ZA961947B - 6-substituted pyrazolo(3,4-d)pyrimidin-4-ones and compositions and methods of use thereof - Google Patents

6-substituted pyrazolo(3,4-d)pyrimidin-4-ones and compositions and methods of use thereof

Info

Publication number
ZA961947B
ZA961947B ZA961947A ZA961947A ZA961947B ZA 961947 B ZA961947 B ZA 961947B ZA 961947 A ZA961947 A ZA 961947A ZA 961947 A ZA961947 A ZA 961947A ZA 961947 B ZA961947 B ZA 961947B
Authority
ZA
South Africa
Prior art keywords
pyrimidin
ones
compositions
methods
substituted pyrazolo
Prior art date
Application number
ZA961947A
Other languages
English (en)
Inventor
Edward R Bacon
Sol J Daum
Baldev Singh
Original Assignee
Sanofi Winthrop Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Winthrop Inc filed Critical Sanofi Winthrop Inc
Publication of ZA961947B publication Critical patent/ZA961947B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA961947A 1995-03-10 1996-03-11 6-substituted pyrazolo(3,4-d)pyrimidin-4-ones and compositions and methods of use thereof ZA961947B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/402,268 US5656629A (en) 1995-03-10 1995-03-10 6-substituted pyrazolo (3,4-d)pyrimidin-4-ones and compositions and methods of use thereof

Publications (1)

Publication Number Publication Date
ZA961947B true ZA961947B (en) 1996-10-07

Family

ID=23591222

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA961947A ZA961947B (en) 1995-03-10 1996-03-11 6-substituted pyrazolo(3,4-d)pyrimidin-4-ones and compositions and methods of use thereof

Country Status (13)

Country Link
US (2) US5656629A (cs)
EP (1) EP0813527A4 (cs)
JP (1) JPH11501923A (cs)
KR (1) KR19980702891A (cs)
AU (1) AU708750B2 (cs)
CA (1) CA2211669A1 (cs)
CZ (1) CZ280597A3 (cs)
HU (1) HUP9801336A3 (cs)
NO (1) NO974151L (cs)
NZ (1) NZ306035A (cs)
PL (1) PL322380A1 (cs)
WO (1) WO1996028429A1 (cs)
ZA (1) ZA961947B (cs)

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DE10328479A1 (de) * 2003-06-25 2005-01-13 Bayer Ag 6-Arylamino-5-cyano-4-pyrimidinone
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US7572799B2 (en) 2003-11-24 2009-08-11 Pfizer Inc Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors
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Also Published As

Publication number Publication date
NO974151D0 (no) 1997-09-09
NZ306035A (en) 1999-07-29
US5656629A (en) 1997-08-12
KR19980702891A (ko) 1998-08-05
AU5418896A (en) 1996-10-02
HUP9801336A2 (hu) 1998-10-28
EP0813527A1 (en) 1997-12-29
WO1996028429A1 (en) 1996-09-19
CZ280597A3 (cs) 1998-04-15
US5977118A (en) 1999-11-02
PL322380A1 (en) 1998-01-19
CA2211669A1 (en) 1996-09-19
MX9706876A (es) 1998-06-28
HUP9801336A3 (en) 2000-07-28
NO974151L (no) 1997-11-04
EP0813527A4 (en) 1998-09-09
JPH11501923A (ja) 1999-02-16
AU708750B2 (en) 1999-08-12

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