ZA200804498B - N4-phenyl-quinazoline-4 -amine derivatives and related compounds as ERBB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases - Google Patents

N4-phenyl-quinazoline-4 -amine derivatives and related compounds as ERBB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

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Publication number
ZA200804498B
ZA200804498B ZA200804498A ZA200804498A ZA200804498B ZA 200804498 B ZA200804498 B ZA 200804498B ZA 200804498 A ZA200804498 A ZA 200804498A ZA 200804498 A ZA200804498 A ZA 200804498A ZA 200804498 B ZA200804498 B ZA 200804498B
Authority
ZA
South Africa
Prior art keywords
treatment
tyrosine kinase
kinase inhibitors
quinazoline
receptor tyrosine
Prior art date
Application number
ZA200804498A
Other languages
English (en)
Inventor
Joseph P Lyssikatos
Fredrik P Marmsater
Zhao Qian
Greschuk Julie Marie
Liu Weidong
Hennings D David
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of ZA200804498B publication Critical patent/ZA200804498B/xx

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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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ZA200804498A 2005-11-15 2006-11-15 N4-phenyl-quinazoline-4 -amine derivatives and related compounds as ERBB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases ZA200804498B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73628905P 2005-11-15 2005-11-15
US81701906P 2006-06-28 2006-06-28

Publications (1)

Publication Number Publication Date
ZA200804498B true ZA200804498B (en) 2009-07-29

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ZA200804498A ZA200804498B (en) 2005-11-15 2006-11-15 N4-phenyl-quinazoline-4 -amine derivatives and related compounds as ERBB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

Country Status (29)

Country Link
US (6) US8648087B2 (no)
EP (2) EP2090575B1 (no)
JP (2) JP5134548B2 (no)
KR (1) KR101086967B1 (no)
CN (2) CN102887891B (no)
AT (2) ATE507224T1 (no)
AU (2) AU2006315383B2 (no)
BR (2) BR122018075851B1 (no)
CA (2) CA2632194C (no)
CY (2) CY1110583T1 (no)
DE (2) DE602006009968D1 (no)
DK (2) DK2090575T3 (no)
ES (2) ES2335535T3 (no)
FI (1) FIC20210022I1 (no)
FR (1) FR21C1031I2 (no)
HK (2) HK1129678A1 (no)
HU (1) HUS2100028I1 (no)
IL (2) IL239149A (no)
LT (1) LTC1971601I2 (no)
LU (1) LUC00217I2 (no)
NL (1) NL301113I2 (no)
NO (1) NO342413B1 (no)
PL (2) PL1971601T3 (no)
PT (2) PT1971601E (no)
RU (2) RU2592703C9 (no)
SG (1) SG152230A1 (no)
SI (2) SI2090575T1 (no)
WO (1) WO2007059257A2 (no)
ZA (1) ZA200804498B (no)

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