BR112013031575A2 - composto peptídico ciclado de estrutura principal, composição farmacêutica, uso de composto, e, processo para a manufatura de um composto. - Google Patents

composto peptídico ciclado de estrutura principal, composição farmacêutica, uso de composto, e, processo para a manufatura de um composto.

Info

Publication number
BR112013031575A2
BR112013031575A2 BR112013031575A BR112013031575A BR112013031575A2 BR 112013031575 A2 BR112013031575 A2 BR 112013031575A2 BR 112013031575 A BR112013031575 A BR 112013031575A BR 112013031575 A BR112013031575 A BR 112013031575A BR 112013031575 A2 BR112013031575 A2 BR 112013031575A2
Authority
BR
Brazil
Prior art keywords
compound
manufacture
pharmaceutical composition
main structure
cyclic peptide
Prior art date
Application number
BR112013031575A
Other languages
English (en)
Other versions
BR112013031575B1 (pt
Inventor
Obrecht Daniel
Otto Gombert Frank
Zimmermann Johann
Original Assignee
Polyphor Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polyphor Ag filed Critical Polyphor Ag
Publication of BR112013031575A2 publication Critical patent/BR112013031575A2/pt
Publication of BR112013031575B1 publication Critical patent/BR112013031575B1/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/047Simultaneous synthesis of different peptide species; Peptide libraries
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links
BR112013031575-0A 2011-06-07 2012-06-06 Composto peptídico ciclado de estrutura principal, composição farmacêutica, uso de um composto, e, processo para a manufatura de um composto BR112013031575B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP2011059402 2011-06-07
EPPCT/EP2011/059402 2011-06-07
PCT/EP2012/060763 WO2012168336A1 (en) 2011-06-07 2012-06-06 Beta - hairpin peptidomimetics as cxc4 antagonists

Publications (2)

Publication Number Publication Date
BR112013031575A2 true BR112013031575A2 (pt) 2017-03-21
BR112013031575B1 BR112013031575B1 (pt) 2021-03-16

Family

ID=46208595

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013031575-0A BR112013031575B1 (pt) 2011-06-07 2012-06-06 Composto peptídico ciclado de estrutura principal, composição farmacêutica, uso de um composto, e, processo para a manufatura de um composto

Country Status (12)

Country Link
US (2) US9079939B2 (pt)
JP (1) JP5957521B2 (pt)
KR (1) KR102091456B1 (pt)
CN (1) CN103703018B (pt)
AU (1) AU2012266355B2 (pt)
BR (1) BR112013031575B1 (pt)
CA (1) CA2838037C (pt)
ES (1) ES2552944T3 (pt)
IL (1) IL229535B (pt)
MX (1) MX343205B (pt)
SG (1) SG195055A1 (pt)
WO (1) WO2012168336A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007079597A1 (en) 2006-01-16 2007-07-19 Polyphor Ltd. Template - fixed peptidomimetics with antimicrobial activity
DE602007008150D1 (de) 2007-02-28 2010-09-09 Polyphor Ltd Templat-fixierte peptidomimetika
US9617308B2 (en) * 2012-06-06 2017-04-11 Polyphor Ag Beta-hairpin peptidomimetics
US20240009266A1 (en) 2020-11-19 2024-01-11 Polyphor Ag Pharmaceutical combinations comprising a peptide cxcr4 inhibitor and a taxane for treating cancer
WO2022184320A2 (en) 2021-03-03 2022-09-09 Spexis Ag Medical use of cyclic peptides
WO2023285677A1 (en) 2021-07-16 2023-01-19 Spexis Ag Pharmaceutical combinations for treating cancer
WO2023285681A1 (en) 2021-07-16 2023-01-19 Spexis Ag Pharmaceutical combinations for treating cancer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995010534A1 (en) 1993-10-14 1995-04-20 Seikagaku Corporation Polypeptide and anti-hiv agent prepared therefrom
AU2003232253A1 (en) * 2003-05-02 2004-11-23 Polyphor Ag Template-fixed beta-hairpin peptidomimetics with cxcr4 antagonizing activity
DE602007008150D1 (de) * 2007-02-28 2010-09-09 Polyphor Ltd Templat-fixierte peptidomimetika
PE20090299A1 (es) * 2007-05-30 2009-03-19 Lilly Co Eli Antagonistas cxcr4 de peptido ciclicos
US8883720B2 (en) * 2008-11-26 2014-11-11 Polyphor Ag Template-fixed beta-hairpin peptidomimetics with CXCR4 antagonizing activity

Also Published As

Publication number Publication date
US20150266924A1 (en) 2015-09-24
US20140213509A1 (en) 2014-07-31
CN103703018A (zh) 2014-04-02
IL229535B (en) 2018-07-31
JP2014516999A (ja) 2014-07-17
SG195055A1 (en) 2013-12-30
WO2012168336A1 (en) 2012-12-13
US9079939B2 (en) 2015-07-14
AU2012266355B2 (en) 2016-06-09
KR102091456B1 (ko) 2020-03-23
US9556231B2 (en) 2017-01-31
MX343205B (es) 2016-10-28
BR112013031575B1 (pt) 2021-03-16
CN103703018B (zh) 2016-10-26
IL229535A0 (en) 2014-01-30
CA2838037A1 (en) 2012-12-13
AU2012266355A1 (en) 2013-12-12
ES2552944T3 (es) 2015-12-03
CA2838037C (en) 2019-09-17
MX2013014229A (es) 2014-01-23
NZ618110A (en) 2014-12-24
JP5957521B2 (ja) 2016-07-27
KR20140041689A (ko) 2014-04-04

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 06/06/2012, OBSERVADAS AS CONDICOES LEGAIS.