ZA200609401B - Sustained release formulations - Google Patents
Sustained release formulations Download PDFInfo
- Publication number
- ZA200609401B ZA200609401B ZA200609401A ZA200609401A ZA200609401B ZA 200609401 B ZA200609401 B ZA 200609401B ZA 200609401 A ZA200609401 A ZA 200609401A ZA 200609401 A ZA200609401 A ZA 200609401A ZA 200609401 B ZA200609401 B ZA 200609401B
- Authority
- ZA
- South Africa
- Prior art keywords
- peptide
- acid ester
- gallic acid
- complex
- salt
- Prior art date
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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US20050271726A1 (en) * | 2004-06-02 | 2005-12-08 | Albert Crum | Immune enhancing compositions and methods of use thereof |
EP1841455A1 (en) | 2005-01-24 | 2007-10-10 | Amgen Inc. | Humanized anti-amyloid antibody |
US7252834B2 (en) | 2005-04-25 | 2007-08-07 | Clemson University Research Foundation (Curf) | Elastin stabilization of connective tissue |
US8236759B2 (en) * | 2005-06-30 | 2012-08-07 | Ipsen Pharma Sas | GLP-1 pharmaceutical compositions |
WO2007117356A2 (en) * | 2006-02-15 | 2007-10-18 | Gammacan Ltd. | Immunoglobulins from vitiligo plasma for melanoma therapy |
EP2498096A1 (en) * | 2006-07-21 | 2012-09-12 | Amgen Inc. | Method of detecting and/or measuring hepcidin in a sample |
TWI454479B (zh) | 2007-03-06 | 2014-10-01 | Amgen Inc | 變異之活動素受體多肽及其用途 |
WO2013106175A1 (en) | 2011-12-19 | 2013-07-18 | Amgen Inc. | Variant activin receptor polypeptides, alone or in combination with chemotherapy, and uses thereof |
MX2009012609A (es) | 2007-05-22 | 2009-12-07 | Amgen Inc | Composiciones y metodos para producir proteinas de fusion bioactivas. |
EP2235058A2 (en) | 2007-12-21 | 2010-10-06 | Amgen, Inc | Anti-amyloid antibodies and uses thereof |
JP2011513220A (ja) * | 2008-02-21 | 2011-04-28 | ヴァトリックス・メディカル・インコーポレーテッド | デリバリービヒクルと組み合わせた結合組織安定剤の適用による動脈瘤の処置 |
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US20100119605A1 (en) * | 2008-11-12 | 2010-05-13 | Isenburg Jason C | Compositions for tissue stabilization |
US8444624B2 (en) * | 2009-10-19 | 2013-05-21 | Vatrix Medical, Inc. | Vascular medical devices with sealing elements and procedures for the treatment of isolated vessel sections |
US8911468B2 (en) | 2011-01-31 | 2014-12-16 | Vatrix Medical, Inc. | Devices, therapeutic compositions and corresponding percutaneous treatment methods for aortic dissection |
PE20140593A1 (es) | 2011-03-16 | 2014-05-10 | Amgen Inc | Inhibidores potentes y selectivos de nav1.3 y nav1.7 |
JP2014516695A (ja) | 2011-05-18 | 2014-07-17 | バトリックス・メディカル・インコーポレイテッド | 血管安定化用被覆バルーン |
JP6426107B2 (ja) | 2012-12-20 | 2018-11-21 | アムジエン・インコーポレーテツド | Apj受容体アゴニストおよびその使用 |
SG11201505960VA (en) | 2013-02-01 | 2015-08-28 | Santa Maria Biotherapeutics Inc | Administration of an anti-activin-a compound to a subject |
WO2014165277A2 (en) | 2013-03-12 | 2014-10-09 | Amgen Inc. | POTENT AND SELECTIVE INHIBITORS OF Nav1.7 |
ES2950789T3 (es) | 2014-06-10 | 2023-10-13 | Amgen Inc | Polipéptidos de apelina |
TW201618783A (zh) | 2014-08-07 | 2016-06-01 | 艾森塔製藥公司 | 以布魯頓(Bruton)氏酪胺酸激酶(BTK)佔據和BTK再合成速率為基礎之治療癌症、免疫和自體免疫疾病及發炎性疾病之方法 |
US11318190B2 (en) | 2017-05-05 | 2022-05-03 | United States Government As Represented By The Department Of Veterans Affairs | Methods and compositions for treating liver disease |
US11654114B2 (en) * | 2017-06-07 | 2023-05-23 | Egy-Nano Pharma, Lp | Oral prolonged drug delivery platforms |
JP7111897B2 (ja) | 2018-08-03 | 2022-08-02 | ネクテロ・メディカル・インコーポレイテッド | 精製ペンタガロイルグルコース及び送達用デバイス |
WO2020227437A1 (en) | 2019-05-06 | 2020-11-12 | Axial Biotherapeutics, Inc. | Sustained release solid dosage forms for modulating the colonic microbiome |
Family Cites Families (30)
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JP2000080027A (ja) * | 1998-09-02 | 2000-03-21 | Taiyo Kagaku Co Ltd | 徐放性製剤 |
US6428818B1 (en) | 1999-03-30 | 2002-08-06 | Purdue Research Foundation | Tea catechin formulations and processes for making same |
EP1225916A1 (en) | 1999-11-01 | 2002-07-31 | University Technology Corporation | Compositions and methods for controlled-release delivery and increased potency of pharmaceuticals via hydrophobic ion-pairing |
US6713506B2 (en) * | 2000-10-11 | 2004-03-30 | University Of South Florida | Tea polyphenol esters and analogs thereof for cancer prevention and treatment |
US6759064B2 (en) | 2001-02-22 | 2004-07-06 | Purdue Research Foundation | Compositions based on vanilloid-catechin synergies for prevention and treatment of cancer |
JP5013152B2 (ja) * | 2001-02-28 | 2012-08-29 | 株式会社ビーエムジー | 蛋白質複合体形成剤 |
US20040142048A1 (en) | 2002-02-22 | 2004-07-22 | Morre Dorothy M. | Compositions based on proanthocyanadin-catechin synergies for prevention and treatment of cancer |
WO2004012522A1 (en) | 2002-07-26 | 2004-02-12 | Dsm Ip Assets B.V. | Compositions comprising lactoferrin |
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2005
- 2005-04-25 DK DK05742315.4T patent/DK1750683T3/da active
- 2005-04-25 CN CN201410023256.4A patent/CN103920162B/zh not_active Expired - Fee Related
- 2005-04-25 EP EP05742315A patent/EP1750683B1/en active Active
- 2005-04-25 AU AU2005237542A patent/AU2005237542B2/en not_active Ceased
- 2005-04-25 US US11/114,473 patent/US7323169B2/en not_active Expired - Fee Related
- 2005-04-25 PT PT57423154T patent/PT1750683E/pt unknown
- 2005-04-25 CN CNA2005800124592A patent/CN1997356A/zh active Pending
- 2005-04-25 ES ES05742315T patent/ES2400687T3/es active Active
- 2005-04-25 PL PL05742315T patent/PL1750683T3/pl unknown
- 2005-04-25 KR KR1020067021346A patent/KR101201638B1/ko not_active IP Right Cessation
- 2005-04-25 CA CA2563185A patent/CA2563185C/en not_active Expired - Fee Related
- 2005-04-25 JP JP2007509735A patent/JP5036533B2/ja not_active Expired - Fee Related
- 2005-04-25 WO PCT/US2005/014254 patent/WO2005105057A1/en active Application Filing
- 2005-04-25 SI SI200531678T patent/SI1750683T1/sl unknown
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- 2006-10-15 IL IL178596A patent/IL178596A/en not_active IP Right Cessation
- 2006-11-13 ZA ZA200609401A patent/ZA200609401B/en unknown
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2007
- 2007-08-13 HK HK07108780.0A patent/HK1103023A1/xx not_active IP Right Cessation
- 2007-08-30 US US11/847,984 patent/US7732399B2/en not_active Expired - Fee Related
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2011
- 2011-09-09 JP JP2011196883A patent/JP5829870B2/ja not_active Expired - Fee Related
- 2011-09-09 JP JP2011196884A patent/JP2012036194A/ja active Pending
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Also Published As
Publication number | Publication date |
---|---|
JP5829870B2 (ja) | 2015-12-09 |
US7323169B2 (en) | 2008-01-29 |
EP1750683A1 (en) | 2007-02-14 |
CN1997356A (zh) | 2007-07-11 |
PL1750683T3 (pl) | 2013-05-31 |
US20050271722A1 (en) | 2005-12-08 |
IL178596A (en) | 2012-06-28 |
IL178596A0 (en) | 2007-02-11 |
US7732399B2 (en) | 2010-06-08 |
WO2005105057A1 (en) | 2005-11-10 |
KR20070026457A (ko) | 2007-03-08 |
SI1750683T1 (sl) | 2013-04-30 |
JP5036533B2 (ja) | 2012-09-26 |
DK1750683T3 (da) | 2013-04-15 |
US20070292506A1 (en) | 2007-12-20 |
JP2012046520A (ja) | 2012-03-08 |
CN103920162B (zh) | 2017-07-11 |
ES2400687T3 (es) | 2013-04-11 |
PT1750683E (pt) | 2013-01-25 |
EP1750683B1 (en) | 2013-01-09 |
CA2563185C (en) | 2010-04-20 |
JP2007534698A (ja) | 2007-11-29 |
HK1103023A1 (en) | 2007-12-14 |
CA2563185A1 (en) | 2005-11-10 |
JP2012036194A (ja) | 2012-02-23 |
AU2005237542A1 (en) | 2005-11-10 |
CN103920162A (zh) | 2014-07-16 |
KR101201638B1 (ko) | 2012-11-15 |
HK1200092A1 (en) | 2015-07-31 |
AU2005237542B2 (en) | 2009-12-17 |
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