ZA200508948B - Substituted pyrazoles - Google Patents

Substituted pyrazoles Download PDF

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Publication number
ZA200508948B
ZA200508948B ZA200508948A ZA200508948A ZA200508948B ZA 200508948 B ZA200508948 B ZA 200508948B ZA 200508948 A ZA200508948 A ZA 200508948A ZA 200508948 A ZA200508948 A ZA 200508948A ZA 200508948 B ZA200508948 B ZA 200508948B
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ZA
South Africa
Prior art keywords
pyrazol
fluorophenyl
biphenyl
methyl
het
Prior art date
Application number
ZA200508948A
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English (en)
Inventor
Schiemann Kai
Arlt Michael
Schadt Oliver
Bartoszyk Gerd
Ackermann Karl-August
Finsinger Dirk
Van Amsterdam Christoph
Seyfried Christoph
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Merck Patent Gmbh
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Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of ZA200508948B publication Critical patent/ZA200508948B/en

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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ZA200508948A 2003-04-05 2005-11-04 Substituted pyrazoles ZA200508948B (en)

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DE10315572A DE10315572A1 (de) 2003-04-05 2003-04-05 Substituierte Pyrazole

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ZA200508948B true ZA200508948B (en) 2007-03-28

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JP4740115B2 (ja) 2011-08-03
CA2521201A1 (en) 2004-10-21
AU2004228120A1 (en) 2004-10-21
CN1768051A (zh) 2006-05-03
JP2006522035A (ja) 2006-09-28
AU2004228120B2 (en) 2010-12-02
AR043837A1 (es) 2005-08-17
WO2004089931A1 (de) 2004-10-21
JP2011148803A (ja) 2011-08-04
MXPA05010652A (es) 2005-12-12
PL377844A1 (pl) 2006-02-20
KR20050119193A (ko) 2005-12-20
DE10315572A1 (de) 2004-10-14
US20060264419A1 (en) 2006-11-23
BRPI0409164A (pt) 2006-04-11

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