MX2010009561A - Compuestos amida, composiciones y usos de los mismos. - Google Patents
Compuestos amida, composiciones y usos de los mismos.Info
- Publication number
- MX2010009561A MX2010009561A MX2010009561A MX2010009561A MX2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A
- Authority
- MX
- Mexico
- Prior art keywords
- compositions
- amide compounds
- compounds
- anxiety
- inflammation
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
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- C07C233/68—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C07C233/69—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
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Abstract
Se proveen compuestos de conformidad con la fórmula 1: (ver fórmula 1) en donde A, B, W, X', L, R1, R3, R4b, y m' son como se definió en la presente invención; se proveen compuestos y composiciones farmacéuticas de los mismos útiles para la prevención y tratamiento de una variedad de condiciones en mamíferos incluyendo humanos, incluyendo a manera de ejemplo no limitante, dolor, inflamación, trastornos cognitivos, ansiedad, depresión, y otros.
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-
2009
- 2009-02-27 MX MX2010009561A patent/MX2010009561A/es active IP Right Grant
- 2009-02-27 EP EP09716825.6A patent/EP2262766B1/en not_active Not-in-force
- 2009-02-27 WO PCT/US2009/001249 patent/WO2009110985A2/en active Application Filing
- 2009-02-27 ES ES09716825.6T patent/ES2557281T3/es active Active
- 2009-02-27 JP JP2010548731A patent/JP5539235B2/ja not_active Expired - Fee Related
- 2009-02-27 CA CA2715835A patent/CA2715835C/en not_active Expired - Fee Related
- 2009-02-27 US US12/312,749 patent/US8946439B2/en not_active Expired - Fee Related
- 2009-02-27 CN CN201410266032.6A patent/CN104058999A/zh active Pending
- 2009-02-27 CN CN200980111248.2A patent/CN101981003B/zh not_active Expired - Fee Related
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2011
- 2011-03-29 HK HK11103167.8A patent/HK1149007A1/xx not_active IP Right Cessation
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2013
- 2013-12-27 JP JP2013272289A patent/JP5916700B2/ja not_active Expired - Fee Related
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Also Published As
Publication number | Publication date |
---|---|
CN101981003B (zh) | 2014-07-02 |
JP5916700B2 (ja) | 2016-05-11 |
WO2009110985A3 (en) | 2010-02-25 |
EP2262766B1 (en) | 2015-11-11 |
US8946439B2 (en) | 2015-02-03 |
JP2014065737A (ja) | 2014-04-17 |
HK1149007A1 (en) | 2011-09-23 |
CA2715835C (en) | 2017-03-21 |
CN101981003A (zh) | 2011-02-23 |
US20110065681A1 (en) | 2011-03-17 |
WO2009110985A2 (en) | 2009-09-11 |
CN104058999A (zh) | 2014-09-24 |
EP2262766A2 (en) | 2010-12-22 |
JP2011514894A (ja) | 2011-05-12 |
JP5539235B2 (ja) | 2014-07-02 |
CA2715835A1 (en) | 2009-09-11 |
US20150266822A1 (en) | 2015-09-24 |
CN104016907A (zh) | 2014-09-03 |
ES2557281T3 (es) | 2016-01-25 |
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