ZA834189B - Dynorphin amide analogs - Google Patents

Dynorphin amide analogs

Info

Publication number
ZA834189B
ZA834189B ZA834189A ZA834189A ZA834189B ZA 834189 B ZA834189 B ZA 834189B ZA 834189 A ZA834189 A ZA 834189A ZA 834189 A ZA834189 A ZA 834189A ZA 834189 B ZA834189 B ZA 834189B
Authority
ZA
South Africa
Prior art keywords
dynorphin
amino acids
compounds
amide analogs
new compounds
Prior art date
Application number
ZA834189A
Other languages
English (en)
Inventor
Nancy M Lee
Horace H Loh
Kang Chang Jaw
Original Assignee
Univ California
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ California filed Critical Univ California
Publication of ZA834189B publication Critical patent/ZA834189B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Polyamides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
ZA834189A 1982-06-10 1983-06-08 Dynorphin amide analogs ZA834189B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/387,005 US4462941A (en) 1982-06-10 1982-06-10 Dynorphin amide analogs

Publications (1)

Publication Number Publication Date
ZA834189B true ZA834189B (en) 1984-02-29

Family

ID=23528034

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA834189A ZA834189B (en) 1982-06-10 1983-06-08 Dynorphin amide analogs

Country Status (15)

Country Link
US (1) US4462941A (de)
EP (1) EP0096592B1 (de)
JP (1) JPS5925365A (de)
KR (1) KR840005080A (de)
AT (1) ATE22449T1 (de)
AU (1) AU1448983A (de)
CA (1) CA1241645A (de)
DE (1) DE3366428D1 (de)
DK (1) DK262683A (de)
FI (1) FI832095L (de)
IL (1) IL68825A0 (de)
IS (1) IS2812A7 (de)
NO (1) NO832107L (de)
PT (1) PT76860B (de)
ZA (1) ZA834189B (de)

Families Citing this family (84)

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US4481191A (en) * 1983-03-30 1984-11-06 The Regents Of The University Of California Method for controlling blood pressure
US4900811A (en) * 1983-07-21 1990-02-13 Scripps Clinic And Research Foundation Synthetic polypeptides corresponding to portions of proteinoids translated from brain-specific mRNAs, receptors, methods and diagnostics using the same
US5242798A (en) * 1983-07-21 1993-09-07 Scripps Clinic And Research Foundation Synthetic polypeptides corresponding to portions of proteinoids translated from brain-specific mRNAs, receptors, methods and diagnostics using the same
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US5482930A (en) * 1993-06-09 1996-01-09 The Regents Of The University Of California Anti-inflammatory composition and method with des-Tyr dynorphin and analogues
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AU7637394A (en) * 1994-08-26 1996-03-22 Avram Goldstein Analgesic method with dynorphin analogues truncated at the n-terminus
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EP1976876A4 (de) * 2005-12-22 2010-01-13 Conjuchem Biotechnologies Inc Verfahren zur herstellung von vorgebildeten konjugaten von albumin und einem therapeutischen mittel
WO2008077194A1 (en) * 2006-12-22 2008-07-03 Xenome Ltd Receptor agonists
US20090099074A1 (en) * 2007-01-10 2009-04-16 Conjuchem Biotechnologies Inc. Modulating food intake
DE102007011485A1 (de) 2007-03-07 2008-09-11 Grünenthal GmbH Darreichungsform mit erschwertem Missbrauch
CA2708762A1 (en) * 2007-12-11 2009-06-18 Conjuchem Biotechnologies Inc. Formulation of insulinotropic peptide conjugates
TWI454288B (zh) 2008-01-25 2014-10-01 Gruenenthal Chemie 藥物劑型
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CN102573805A (zh) 2009-07-22 2012-07-11 格吕伦塔尔有限公司 热熔挤出的控制释放剂型
ES2560210T3 (es) 2009-07-22 2016-02-17 Grünenthal GmbH Forma de dosificación resistente a la manipulación para opiádes sensibles a la oxidación
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TWI516286B (zh) 2010-09-02 2016-01-11 歌林達股份有限公司 含陰離子聚合物之抗破碎劑型
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Family Cites Families (4)

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Publication number Priority date Publication date Assignee Title
JPS5572153A (en) * 1978-11-26 1980-05-30 Shionogi & Co Ltd Undecapeptide
US4396606A (en) * 1979-11-05 1983-08-02 Addiction Research Foundation Novel polypeptide analgesics
US4361553A (en) * 1981-05-18 1982-11-30 Regents Of The University Of California Therapeutic uses of dynorphin
JPS5815946A (ja) 1981-07-21 1983-01-29 Eisai Co Ltd 新規ヘプタデカペプタイド

Also Published As

Publication number Publication date
EP0096592A1 (de) 1983-12-21
DK262683D0 (da) 1983-06-09
JPS5925365A (ja) 1984-02-09
IL68825A0 (en) 1983-09-30
US4462941A (en) 1984-07-31
JPH0427995B2 (de) 1992-05-13
CA1241645A (en) 1988-09-06
KR840005080A (ko) 1984-11-03
ATE22449T1 (de) 1986-10-15
AU1448983A (en) 1983-12-15
PT76860A (en) 1983-07-01
NO832107L (no) 1983-12-12
IS2812A7 (is) 1983-10-07
EP0096592B1 (de) 1986-09-24
DE3366428D1 (en) 1986-10-30
DK262683A (da) 1983-12-11
FI832095A0 (fi) 1983-06-10
PT76860B (en) 1986-01-27
FI832095L (fi) 1983-12-11

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