmaceuticas, metodo y aparato para su produccion AR079536A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09179877A EP2340812A1 (en) 2009-12-18 2009-12-18 Granules for pharmaceutical preparations, methods and apparatus for their production

Publications (1)

Publication Number Publication Date
AR079536A1 true AR079536A1 (es) 2012-02-01

Family

ID=42110308

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100104755A AR079536A1 (es) 2009-12-18 2010-12-20 Granulos para preparaciones farmaceuticas, metodo y aparato para su produccion

Country Status (27)

Country Link
US (2) US8765185B2 (es)
EP (2) EP2340812A1 (es)
JP (1) JP5593396B2 (es)
KR (1) KR101882880B1 (es)
CN (2) CN105769772A (es)
AR (1) AR079536A1 (es)
AU (1) AU2010332884B2 (es)
BR (1) BR112012014935B1 (es)
CA (1) CA2784235C (es)
DK (1) DK2512453T3 (es)
ES (1) ES2612870T3 (es)
HR (1) HRP20161639T1 (es)
HU (1) HUE031228T2 (es)
IL (1) IL220319A (es)
JO (1) JO3762B1 (es)
LT (1) LT2512453T (es)
MX (2) MX2012006851A (es)
NL (1) NL1038373C2 (es)
NZ (1) NZ600582A (es)
PL (1) PL2512453T3 (es)
PT (1) PT2512453T (es)
RS (1) RS55438B1 (es)
RU (1) RU2584349C2 (es)
SI (1) SI2512453T1 (es)
TW (1) TWI511723B (es)
WO (1) WO2011073245A2 (es)
ZA (1) ZA201204441B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2520197A1 (en) 2003-04-23 2004-11-04 Ferring B.V. Sachet for a pharmaceutical composition
DK3628319T3 (da) 2008-10-02 2024-03-04 Salix Pharmaceuticals Ltd Behandling af hepatisk encefalopati ved anvendelse af rifaximin
EP2340812A1 (en) 2009-12-18 2011-07-06 Ferring International Center S.A. Granules for pharmaceutical preparations, methods and apparatus for their production
US20140141075A1 (en) 2012-11-21 2014-05-22 Warner Chilcott Company, Llc 5-aminosalicylic acid capsule formulation
DE202017102645U1 (de) * 2017-05-03 2018-08-06 Romaco Kilian Gmbh Ablaufvorrichtung für Presslinge einer Rundläufer-Tablettenpresse sowie Rundläufer-Tablettenpresse mit Ablaufvorrichtung
RU2667637C1 (ru) * 2017-06-26 2018-09-21 Гермес Арцнаймиттель ГмбХ Фармацевтическая композиция для перорального применения, содержащая n-ацетилцистеин с маскированным вкусом
ES2938608T3 (es) 2017-09-20 2023-04-13 Tillotts Pharma Ag Método para preparar una forma farmacéutica sólida que comprende anticuerpos mediante granulación en húmedo, extrusión y esferonización
ES2938609T3 (es) 2017-09-20 2023-04-13 Tillotts Pharma Ag Preparación de formas farmacéuticas sólidas que comprenden anticuerpos mediante estratificación de solución/suspensión
EP3459529A1 (en) 2017-09-20 2019-03-27 Tillotts Pharma Ag Preparation of sustained release solid dosage forms comprising antibodies by spray drying
KR102161235B1 (ko) * 2020-07-22 2020-09-29 주식회사 피티케이 이송 일체형 과립 제조 장치 및 방법
CN114472139A (zh) * 2022-01-04 2022-05-13 安徽宏信药业发展有限公司 一种中药药丸干燥筛选装置
CN115445902B (zh) * 2022-09-21 2023-06-06 重庆科技学院 一种条形颗粒物三维尺寸分选方法及装置
CN116942532B (zh) * 2023-09-20 2023-12-12 北京爱力佳医药科技有限公司 一种粉状药物制备装置

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57500432A (es) 1980-03-20 1982-03-11
US4720473A (en) * 1986-03-10 1988-01-19 Cri International, Inc. Production of improved catalyst-type particles using length and density grading
CA1294943C (en) * 1986-03-10 1992-01-28 J. Gary Welch Production of improved catalyst-type particles using length and density grading
JPH0827133B2 (ja) 1993-07-13 1996-03-21 不二パウダル株式会社 湿潤粉粒体の処理装置
HU228856B1 (en) 1995-12-21 2013-06-28 Ferring Farma Lab Modified release oral pharmaceutical composition containing 5-asa for the treatment of bowel diseases
US6004581A (en) 1995-12-21 1999-12-21 Farmaceutisk Laboratorium Ferring A/S Modified release oral pharmaceutical composition and method for the treatment of bowel diseases
AUPO637197A0 (en) 1997-04-23 1997-05-15 F.H. Faulding & Co. Limited Taste-masked pharmaceutical compositions
DE19724181A1 (de) * 1997-06-09 1998-12-10 Bayer Ag Multiple-unit-retard-Zubereitungen und Verfahren zu ihrer Herstellung
JP2000128774A (ja) 1998-10-26 2000-05-09 Tanabe Seiyaku Co Ltd 薬物を含有する球形微粒子の製法
US6146685A (en) 1998-11-05 2000-11-14 Delsys Pharmaceutical Corporation Method of deposition a dry powder and dispensing device
CA2360655C (en) * 1999-01-29 2007-03-20 Losan Pharma Gmbh Pharmaceutical compositions
US6735487B1 (en) 1999-07-01 2004-05-11 Ods Properties, Inc. Interactive wagering system with promotions
GB0113841D0 (en) * 2001-06-07 2001-08-01 Boots Co Plc Therapeutic agents
AR036797A1 (es) 2001-10-15 2004-10-06 Ferring Bv Un metodo para preparar una composicion farmaceutica que comprende acido 5-aminosalicilico para utilizar en el tratamiento de colitis ulcerosa y enfermedades de crohn
DE60130270T2 (de) 2001-10-15 2008-05-29 Ferring B.V. Verfahren zur herstellung einer pharmazeutischen zubereitung mit 5-aminosalicylsäure zur verwendung bei der behandlung von colitis ulcerosa und morbus crohn
US7445796B2 (en) 2002-08-19 2008-11-04 L. Perrigo Company Pharmaceutically active particles of a monomodal particle size distribution and method
EP1470819A1 (en) * 2003-04-23 2004-10-27 Ferring B.V. High drug load mesalazine sachet
CA2520197A1 (en) 2003-04-23 2004-11-04 Ferring B.V. Sachet for a pharmaceutical composition
EP1547601A1 (en) * 2003-12-23 2005-06-29 Ferring B.V. Coating method
US7207505B2 (en) 2004-06-04 2007-04-24 Bender Martin P Method for producing small granules
DE102004028977A1 (de) * 2004-06-16 2006-01-05 Add Advanced Drug Delivery Technologies Ltd. Neutralpellets
WO2007061717A2 (en) 2005-11-17 2007-05-31 Teva Pharmaceutical Industries, Ltd. Methods for isolating propargylated aminoindans
EP2340812A1 (en) 2009-12-18 2011-07-06 Ferring International Center S.A. Granules for pharmaceutical preparations, methods and apparatus for their production

Also Published As

Publication number Publication date
US20130022681A1 (en) 2013-01-24
EP2512453A2 (en) 2012-10-24
CN105769772A (zh) 2016-07-20
NZ600582A (en) 2014-09-26
BR112012014935B1 (pt) 2021-12-21
TW201125556A (en) 2011-08-01
EP2340812A1 (en) 2011-07-06
LT2512453T (lt) 2016-12-27
MX351365B (es) 2017-10-12
RU2584349C2 (ru) 2016-05-20
US8765185B2 (en) 2014-07-01
ZA201204441B (en) 2013-02-27
MX2012006851A (es) 2012-08-31
WO2011073245A2 (en) 2011-06-23
IL220319A (en) 2016-03-31
PT2512453T (pt) 2016-12-16
TWI511723B (zh) 2015-12-11
ES2612870T3 (es) 2017-05-19
CA2784235C (en) 2019-01-15
KR101882880B1 (ko) 2018-07-27
CN102791257B (zh) 2017-03-01
CA2784235A1 (en) 2011-06-23
JP5593396B2 (ja) 2014-09-24
DK2512453T3 (en) 2017-01-09
IL220319A0 (en) 2012-08-30
EP2512453B1 (en) 2016-11-09
HUE031228T2 (en) 2017-07-28
BR112012014935A2 (pt) 2016-03-08
WO2011073245A3 (en) 2011-08-11
US9114083B2 (en) 2015-08-25
AU2010332884A1 (en) 2012-07-05
KR20120102775A (ko) 2012-09-18
AU2010332884B2 (en) 2015-12-10
SI2512453T1 (sl) 2017-02-28
CN102791257A (zh) 2012-11-21
RU2012124834A (ru) 2014-01-27
HRP20161639T1 (hr) 2017-02-10
RS55438B1 (sr) 2017-04-28
PL2512453T3 (pl) 2017-03-31
NL1038373C2 (en) 2011-06-21
JO3762B1 (ar) 2021-01-31
US20140328934A1 (en) 2014-11-06
JP2013514312A (ja) 2013-04-25

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