KR20050119193A - 치환된 피라졸 - Google Patents

치환된 피라졸 Download PDF

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Publication number
KR20050119193A
KR20050119193A KR1020057018895A KR20057018895A KR20050119193A KR 20050119193 A KR20050119193 A KR 20050119193A KR 1020057018895 A KR1020057018895 A KR 1020057018895A KR 20057018895 A KR20057018895 A KR 20057018895A KR 20050119193 A KR20050119193 A KR 20050119193A
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South Korea
Prior art keywords
pyrazol
fluorophenyl
ylmethyl
biphenyl
methyl
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KR1020057018895A
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English (en)
Korean (ko)
Inventor
카이 쉬만
칼-아우구스트 아케르만
미카엘 아를트
디르크 핀싱어
올리버 샤트
크리스토프 반 암스테르담
게르트 바르토스지크
크리스토프 자이프리트
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메르크 파텐트 게엠베하
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Publication of KR20050119193A publication Critical patent/KR20050119193A/ko
Withdrawn legal-status Critical Current

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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KR1020057018895A 2003-04-05 2004-03-08 치환된 피라졸 Withdrawn KR20050119193A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10315572A DE10315572A1 (de) 2003-04-05 2003-04-05 Substituierte Pyrazole
DE10315572.4 2003-04-05

Publications (1)

Publication Number Publication Date
KR20050119193A true KR20050119193A (ko) 2005-12-20

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EP1626967A1 (de) 2006-02-22
AU2004228120A1 (en) 2004-10-21
AR043837A1 (es) 2005-08-17
JP2011148803A (ja) 2011-08-04
WO2004089931A1 (de) 2004-10-21
ZA200508948B (en) 2007-03-28
JP4740115B2 (ja) 2011-08-03
BRPI0409164A (pt) 2006-04-11
PL377844A1 (pl) 2006-02-20
CA2521201A1 (en) 2004-10-21
MXPA05010652A (es) 2005-12-12
CN1768051A (zh) 2006-05-03
AU2004228120B2 (en) 2010-12-02
US20060264419A1 (en) 2006-11-23
DE10315572A1 (de) 2004-10-14
JP2006522035A (ja) 2006-09-28

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