AR057071A1 - Producto de combinacion que comprende arilpirazoles sustituidos - Google Patents
Producto de combinacion que comprende arilpirazoles sustituidosInfo
- Publication number
- AR057071A1 AR057071A1 ARP060102546A ARP060102546A AR057071A1 AR 057071 A1 AR057071 A1 AR 057071A1 AR P060102546 A ARP060102546 A AR P060102546A AR P060102546 A ARP060102546 A AR P060102546A AR 057071 A1 AR057071 A1 AR 057071A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- alkylamino
- fluorine
- haloalkyl
- halo
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/24—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with two or more hetero atoms
- A01N43/32—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with two or more hetero atoms six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
- C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
- C07D327/06—Six-membered rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Abstract
Esta presente se refiere un un producto de combinacion que comprende una serie de 1-aril-4-ciclopropilpirazoles en los que hay al menos un fluor unido al anillo ciclopropilo, y uno o más agentes terapéuticos adicionales, particularmente agentes antiparasitarios. Reivindicacion 1: Un producto de combinacion caracterizado porque comprende un compuesto de formula (1); en la que: R1 es CF3, OCF2H, OCF3, -SCF3, -SOCF3, -SO2CF3, o SF5; R2 es H, fluor, o alquilo C1-4 opcionalmente sustituido con 1 un 5 átomos de halogeno seleccionados independientemente entre cloro y fluor; R3, R4, R5, y R6 representan independientemente H, alquilo C1-4 opcionalmente sustituido con 1 un 5 grupos halogeno seleccionados independientemente entre cloro y fluor, o un cloro o fluor; R7 es Cl o fluor; X es CR8 o N, donde R8 es Cl o fluor; y R9 es NRaRb; Ra se selecciona entre hidrogeno, alquilo C1-6, alquenilo C2-6, cicloalquilo C3-8, C(O)O-alquiloC1-6 y alcanoilo C1-6, donde cada uno de los grupos anteriores puede incluir uno o más sustituyentes opcionales cuando sea químicamente posible seleccionados independientemente entre halo, het, fenilo, hidroxi, -C(O)OH, -C(O)O-alquiloC1-6, alquilo C1-6, haloalquilo C1-6, cicloalquilo C3-8, alcoxi C1-6, haloalcoxi C1-6, amino, alquilamino C1-6 y di-alquilaminoC1-6; Rb se selecciona entre hidrogeno, alquilo C1-6, alquenilo C2-6, alcanoilo C1-6 y C(O)O-alquiloC1-6, donde cada uno de los grupos anteriores puede incluir uno o más sustituyentes opcionales cuando sea químicamente posible seleccionados independientemente entre halo, fenilo, hidroxi, -COOH, -C(O)O-alquilo C1-6, alquilo C1-6, haloalquilo C1-6, cicloalquilo C3-8, alcoxi C1-6, haloalcoxi C1-6, amino, alquilamino C1-6 y di- alquilaminoC1-6; o Ra y Rb junto con el átomo de N al que están unidos pueden formar un anillo heterocíclico de tres a siete miembros que contiene uno o más átomos N, O o S adicionales y donde dicho anillo heterocíclico puede tener uno o más sustituyentes opcionales seleccionados entre oxo, halo, het, fenilo, hidroxi, -COOH, -C(O)O-alquiloC1-6, alquilo C1-6, haloalquilo C1-6, cicloalquilo C3-6, alcoxi C1-6, haloalcoxi C1-6, amino, alquilamino C1-6 y di-alquilaminoC1-6; y het representa un grupo heterocíclico de cuatro a siete miembros, que es aromático o no aromático y que contiene uno o más heteroátomos seleccionados entre nitrogeno, oxígeno, azufre y mezclas de los mismos, y donde dicho anillo heterocíclico está opcionalmente sustituidos, donde la valencia lo permita, con uno o más sustituyentes seleccionados entre halo, ciano, nitro, alquilo C1-6, haloalquilo C1-6, alcoxi C1-6, OC(O)-alquiloC1-6, C(O)-alquiloC1-6, C(O)O-alquiloC1-6 y NRcRd, donde Rc y Rd se seleccionan independientemente entre hidrogeno, alquilo C1-6 y alquenilo C2-6, donde cada uno de los grupos anteriores puede incluir uno o más sustituyentes opcionales cuando sea químicamente posible seleccionados independientemente entre halo, fenilo, hidroxi, -COOH, C(O)O-alquiloC1-6, alquilo C1-6, haloalquilo C1-6, cicloalquilo C3-8, alcoxi C1-6, haloalcoxi C1-6, amino, alquilaminoC1-6 y di-alquilaminoC1-6; o una sal farmacéuticamente aceptable o profármaco del mismo; con la condicion de que al menos uno de R2, R3, R4, R5, o R6 sea fluor, con uno o más agentes terapéuticas distintos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11/153,103 US7514464B2 (en) | 2003-12-18 | 2005-06-15 | Substituted arylpyrazoles |
Publications (1)
Publication Number | Publication Date |
---|---|
AR057071A1 true AR057071A1 (es) | 2007-11-14 |
Family
ID=36925247
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP060102546A AR057071A1 (es) | 2005-06-15 | 2006-06-15 | Producto de combinacion que comprende arilpirazoles sustituidos |
Country Status (16)
Country | Link |
---|---|
US (4) | US7514464B2 (es) |
EP (1) | EP1901608A1 (es) |
JP (1) | JP2007008930A (es) |
KR (1) | KR20080016646A (es) |
CN (1) | CN101203134A (es) |
AR (1) | AR057071A1 (es) |
AU (1) | AU2006257645B2 (es) |
BR (1) | BRPI0613709A2 (es) |
CA (1) | CA2612286C (es) |
IL (1) | IL187556A0 (es) |
MX (1) | MX2007015115A (es) |
NO (1) | NO20076109L (es) |
RU (1) | RU2381218C2 (es) |
TW (1) | TW200716600A (es) |
WO (1) | WO2006134466A1 (es) |
ZA (1) | ZA200710133B (es) |
Families Citing this family (65)
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US7514464B2 (en) * | 2003-12-18 | 2009-04-07 | Pfizer Limited | Substituted arylpyrazoles |
DE102004053964A1 (de) * | 2004-11-09 | 2006-05-11 | Bayer Healthcare Ag | Mittel gegen Demodikose |
GB0501220D0 (en) * | 2005-01-21 | 2005-03-02 | Norbrook Lab Ltd | Anthelmintic composition |
US20080176865A1 (en) * | 2005-06-15 | 2008-07-24 | Pfizer Limited | Substituted arylpyrazoles |
US7645786B2 (en) * | 2005-06-15 | 2010-01-12 | Pfizer Inc. | Substituted arylpyrazoles |
US20080146643A1 (en) * | 2005-06-15 | 2008-06-19 | Pfizer Limited | Combination |
US20070149464A1 (en) * | 2005-06-15 | 2007-06-28 | Pfizer Inc. | Combination |
ES2338699T3 (es) * | 2005-06-15 | 2010-05-11 | Pfizer Limited | Arilpirazoles sustituidos para uso contra parasitos. |
DE102006061538A1 (de) | 2006-12-27 | 2008-07-03 | Bayer Healthcare Ag | Kombinationsprodukt zur Bekämpfung von Parasiten an Tieren |
DE102006061537A1 (de) | 2006-12-27 | 2008-07-03 | Bayer Healthcare Ag | Mittel zur Bekämpfung von Parasiten an Tieren |
CN101600687B (zh) * | 2007-02-09 | 2012-10-31 | 辉瑞股份有限公司 | 抗寄生物剂 |
KR20110098012A (ko) * | 2007-02-09 | 2011-08-31 | 화이자 리미티드 | 구충제 |
CN101873800A (zh) * | 2007-11-28 | 2010-10-27 | 日本农药株式会社 | 农业和园艺杀虫剂组合物 |
US7986196B2 (en) | 2008-07-07 | 2011-07-26 | Bae Systems Information And Electronic Systems Integration Inc. | Method and apparatus for digital synthesis of long multi-cycle microwave pulses |
GB0905365D0 (en) | 2009-03-27 | 2009-05-13 | Norbrook Lab Ltd | A topical parasiticide composition |
EP2266973A1 (de) | 2009-05-29 | 2010-12-29 | Bayer CropScience AG | Pyrazinylpyrazole |
WO2011057984A1 (de) | 2009-11-11 | 2011-05-19 | Bayer Cropscience Ag | Neue diazinyl-pyrazolylverbindungen |
CN101919856B (zh) * | 2010-05-05 | 2012-02-29 | 四川宝盛康药业有限公司 | 一种包含阿苯达唑的颗粒剂及其应用和制备方法 |
CN101919857B (zh) * | 2010-05-05 | 2012-05-30 | 四川宝盛康药业有限公司 | 一种复方阿苯达唑咀嚼片及其应用和制备方法 |
CN102453043A (zh) * | 2010-10-28 | 2012-05-16 | 桂林南药股份有限公司 | 右旋四咪唑碱的消旋方法 |
WO2012061288A1 (en) | 2010-11-03 | 2012-05-10 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
CN105360131A (zh) * | 2010-11-03 | 2016-03-02 | 陶氏益农公司 | 杀虫组合物和与其相关的方法 |
BR112013027291B1 (pt) * | 2011-04-25 | 2021-01-19 | Keki Hormusji Gharda | processo para a preparação de derivados de dicianocarboxilato |
EP2725899B1 (de) | 2011-06-30 | 2016-09-28 | Hansen-AB GmbH | Mittel zur bekämpfung von parasiten an tieren |
CA2852688C (en) | 2011-10-26 | 2021-06-29 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
JO3626B1 (ar) | 2012-02-23 | 2020-08-27 | Merial Inc | تركيبات موضعية تحتوي على فيبرونيل و بيرميثرين و طرق استخدامها |
BR112014026746A2 (pt) | 2012-04-27 | 2017-06-27 | Dow Agrosciences Llc | composições pesticidas e processos relacionados com as mesmas |
US9282739B2 (en) | 2012-04-27 | 2016-03-15 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
US9708288B2 (en) | 2012-04-27 | 2017-07-18 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
MX363173B (es) * | 2012-12-12 | 2019-03-12 | Zoetis Services Llc | Composiciones inyectables de fenilpirazol. |
BR102013021210B1 (pt) | 2013-01-25 | 2015-12-01 | Fundação Universidade Fed De São Carlos | processo de obtenção de nanopartículas biopoliméricas contendo óleo e extratos de azadirachta indica a. juss (neem), nanopartículas biopoliméricas e micropartículas em pó |
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2005
- 2005-06-15 US US11/153,103 patent/US7514464B2/en not_active Expired - Fee Related
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2006
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- 2006-06-06 US US11/917,389 patent/US7902232B2/en not_active Expired - Fee Related
- 2006-06-06 KR KR1020077029362A patent/KR20080016646A/ko not_active Application Discontinuation
- 2006-06-06 BR BRPI0613709-1A patent/BRPI0613709A2/pt not_active IP Right Cessation
- 2006-06-06 RU RU2007146113/04A patent/RU2381218C2/ru not_active IP Right Cessation
- 2006-06-06 AU AU2006257645A patent/AU2006257645B2/en not_active Ceased
- 2006-06-06 WO PCT/IB2006/001579 patent/WO2006134466A1/en active Application Filing
- 2006-06-06 EP EP06744833A patent/EP1901608A1/en not_active Withdrawn
- 2006-06-06 MX MX2007015115A patent/MX2007015115A/es active IP Right Grant
- 2006-06-14 TW TW095121209A patent/TW200716600A/zh unknown
- 2006-06-15 JP JP2006165812A patent/JP2007008930A/ja not_active Withdrawn
- 2006-06-15 AR ARP060102546A patent/AR057071A1/es unknown
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US20060014802A1 (en) | 2006-01-19 |
JP2007008930A (ja) | 2007-01-18 |
RU2381218C2 (ru) | 2010-02-10 |
CA2612286A1 (en) | 2006-12-21 |
CA2612286C (en) | 2011-04-26 |
EP1901608A1 (en) | 2008-03-26 |
TW200716600A (en) | 2007-05-01 |
ZA200710133B (en) | 2009-03-25 |
CN101203134A (zh) | 2008-06-18 |
US7902232B2 (en) | 2011-03-08 |
US7960426B2 (en) | 2011-06-14 |
US20090312371A1 (en) | 2009-12-17 |
RU2007146113A (ru) | 2009-07-20 |
AU2006257645A1 (en) | 2006-12-21 |
WO2006134466A1 (en) | 2006-12-21 |
AU2006257645B2 (en) | 2009-11-05 |
NO20076109L (no) | 2007-12-28 |
MX2007015115A (es) | 2008-04-10 |
US20110196011A1 (en) | 2011-08-11 |
KR20080016646A (ko) | 2008-02-21 |
US20090137524A1 (en) | 2009-05-28 |
IL187556A0 (en) | 2008-03-20 |
US7514464B2 (en) | 2009-04-07 |
BRPI0613709A2 (pt) | 2011-02-01 |
US8084486B2 (en) | 2011-12-27 |
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