ZA200604788B - Benzylether amine compounds usefl as CCR-5 antagonists - Google Patents
Benzylether amine compounds usefl as CCR-5 antagonistsInfo
- Publication number
- ZA200604788B ZA200604788B ZA200604788A ZA200604788A ZA200604788B ZA 200604788 B ZA200604788 B ZA 200604788B ZA 200604788 A ZA200604788 A ZA 200604788A ZA 200604788 A ZA200604788 A ZA 200604788A ZA 200604788 B ZA200604788 B ZA 200604788B
- Authority
- ZA
- South Africa
- Prior art keywords
- usefl
- benzylether
- ccr
- antagonists
- amine compounds
- Prior art date
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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- C07D211/38—Halogen atoms or nitro radicals
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
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US7754725B2 (en) | 2006-03-01 | 2010-07-13 | Astex Therapeutics Ltd. | Dihydroxyphenyl isoindolymethanones |
WO2008044041A1 (en) | 2006-10-12 | 2008-04-17 | Astex Therapeutics Limited | Pharmaceutical combinations |
JP5721949B2 (ja) | 2006-10-12 | 2015-05-20 | アステックス、セラピューティックス、リミテッドAstex Therapeutics Limited | 複合薬剤 |
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JP5518478B2 (ja) | 2006-10-12 | 2014-06-11 | アステックス、セラピューティックス、リミテッド | 医薬化合物 |
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US8026365B2 (en) | 2007-05-25 | 2011-09-27 | Hoffman-La Roche Inc. | 4,4-disubstituted piperidine derivatives |
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EP2513115B1 (en) | 2009-12-18 | 2013-10-09 | Basilea Pharmaceutica AG | Tricyclic antibiotics |
US8791100B2 (en) * | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
CN103635474B (zh) | 2011-06-17 | 2016-04-27 | 巴斯利尔药物股份公司 | 三环抗生素 |
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-
2004
- 2004-11-08 EP EP04810567A patent/EP1687268A1/en not_active Withdrawn
- 2004-11-08 RU RU2006120084/04A patent/RU2006120084A/ru not_active Application Discontinuation
- 2004-11-08 US US10/984,430 patent/US20050101644A1/en not_active Abandoned
- 2004-11-08 AU AU2004289690A patent/AU2004289690A1/en not_active Abandoned
- 2004-11-08 WO PCT/US2004/037258 patent/WO2005047249A1/en active Application Filing
- 2004-11-08 KR KR1020067011398A patent/KR20060123292A/ko not_active Application Discontinuation
- 2004-11-08 CN CNA2004800402095A patent/CN1902171A/zh active Pending
- 2004-11-08 BR BRPI0415874-1A patent/BRPI0415874A/pt not_active Application Discontinuation
- 2004-11-08 CA CA002543913A patent/CA2543913A1/en not_active Abandoned
- 2004-11-08 JP JP2006539723A patent/JP2007513082A/ja active Pending
-
2006
- 2006-04-26 IL IL175227A patent/IL175227A0/en unknown
- 2006-06-09 ZA ZA200604788A patent/ZA200604788B/xx unknown
- 2006-06-09 NO NO20062677A patent/NO20062677L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
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CN1902171A (zh) | 2007-01-24 |
WO2005047249A1 (en) | 2005-05-26 |
RU2006120084A (ru) | 2008-01-10 |
NO20062677L (no) | 2006-08-09 |
EP1687268A1 (en) | 2006-08-09 |
US20050101644A1 (en) | 2005-05-12 |
AU2004289690A1 (en) | 2005-05-26 |
CA2543913A1 (en) | 2005-05-26 |
KR20060123292A (ko) | 2006-12-01 |
JP2007513082A (ja) | 2007-05-24 |
BRPI0415874A (pt) | 2007-01-09 |
IL175227A0 (en) | 2006-09-05 |
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