RU2357968C1 - Кристаллические формы производной имидазола - Google Patents
Кристаллические формы производной имидазола Download PDFInfo
- Publication number
- RU2357968C1 RU2357968C1 RU2007133802/04A RU2007133802A RU2357968C1 RU 2357968 C1 RU2357968 C1 RU 2357968C1 RU 2007133802/04 A RU2007133802/04 A RU 2007133802/04A RU 2007133802 A RU2007133802 A RU 2007133802A RU 2357968 C1 RU2357968 C1 RU 2357968C1
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- RU
- Russia
- Prior art keywords
- ethyl
- dimethyl
- phenyl
- amino
- imidazo
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Molecular Biology (AREA)
- Ophthalmology & Optometry (AREA)
- Orthopedic Medicine & Surgery (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66059205P | 2005-03-11 | 2005-03-11 | |
| US60/660,592 | 2005-03-11 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2007133802A RU2007133802A (ru) | 2009-03-20 |
| RU2357968C1 true RU2357968C1 (ru) | 2009-06-10 |
Family
ID=36649530
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2007133802/04A RU2357968C1 (ru) | 2005-03-11 | 2006-03-01 | Кристаллические формы производной имидазола |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7960407B2 (enExample) |
| EP (1) | EP1861400B1 (enExample) |
| JP (1) | JP5069415B2 (enExample) |
| KR (1) | KR100911073B1 (enExample) |
| CN (1) | CN101137656B (enExample) |
| AR (1) | AR055567A1 (enExample) |
| AT (1) | ATE469150T1 (enExample) |
| AU (1) | AU2006221699A1 (enExample) |
| BE (1) | BE2018C028I2 (enExample) |
| BR (1) | BRPI0608819B8 (enExample) |
| CA (1) | CA2600510C (enExample) |
| DE (1) | DE602006014516D1 (enExample) |
| ES (1) | ES2344310T3 (enExample) |
| FR (1) | FR18C1028I2 (enExample) |
| IL (1) | IL185145A0 (enExample) |
| IN (1) | IN2014DN09939A (enExample) |
| MX (1) | MX2007011110A (enExample) |
| NL (1) | NL300944I2 (enExample) |
| PL (1) | PL1861400T3 (enExample) |
| RU (1) | RU2357968C1 (enExample) |
| TW (1) | TW200643021A (enExample) |
| WO (1) | WO2006095268A1 (enExample) |
| ZA (1) | ZA200707568B (enExample) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012115538A1 (ru) | 2011-02-21 | 2012-08-30 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном |
| RU2464042C1 (ru) * | 2011-03-31 | 2012-10-20 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО |
| RU2663620C2 (ru) * | 2013-03-19 | 2018-08-07 | Аскат Инк. | Применение рецептора антагониста ер4 для лечения хрящевой болезни |
| RU2811411C2 (ru) * | 2014-03-06 | 2024-01-11 | Аратана Терапьютикс, Инк. | Композиции грапипранта и способы их применения |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102224154A (zh) | 2008-09-25 | 2011-10-19 | 默克弗罗斯特加拿大有限公司 | 作为EP4受体拮抗剂的β-咔啉磺酰脲衍生物 |
| ES2698508T3 (es) | 2009-04-22 | 2019-02-05 | Askat Inc | Sustancia antagonista del receptor EP4 selectivo para el tratamiento del cáncer |
| MX341482B (es) * | 2010-02-22 | 2016-08-22 | Raqualia Pharma Inc | Antagonistas del receptor ep4 y su uso en el tratamiento de enfermedades mediadas por la il-23. |
| US10391086B2 (en) | 2013-03-19 | 2019-08-27 | Askat Inc. | Use of EP4 receptor antagonists in the treatment of cartilage disease |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2012115538A1 (ru) | 2011-02-21 | 2012-08-30 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном |
| RU2464042C1 (ru) * | 2011-03-31 | 2012-10-20 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО |
| RU2663620C2 (ru) * | 2013-03-19 | 2018-08-07 | Аскат Инк. | Применение рецептора антагониста ер4 для лечения хрящевой болезни |
| RU2811411C2 (ru) * | 2014-03-06 | 2024-01-11 | Аратана Терапьютикс, Инк. | Композиции грапипранта и способы их применения |
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