ZA200603355B - Use of cyclic anabaenopeptin-type peptides for the treatment of a condition wherein inhibition of carboxypeptidase U is beneficial, novel anabaenopeptin derivatives and intermediates thereof - Google Patents
Use of cyclic anabaenopeptin-type peptides for the treatment of a condition wherein inhibition of carboxypeptidase U is beneficial, novel anabaenopeptin derivatives and intermediates thereof Download PDFInfo
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- ZA200603355B ZA200603355B ZA200603355A ZA200603355A ZA200603355B ZA 200603355 B ZA200603355 B ZA 200603355B ZA 200603355 A ZA200603355 A ZA 200603355A ZA 200603355 A ZA200603355 A ZA 200603355A ZA 200603355 B ZA200603355 B ZA 200603355B
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P41/00—Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Diabetes (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Physical Education & Sports Medicine (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Toxicology (AREA)
- Psychology (AREA)
- Vascular Medicine (AREA)
- Surgery (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0302853A SE0302853D0 (sv) | 2003-10-29 | 2003-10-29 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200603355B true ZA200603355B (en) | 2007-07-25 |
Family
ID=29580155
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200603355A ZA200603355B (en) | 2003-10-29 | 2006-04-26 | Use of cyclic anabaenopeptin-type peptides for the treatment of a condition wherein inhibition of carboxypeptidase U is beneficial, novel anabaenopeptin derivatives and intermediates thereof |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US20080039376A1 (fr) |
| EP (1) | EP1689424A1 (fr) |
| JP (1) | JP2008501622A (fr) |
| KR (1) | KR20060132596A (fr) |
| CN (1) | CN1897963A (fr) |
| AR (1) | AR046612A1 (fr) |
| AU (1) | AU2004283643B2 (fr) |
| BR (1) | BRPI0415964A (fr) |
| CA (1) | CA2543630A1 (fr) |
| CO (1) | CO5690614A2 (fr) |
| IL (1) | IL175198A0 (fr) |
| IS (1) | IS8471A (fr) |
| MY (1) | MY143363A (fr) |
| NO (1) | NO20061999L (fr) |
| RU (1) | RU2365594C2 (fr) |
| SA (1) | SA05250463B1 (fr) |
| SE (1) | SE0302853D0 (fr) |
| TW (1) | TW200524576A (fr) |
| UA (1) | UA85199C2 (fr) |
| UY (1) | UY28585A1 (fr) |
| WO (1) | WO2005039617A1 (fr) |
| ZA (1) | ZA200603355B (fr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016053901A1 (fr) | 2014-09-30 | 2016-04-07 | Apple Inc | Structures d'entrée sensibles à la force configurables pour dispositifs électroniques |
| TWI628569B (zh) | 2015-09-30 | 2018-07-01 | 蘋果公司 | 具有適應性輸入列之鍵盤 |
| RS63143B1 (sr) | 2016-06-01 | 2022-05-31 | Athira Pharma Inc | Jedinjenja |
| US10732743B2 (en) | 2017-07-18 | 2020-08-04 | Apple Inc. | Concealable input region for an electronic device having microperforations |
| US20210130409A1 (en) * | 2017-09-01 | 2021-05-06 | Alsonex Pty Ltd | Method for the Solid-Phase Synthesis of Cyclic Pentapeptides |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9524630D0 (en) * | 1994-12-24 | 1996-01-31 | Zeneca Ltd | Chemical compounds |
| BR0113289A (pt) * | 2000-08-17 | 2003-06-17 | Pfizer | Imidazóis substituìdos como inibidores de tafia |
-
2003
- 2003-10-29 SE SE0302853A patent/SE0302853D0/xx unknown
-
2004
- 2004-10-27 MY MYPI20044426A patent/MY143363A/en unknown
- 2004-10-28 RU RU2006117821/04A patent/RU2365594C2/ru not_active IP Right Cessation
- 2004-10-28 KR KR1020067010392A patent/KR20060132596A/ko not_active Application Discontinuation
- 2004-10-28 AU AU2004283643A patent/AU2004283643B2/en not_active Ceased
- 2004-10-28 UY UY28585A patent/UY28585A1/es not_active Application Discontinuation
- 2004-10-28 UA UAA200604776A patent/UA85199C2/ru unknown
- 2004-10-28 CN CNA2004800390596A patent/CN1897963A/zh active Pending
- 2004-10-28 WO PCT/SE2004/001568 patent/WO2005039617A1/fr active Application Filing
- 2004-10-28 US US10/578,022 patent/US20080039376A1/en not_active Abandoned
- 2004-10-28 BR BRPI0415964-0A patent/BRPI0415964A/pt not_active IP Right Cessation
- 2004-10-28 CA CA002543630A patent/CA2543630A1/fr not_active Abandoned
- 2004-10-28 EP EP04793868A patent/EP1689424A1/fr not_active Withdrawn
- 2004-10-28 JP JP2006537936A patent/JP2008501622A/ja not_active Withdrawn
- 2004-10-29 TW TW093132865A patent/TW200524576A/zh unknown
- 2004-11-01 AR ARP040104004A patent/AR046612A1/es unknown
-
2005
- 2005-01-29 SA SA05250463A patent/SA05250463B1/ar unknown
-
2006
- 2006-04-25 IL IL175198A patent/IL175198A0/en unknown
- 2006-04-26 ZA ZA200603355A patent/ZA200603355B/en unknown
- 2006-05-04 NO NO20061999A patent/NO20061999L/no not_active Application Discontinuation
- 2006-05-16 IS IS8471A patent/IS8471A/is unknown
- 2006-05-23 CO CO06049388A patent/CO5690614A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IS8471A (is) | 2006-05-16 |
| IL175198A0 (en) | 2006-09-05 |
| RU2006117821A (ru) | 2007-12-10 |
| SA05250463B1 (ar) | 2009-02-07 |
| CO5690614A2 (es) | 2006-10-31 |
| CN1897963A (zh) | 2007-01-17 |
| KR20060132596A (ko) | 2006-12-21 |
| NO20061999L (no) | 2006-07-27 |
| CA2543630A1 (fr) | 2005-05-06 |
| JP2008501622A (ja) | 2008-01-24 |
| US20080039376A1 (en) | 2008-02-14 |
| WO2005039617A1 (fr) | 2005-05-06 |
| AU2004283643B2 (en) | 2008-07-10 |
| EP1689424A1 (fr) | 2006-08-16 |
| SE0302853D0 (sv) | 2003-10-29 |
| AR046612A1 (es) | 2005-12-14 |
| MY143363A (en) | 2011-04-29 |
| BRPI0415964A (pt) | 2007-01-23 |
| UA85199C2 (ru) | 2009-01-12 |
| RU2365594C2 (ru) | 2009-08-27 |
| SA05250463A (ar) | 2005-12-03 |
| AU2004283643A1 (en) | 2005-05-06 |
| TW200524576A (en) | 2005-08-01 |
| UY28585A1 (es) | 2005-05-31 |
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