AR035392A1 - Moduladores del receptor de adenosina - Google Patents

Moduladores del receptor de adenosina

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Publication number
AR035392A1
AR035392A1 ARP010100801A ARP010100801A AR035392A1 AR 035392 A1 AR035392 A1 AR 035392A1 AR P010100801 A ARP010100801 A AR P010100801A AR P010100801 A ARP010100801 A AR P010100801A AR 035392 A1 AR035392 A1 AR 035392A1
Authority
AR
Argentina
Prior art keywords
adenosine
receiver modulators
modulators
adenosine receiver
cardioprotective
Prior art date
Application number
ARP010100801A
Other languages
English (en)
Inventor
Gerda Huber-Trottmann
Gavin John Kilpatrick
Roger David Norcross
Edilio Maurizio Borroni
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR035392A1 publication Critical patent/AR035392A1/es

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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D239/42—One nitrogen atom
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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Abstract

Compuestos cíclicos heteroaromáticos, que contienen al mínimo un átomo de nitrógeno, y su uso en la elaboración de medicamentos para el tratamiento de enfermedades, relacionadas con moduladores del receptor de adenosina, tales como Alzheimer, Parkinson, neuroprotección, esquizofrenia, ansiedad, dolor insuficiencia respiratoria, depresión, asma, respuestas alérgicas, hipoxia, isquemia, epilepsia, sustancias de abuso, sedación y que puede ser relajantes musculares antipsicóticos, antiepilépticos, anticonvulsivos y agentes cardioprotectores
ARP010100801A 2000-02-25 2001-02-22 Moduladores del receptor de adenosina AR035392A1 (es)

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