AR055567A1 - Formas de crital de un derivado de imidazol y composicion farmaceutica - Google Patents

Formas de crital de un derivado de imidazol y composicion farmaceutica

Info

Publication number
AR055567A1
AR055567A1 ARP060100886A ARP060100886A AR055567A1 AR 055567 A1 AR055567 A1 AR 055567A1 AR P060100886 A ARP060100886 A AR P060100886A AR P060100886 A ARP060100886 A AR P060100886A AR 055567 A1 AR055567 A1 AR 055567A1
Authority
AR
Argentina
Prior art keywords
ethyl
forms
criminal
pharmaceutical
tit
Prior art date
Application number
ARP060100886A
Other languages
English (en)
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AR055567A1 publication Critical patent/AR055567A1/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Nutrition Science (AREA)
  • Pregnancy & Childbirth (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
ARP060100886A 2005-03-11 2006-03-09 Formas de crital de un derivado de imidazol y composicion farmaceutica AR055567A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US66059205P 2005-03-11 2005-03-11

Publications (1)

Publication Number Publication Date
AR055567A1 true AR055567A1 (es) 2007-08-22

Family

ID=36649530

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060100886A AR055567A1 (es) 2005-03-11 2006-03-09 Formas de crital de un derivado de imidazol y composicion farmaceutica

Country Status (21)

Country Link
US (1) US7960407B2 (enExample)
EP (1) EP1861400B1 (enExample)
JP (1) JP5069415B2 (enExample)
KR (1) KR100911073B1 (enExample)
CN (1) CN101137656B (enExample)
AR (1) AR055567A1 (enExample)
AT (1) ATE469150T1 (enExample)
AU (1) AU2006221699A1 (enExample)
BR (1) BRPI0608819B8 (enExample)
CA (1) CA2600510C (enExample)
DE (1) DE602006014516D1 (enExample)
ES (1) ES2344310T3 (enExample)
IL (1) IL185145A0 (enExample)
IN (1) IN2014DN09939A (enExample)
MX (1) MX2007011110A (enExample)
NL (1) NL300944I2 (enExample)
PL (1) PL1861400T3 (enExample)
RU (1) RU2357968C1 (enExample)
TW (1) TW200643021A (enExample)
WO (1) WO2006095268A1 (enExample)
ZA (1) ZA200707568B (enExample)

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CA2737618A1 (en) * 2008-09-25 2010-04-01 Merck Frosst Canada Ltd. Beta-carboline sulphonylurea derivatives as ep4 receptor antagonists
MX345032B (es) * 2009-04-22 2017-01-12 Raqualia Pharma Inc Antagonistas del receptor ep4 para el tratamiento de cáncer.
ES2600355T3 (es) * 2010-02-22 2017-02-08 Raqualia Pharma Inc. Uso de un antagonista del receptor EP4 en el tratamiento de dermatitis de contacto alérgica y psoriasis
RU2451680C1 (ru) 2011-02-21 2012-05-27 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном, способ его получения (варианты), фармацевтическая композиция и лекарственное средство
RU2464042C1 (ru) * 2011-03-31 2012-10-20 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО
RU2663620C2 (ru) 2013-03-19 2018-08-07 Аскат Инк. Применение рецептора антагониста ер4 для лечения хрящевой болезни
US10391086B2 (en) 2013-03-19 2019-08-27 Askat Inc. Use of EP4 receptor antagonists in the treatment of cartilage disease
US12109218B2 (en) 2014-12-09 2024-10-08 Aratana Therapeutics, Inc. Compositions of grapiprant and methods for using the same
CN107501262A (zh) * 2014-03-06 2017-12-22 阿莱塔纳治疗学股份有限公司 Grapiprant的结晶形式
TWI708606B (zh) * 2014-03-06 2020-11-01 美商雅瑞塔那醫療公司 格拉匹綸(grapiprant)組合物及其使用方法
US10342785B2 (en) 2016-11-04 2019-07-09 Askat Inc. Use of EP4 receptor antagonists for the treatment of NASH-associated liver cancer
CA3096546A1 (en) 2018-04-16 2019-10-24 Arrys Therapeutics, Inc. Ep4 inhibitors and use thereof
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