AR016044A1 - Composiciones farmaceuticas que comprenden cantidades antialergenicas efectivas de descarboniletoxiloratadina - Google Patents

Composiciones farmaceuticas que comprenden cantidades antialergenicas efectivas de descarboniletoxiloratadina

Info

Publication number
AR016044A1
AR016044A1 ARP990103342A ARP990103342A AR016044A1 AR 016044 A1 AR016044 A1 AR 016044A1 AR P990103342 A ARP990103342 A AR P990103342A AR P990103342 A ARP990103342 A AR P990103342A AR 016044 A1 AR016044 A1 AR 016044A1
Authority
AR
Argentina
Prior art keywords
pharmaceutical compositions
dcl
decarbonyletoxyloratadine
antialergenic
amounts
Prior art date
Application number
ARP990103342A
Other languages
English (en)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22348307&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR016044(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of AR016044A1 publication Critical patent/AR016044A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se describen composiciones farmacéuticas que contienen 8-cloro-6,11-dihidro-11-(4-piperidiliden)-5H-benzo[5,6]-ciclohepta[1,2-b]piridina (DCL) y unacantidad protectora de DCL de una sal básica farmacéuticamente aceptable como ser fosfato dibásico decalcio y una cantidad de por lo menos un desintegrante,preferentemente dos desintegrantes como ser celulosa microcristalina y almidon suficiente para proveer una disolucion de por lo menos 80% en peso dela composicion farmacéutica en aproximadamente45 minutos y describe el uso de DCL para preparar una composicion farmacéutica para tratar reaccionesalérgicas en mamíferos como ser el hombre.
ARP990103342A 1998-07-10 1999-07-08 Composiciones farmaceuticas que comprenden cantidades antialergenicas efectivas de descarboniletoxiloratadina AR016044A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11323298A 1998-07-10 1998-07-10

Publications (1)

Publication Number Publication Date
AR016044A1 true AR016044A1 (es) 2001-06-20

Family

ID=22348307

Family Applications (4)

Application Number Title Priority Date Filing Date
ARP990103342A AR016044A1 (es) 1998-07-10 1999-07-08 Composiciones farmaceuticas que comprenden cantidades antialergenicas efectivas de descarboniletoxiloratadina
ARP000103668A AR021158A2 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]-ciclohepta[1,2-b]piridina
ARP000103667A AR021157A2 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]ciclohepta[1,2-b]piridina
ARP000103669A AR021159A1 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]-ciclohepta[1,2-b]piridina

Family Applications After (3)

Application Number Title Priority Date Filing Date
ARP000103668A AR021158A2 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]-ciclohepta[1,2-b]piridina
ARP000103667A AR021157A2 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]ciclohepta[1,2-b]piridina
ARP000103669A AR021159A1 (es) 1998-07-10 2000-07-17 Composiciones orales de 8-cloro-6,11-dihidro-11-(4-piperidilidin)-5h-benzo[5,6]-ciclohepta[1,2-b]piridina

Country Status (28)

Country Link
EP (3) EP2055303A3 (es)
JP (4) JP3224379B1 (es)
KR (1) KR100420641B1 (es)
CN (1) CN1145485C (es)
AR (4) AR016044A1 (es)
AT (2) ATE432075T1 (es)
AU (1) AU741201B2 (es)
BR (1) BR9910449A (es)
CA (2) CA2377178A1 (es)
CY (1) CY1109279T1 (es)
CZ (1) CZ300843B6 (es)
DE (2) DE69916042T2 (es)
DK (2) DK1380297T3 (es)
ES (2) ES2214871T3 (es)
HK (1) HK1030361A1 (es)
HU (1) HU228448B1 (es)
ID (1) ID28645A (es)
IL (1) IL139407A0 (es)
MY (1) MY116038A (es)
NO (1) NO331454B1 (es)
NZ (2) NZ507885A (es)
PE (1) PE20000761A1 (es)
PL (1) PL199390B1 (es)
PT (2) PT1380297E (es)
SK (1) SK288240B6 (es)
TW (1) TW575424B (es)
WO (1) WO2000002560A1 (es)
ZA (1) ZA200006224B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK287684B6 (sk) 1999-12-20 2011-06-06 Schering Corporation Pevná orálna farmaceutická dávková forma s predĺženým uvoľňovaním
AU2276801A (en) 1999-12-20 2001-07-03 Schering Corporation Extended release oral dosage composition
US7405223B2 (en) 2000-02-03 2008-07-29 Schering Corporation Treating allergic and inflammatory conditions
US7507714B2 (en) 2000-09-27 2009-03-24 Bayer Corporation Pituitary adenylate cyclase activating peptide (PACAP) receptor 3 (R3) agonists and their pharmacological methods of use
WO2006008512A2 (en) * 2004-07-16 2006-01-26 Cipla Limited Anti-histaminic composition
CA2647605A1 (en) 2006-03-31 2007-10-11 Research Foundation Itsuu Laboratory Novel compound having heterocyclic ring
JP5409382B2 (ja) 2007-11-21 2014-02-05 大日本住友製薬株式会社 口腔内崩壊錠
TR200806298A2 (tr) 2008-08-22 2010-03-22 Bi̇lgi̇ç Mahmut Farmasötik formülasyon
EP2269586B1 (en) 2009-07-01 2011-09-21 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical composition comprising desloratadine
EP2568970B1 (en) 2010-05-10 2018-12-05 Laboratorios Lesvi, S.L. Stable pharmaceutical formulations containing an antihistaminic

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985003707A1 (en) 1984-02-15 1985-08-29 Schering Corporation 8-CHLORO-6,11-DIHYDRO-11-(4-PIPERIDYLIDENE)-5H-BENZO AD5,6 BDCYCLOHEPTA AD1,2-b BDPYRIDINE AND ITS SALTS, PROCESSES FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS
US4657716A (en) 1984-03-19 1987-04-14 Lim Kunststoff Technologie Gesellschaft Method of making elastomeric shoe soles
US4990535A (en) * 1989-05-03 1991-02-05 Schering Corporation Pharmaceutical composition comprising loratadine, ibuprofen and pseudoephedrine
US5595997A (en) * 1994-12-30 1997-01-21 Sepracor Inc. Methods and compositions for treating allergic rhinitis and other disorders using descarboethoxyloratadine
PE71699A1 (es) * 1997-02-07 1999-08-03 Sepracor Inc Composicion farmaceutica de descarboetoxiloratadina sin lactosa, no higroscopica y anhidra

Also Published As

Publication number Publication date
DE69916042T2 (de) 2004-11-11
DE69940932D1 (de) 2009-07-09
CY1109279T1 (el) 2012-05-23
CN1145485C (zh) 2004-04-14
WO2000002560A1 (en) 2000-01-20
CA2377178A1 (en) 2000-01-20
EP1380297B1 (en) 2009-05-27
HK1030361A1 (en) 2001-05-04
PT1073438E (pt) 2004-07-30
TW575424B (en) 2004-02-11
JP3224379B1 (ja) 2001-10-29
HU228448B1 (en) 2013-03-28
EP1380297A1 (en) 2004-01-14
CA2325014C (en) 2002-05-28
JP4160739B2 (ja) 2008-10-08
NZ512916A (en) 2003-03-28
AR021159A1 (es) 2002-06-12
ATE432075T1 (de) 2009-06-15
NZ507885A (en) 2001-08-31
CN1303284A (zh) 2001-07-11
AU741201B2 (en) 2001-11-22
EP2055303A2 (en) 2009-05-06
KR20010043402A (ko) 2001-05-25
EP1073438A1 (en) 2001-02-07
MY116038A (en) 2003-10-31
IL139407A0 (en) 2001-11-25
PT1380297E (pt) 2009-07-06
DK1073438T3 (da) 2004-05-10
HUP0101900A2 (hu) 2001-11-28
PE20000761A1 (es) 2000-08-31
ZA200006224B (en) 2001-11-01
NO20005485D0 (no) 2000-10-31
IL139407A (en) 2001-10-31
JP2005298524A (ja) 2005-10-27
DK1380297T3 (da) 2009-08-17
BR9910449A (pt) 2001-01-02
PL199390B1 (pl) 2008-09-30
NO331454B1 (no) 2012-01-09
AU4953199A (en) 2000-02-01
ID28645A (id) 2001-06-21
CZ20004056A3 (cs) 2001-03-14
DE69916042D1 (de) 2004-05-06
JP2002068983A (ja) 2002-03-08
AR021158A2 (es) 2002-06-12
JP2010265329A (ja) 2010-11-25
ATE262904T1 (de) 2004-04-15
JP4621082B2 (ja) 2011-01-26
EP1073438B1 (en) 2004-03-31
JP2002520285A (ja) 2002-07-09
CZ300843B6 (cs) 2009-08-26
KR100420641B1 (ko) 2004-03-02
EP2055303A3 (en) 2009-12-16
NO20005485L (no) 2001-03-09
HUP0101900A3 (en) 2003-01-28
ES2214871T3 (es) 2004-09-16
CA2325014A1 (en) 2000-01-20
SK17112000A3 (sk) 2001-12-03
PL344045A1 (en) 2001-09-24
AR021157A2 (es) 2002-06-12
ES2326214T3 (es) 2009-10-05
SK288240B6 (sk) 2015-02-03

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