AR055567A1 - Formas de crital de un derivado de imidazol y composicion farmaceutica - Google Patents
Formas de crital de un derivado de imidazol y composicion farmaceuticaInfo
- Publication number
- AR055567A1 AR055567A1 ARP060100886A ARP060100886A AR055567A1 AR 055567 A1 AR055567 A1 AR 055567A1 AR P060100886 A ARP060100886 A AR P060100886A AR P060100886 A ARP060100886 A AR P060100886A AR 055567 A1 AR055567 A1 AR 055567A1
- Authority
- AR
- Argentina
- Prior art keywords
- ethyl
- forms
- criminal
- pharmaceutical
- tit
- Prior art date
Links
- RAXXELZNTBOGNW-UHFFFAOYSA-N 1H-imidazole Chemical class C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 title 1
- HZVLFTCYCLXTGV-UHFFFAOYSA-N 1-[2-[4-(2-ethyl-4,6-dimethylimidazo[4,5-c]pyridin-1-yl)phenyl]ethyl]-3-(4-methylphenyl)sulfonylurea Chemical compound CCC1=NC2=C(C)N=C(C)C=C2N1C(C=C1)=CC=C1CCNC(=O)NS(=O)(=O)C1=CC=C(C)C=C1 HZVLFTCYCLXTGV-UHFFFAOYSA-N 0.000 abstract 2
- 238000000634 powder X-ray diffraction Methods 0.000 abstract 2
- 230000005855 radiation Effects 0.000 abstract 2
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Virology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Molecular Biology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Gynecology & Obstetrics (AREA)
- Nutrition Science (AREA)
- Pregnancy & Childbirth (AREA)
- Obesity (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66059205P | 2005-03-11 | 2005-03-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR055567A1 true AR055567A1 (es) | 2007-08-22 |
Family
ID=36649530
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060100886A AR055567A1 (es) | 2005-03-11 | 2006-03-09 | Formas de crital de un derivado de imidazol y composicion farmaceutica |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US7960407B2 (enExample) |
| EP (1) | EP1861400B1 (enExample) |
| JP (1) | JP5069415B2 (enExample) |
| KR (1) | KR100911073B1 (enExample) |
| CN (1) | CN101137656B (enExample) |
| AR (1) | AR055567A1 (enExample) |
| AT (1) | ATE469150T1 (enExample) |
| AU (1) | AU2006221699A1 (enExample) |
| BR (1) | BRPI0608819B8 (enExample) |
| CA (1) | CA2600510C (enExample) |
| DE (1) | DE602006014516D1 (enExample) |
| ES (1) | ES2344310T3 (enExample) |
| IL (1) | IL185145A0 (enExample) |
| IN (1) | IN2014DN09939A (enExample) |
| MX (1) | MX2007011110A (enExample) |
| NL (1) | NL300944I2 (enExample) |
| PL (1) | PL1861400T3 (enExample) |
| RU (1) | RU2357968C1 (enExample) |
| TW (1) | TW200643021A (enExample) |
| WO (1) | WO2006095268A1 (enExample) |
| ZA (1) | ZA200707568B (enExample) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2737618A1 (en) * | 2008-09-25 | 2010-04-01 | Merck Frosst Canada Ltd. | Beta-carboline sulphonylurea derivatives as ep4 receptor antagonists |
| MX345032B (es) * | 2009-04-22 | 2017-01-12 | Raqualia Pharma Inc | Antagonistas del receptor ep4 para el tratamiento de cáncer. |
| ES2600355T3 (es) * | 2010-02-22 | 2017-02-08 | Raqualia Pharma Inc. | Uso de un antagonista del receptor EP4 en el tratamiento de dermatitis de contacto alérgica y psoriasis |
| RU2451680C1 (ru) | 2011-02-21 | 2012-05-27 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном, способ его получения (варианты), фармацевтическая композиция и лекарственное средство |
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| CA3107023A1 (en) * | 2018-07-11 | 2020-01-16 | Arrys Therapeutics, Inc. | Ep4 inhibitors and synthesis thereof |
| MX2021009251A (es) | 2019-01-30 | 2021-09-21 | Avista Pharma Solutions Inc | Proceso de sintesis y nuevos compuestos intermedios. |
| WO2020160075A1 (en) | 2019-01-30 | 2020-08-06 | Avista Pharma Solutions, Inc. | Chemical compounds |
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| IL110296A (en) * | 1993-07-16 | 1999-12-31 | Smithkline Beecham Corp | Imidazole compounds process for their preparation and pharmaceutical compositions containing them |
| HN2001000224A (es) | 2000-10-19 | 2002-06-13 | Pfizer | Compuestos de imidazol condensado con arilo o heteroarilo como agentes anti - inflamatorios y analgesicos. |
| IL164263A0 (en) * | 2002-04-12 | 2005-12-18 | Pfizer | Use of ep4 receptor ligands on the treatment of il-6 involved diseases |
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- 2006-03-01 CN CN2006800079642A patent/CN101137656B/zh active Active
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| RU2007133802A (ru) | 2009-03-20 |
| DE602006014516D1 (enExample) | 2010-07-08 |
| BRPI0608819A8 (pt) | 2017-10-10 |
| US20090018158A1 (en) | 2009-01-15 |
| ES2344310T3 (es) | 2010-08-24 |
| IL185145A0 (en) | 2007-12-03 |
| US7960407B2 (en) | 2011-06-14 |
| JP2006249089A (ja) | 2006-09-21 |
| AU2006221699A1 (en) | 2006-09-14 |
| IN2014DN09939A (enExample) | 2015-08-14 |
| BRPI0608819B1 (pt) | 2019-11-12 |
| CA2600510A1 (en) | 2006-09-14 |
| ZA200707568B (en) | 2009-09-30 |
| KR20070103484A (ko) | 2007-10-23 |
| EP1861400A1 (en) | 2007-12-05 |
| WO2006095268A1 (en) | 2006-09-14 |
| BRPI0608819B8 (pt) | 2021-05-25 |
| MX2007011110A (es) | 2008-02-21 |
| TW200643021A (en) | 2006-12-16 |
| ATE469150T1 (de) | 2010-06-15 |
| PL1861400T3 (pl) | 2010-09-30 |
| CA2600510C (en) | 2010-11-02 |
| CN101137656B (zh) | 2010-12-22 |
| JP5069415B2 (ja) | 2012-11-07 |
| EP1861400B1 (en) | 2010-05-26 |
| KR100911073B1 (ko) | 2009-08-06 |
| BRPI0608819A2 (pt) | 2010-01-26 |
| RU2357968C1 (ru) | 2009-06-10 |
| NL300944I2 (nl) | 2018-08-07 |
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